sistema nervoso perifÉrico parte iv
TRANSCRIPT
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5 – HT E FARMACOLOGIA DA
ENXAQUECAProfessora Me. Carina Godoy Picelli
FARMACOLOGIA
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ENXAQUECA
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5 -HIDROXITRIPTAMINA
ENTEROAMINA, EXTRATOS DE INTESTINOSEROTONINA, SORO
SISTEMA NERVOSO CENTRALHORMÔNIO LOCAL
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5 - HIDROXITRIPTAMINA
TECIDOS:
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INGESTÃO DE SEROTONINA?!
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SNE: motilidade, peristaltismo, secreções, sensibilidade
CONTRAÇÃO
ARTÉRIAS: VASOCONSTRIÇÃO
AGREGAÇÃO PLAQUETÁRIA
DOR
HUMOR
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5 - HIDROXITRIPTAMINA
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ALCALÓIDES DE ERGOT
ERGOTAMINA: PROFILAXIA DA ENXAQUECAERGOMETRINA:PREVENÇÃO DE HEMORRAGIA PÓS PARTOMETISERGIDA: PROFILAXIA DA ENXAQUECABROMOCRIPTINA: PARKINSON, DISTÚRBIOS ENDÓCRINOS
MECANISMO DE AÇÃO: RECEPTORES 5 –HT, DOPAMINA E ADRENÉRGICOS(AGONISTAS, ANTAGONISTAS, AGONISTAS PARCIAIS)
EFEITOS ADVERSOS: NÁUSEAS, VÔMITO, VASOCONSTRIÇÃO
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ENXAQUECA
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CAUSAS
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FISIOPATOLOGIA
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TRATAMENTO ENXAQUECA
CRISE AGUDAANALGÉSICOS COMUNS (ASPIRINA, PARACETAMOL)ERGOTAMINA (AGONISTA PARCIAL RECEPTOR 5 – HT1)SUMATRIPTANO, ZOLMITRIPTANO (AGONISTAS 5 – HT1)
PROFILAXIA ANTAGONISTAS BETA-ADRENÉRGICOS (PROPANOLOL, METOPROLOL)PIZOTIFENO, CIPROEPTADINA, METISERGIDA (ANTAGONISTA RECEPTOR 5 – HT2)ANTIDEPRESSIVOS TRICÍCLICOS (AMITRIPTILINA, NORTRIPTILINA)ANTAGONISTAS DE CÁLCIO (VERAPAMIL)
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ERGOT
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