supplemental figure 1 · supplemental table 1 kd (nm) birinapant avpi (smac) ciap1 bir3
TRANSCRIPT
Supplemental Figure 1
Supplemental Figure 2
A B
Supplemental Figure 3A
B
Supplemental Figure 4
F (p
g/m
L)
300
400
500SK-OV-3EVSA-TA375HeLa
Secr
eted
TN
F
100
200
300 HeLa
1 μM Birinapant No Treatment0
Supplemental Figure 5
Supplemental Figure 6
A
B
Supplemental Figure 7
Supplemental Table 1
Kd (nM)Birinapant AVPI (Smac)
cIAP1 BIR3 <1 2cIAP2 BIR3 36 20XIAP BIR3 45 130ML-IAP BIR <1 900
Kd, dissociation constant; cIAP, cellular inhibitor of apoptosis; XIAP, X-linked inhibitor of apoptosis; ML-IAP, melanoma inhibitor of apoptosis.