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Page 1: Tech Help: Email: tech@biovision.com | Toll Free: 800.891 ...biolinkk.com/.../uploads/2018/09/Enzyme-Inhibitors-Mini-Brochure.pdf · 2 Ordering: Email: orders@biovision.com Tel:408.493.1800

Tech Help: Email: [email protected] | Toll Free: 800.891.9699 (US Only) |

Page 2: Tech Help: Email: tech@biovision.com | Toll Free: 800.891 ...biolinkk.com/.../uploads/2018/09/Enzyme-Inhibitors-Mini-Brochure.pdf · 2 Ordering: Email: orders@biovision.com Tel:408.493.1800

2Ordering: Email: [email protected] | Tel:408.493.1800 | Web: www.biovision.com 2

ACE (Angiotensin-Converting Enzyme) Inhibitors

Product Name Cat. No. Size CAS. No.Arecoline hydrobromide B1824 100 mg, 500 mg 300-08-3Avasimibe 9506 5 mg, 25 mg 166518-60-1Naringenin 1772 250 mg, 1 g 480-41-1Pellitorine 2053 1 mg, 5 mg 18836-52-7Penicillide B1245 250 µg, 1 mg 55303-92-9Pyripyropene A B1910 500 µg, 1 mg 147444-03-9Terpendole C 2214 250 µg, 1 mg 156967-65-6TMP-153 B1181 10 mg, 50 mg 128831-46-9

ACAT (Acyl-CoA cholesteryl Acyl Transferase) Inhibitors

Product Name Cat. No. Size CAS. No.ACC2 Inhibitor 1717 1 mg, 5 mg N/ACP-640186 9422 5 mg, 25 mg 591778-68-6CP-640186 hydrochloride B1254 5 mg, 25 mg 591778-70-0

ACC (Acetyl-CoA Carboxylase) Inhibitors

Product Name Cat. No. Size CAS. No.2',5'-Dideoxyadenosine 2770 5 mg, 25 mg 6698-26-6KH7 2350 5 mg, 25 mg 330676-02-3PACAP (human, chicken, mouse, ovine, porcine, rat) (6-38) B1562 100 μg, 500 μg 143748-18-9

SQ 22536 2019 5 mg, 25 mg 17318-31-9

Adenylase Cyclase Inhibitors

Product Name Cat. No. Size CAS. No.AKR1C3 Inhibitor I 2403 5 mg, 25 mg N/AAKR1C3 Inhibitor II 2404 5 mg, 25 mg N/AAKR1C3 Inhibitor III 2424 5 mg, 25 mg N/A

AKR (Aldo-Keto Reductase) Inhibitors

Product Name Cat. No. Size CAS. No.ARN-509 9535 5 mg, 25 mg 956104-40-8MDV-3100 9479 10 mg, 50 mg 915087-33-1ODM-201 9668 5 mg, 25 mg 1297538-32-9

Androgen Receptor Antagonists

Angiogenesis Inhibitors

Product Name Cat. No. Size CAS. No.BIBS39 B1071 5 mg, 25 mg 133085-33-3 EXP-3174 9672 5 mg, 25 mg 124750-92-1Losartan potassium 2750 50 mg, 250 mg 124750-99-8Valsartan 2004 25 mg, 100 mg, 500 mg 137862-53-4

Angiotensin Receptor Antagonists

Product Name Cat. No. Size CAS. No.ACE2 Inhibitor, DX600 9687 100 µg, 500 µg, 1 mg N/ACaptopril B1187 1 g, 5 g 62571-86-2

Product Name Cat. No. Size CAS. No.BEC 2359 1 mg, 5 mg 63107-40-4

Arginase Inhibitors

Product Name Cat. No. Size CAS. No.Exemestane 9473 5 mg, 25 mg 107868-30-4

Aromatase Inhibitors

Product Name Cat. No. Size CAS. No.Bafilomycin A1 1829 50 µg, 250 µg 88899-55-2(-)-Blebbistatin 2406 1 mg, 5 mg 856925-71-8(+)-Blebbistatin 2407 1 mg, 5 mg 1177356-70-5(±)-Blebbistatin 2405 5 mg, 25 mg 674289-55-5Bufalin 2509 10 mg, 50 mg 465-21-4

ATPase Inhibitors

Product Name Cat. No. Size CAS. No.ATM Kinase Inhibitor, KU-55933 1685 5 mg 587871-26-9Bafilomycin A1 1829 50 µg, 250 µg 88899-55-2Chloroquine Diphosphate 1825 100 mg, 500 mg 50-63-5EZSolution™ Gö 6976 1785 500 µg 136194-77-9Gö 6976 1711 500 µg 136194-77-93-Methyladenine 2249 25 mg, 100 mg 5142-23-4Spautin-1 2037 5 mg, 25 mg 1262888-28-7

Autophagy Inhibitors

Product Name Cat. No. Size CAS. No.A-1155463 B1821 5 mg, 25 mg 1235034-55-5 A-1210477 B1826 5 mg, 25 mg 1668553-26-1A-1331852 B1948 5 mg, 25 mg 1430844-80-6

Bcl-2 (B-cell lymphoma 2) Inhibitors

Enzyme InhibitorsEnzymes are biological catalysts that drive various reactions within a cell. They are required for nearly every function of a living cell/organism from digestion of food to the synthesis of DNA. Enzymes are usually very specific as to which reactions they catalyze and the substrates that are involved. Enzyme activity can be modulated by different classes of molecules. Enzyme Inhibitors are molecules that bind to the enzyme and decrease or completely stop their function. Since blocking the activity of an enzyme can have profound effects on the downstream cellular events sometimes with pathological or disease consequences, enzyme inhibition is a crucial component of new drug design. The discovery of new and potent enzyme inhibitors and developing better classes of inhibitors constitutes a dynamic branch of biochemical and pharmacological research in the area of Diabetes, Cancer, HIV and many more. BioVision offers a comprehensive collection of more than 800 enzyme inhibitors covering all the core biological/pharmacological research areas.

Product Name Cat. No. Size CAS. No.Angiostatin Human 4919 100 μg, 500 μg N/AAngiostatin K1-3, human recombinant 4920 20 μg, 100 μg, 1 mg N/ABIBF1120 2167 5 mg, 25 mg 928326-83-4Borrelidin 2367 250 µg, 1 mg 7184-60-3Castanospermine 2293 10 mg, 50 mg 79831-76-8

Product Name Cat. No. Size CAS. No.Endostatin, human recombinant 4759 20 μg, 100 μg, 1 mg N/AEndostatin, human recombinant 4799 100 μg, 1 mg N/AFumagillin 2368 1 mg, 5 mg 23110-15-8Isoxanthohumol 2529 5 mg, 25 mg 70872-29-62-Methoxyestradiol 2166 5 mg, 25 mg 362-07-2SKLB610 2610 5 mg, 25 mg 1125780-41-7Thiabendazole 2161 1 g 148-79-8Tranilast 1876 10 mg, 50 mg 53902-12-8

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Product Name Cat. No. Size CAS. No.DMH-1 9542 5 mg, 25 mg 1206711-16-1EZSolution™ LDN193189 2092 5 mg 1062368-24-4LDN193189 1995 5 mg, 25 mg 1062368-24-4

BMP (Bone Morphogenetic Protein) Inhibitors

Product Name Cat. No. Size CAS. No.Alendronate sodium 2168 50 mg, 250 mg 121268-17-5Pamidronate disodium 1884 50 mg, 250 mg 57248-88-1Zoledronic acid hydrate 2653 10 mg, 50 mg 165800-06-6

Bone Resorption Inhibitors

Bromodomain InhibitorsProduct Name Cat. No. Size CAS. No.BAZ2-ICR B1865 5 mg, 25 mg 1665195-94-7 BI-7273 B1879 5 mg, 25 mg 1883429-21-7BI-9564 B1880 5 mg, 25 mg 1883429-22-8Bromodomain Inhibitor, (+)-JQ1 2070 1 mg, 5 mg 1268524-70-4Bromosporine 2652 1 mg, 5 mg 1619994-69-2CPI-0610 B1201 5 mg, 25 mg 1380087-89-7 CPI-203 9404 1 mg, 5 mg 1446144-04-2GSK-2801 9553 5 mg, 25 mg 1619994-68-1I-BET151 2220 1 mg, 5 mg 1300031-49-5I-BET726 B1569 5 mg, 25 mg 1300031-52-0I-BET762 2628 1 mg, 5 mg 1260907-17-2I-CBP112 9405 1 mg, 5 mg N/AEZSolution™ (+)-JQ1 2091 1 mg 1268524-70-4(-)-JQ1 2384 1 mg 1268524-71-5Mivebresib B1564 5 mg, 25 mg 1445993-26-9 MS436 2680 5 mg, 25 mg 1395084-25-9OF-1 9592 5 mg, 25 mg 919973-83-4OTX015 2651 1 mg, 5 mg 202590-98-5PFI-1 2203 1 mg, 5 mg 1403764-72-6PFI-3 2895 5 mg, 25 mg 1819363-80-8RVX-208 9408 1 mg, 5 mg 1044870-39-4SGC-CBP30 9554 5 mg, 25 mg 1613695-14-9

Product Name Cat. No. Size CAS. No.EZSolutioin™ Calpain Inhibitor I, ALLN 2544 5 mg 110044-82-1Calpain Inhibitor I, ALLN 1834 5 mg, 25 mg 110044-82-1Calpain Inhibitor II, ALLM 1835 5 mg, 25 mg 136632-32-1Calpain Inhibitor Z-LLY-FMK 1125 20 µl (10 mM) 133410-84-1Calpain Inhibitor, Z-LLY-FMK B1506 250 μg, 1 mg 133410-84-1

Calpain Inhibitors

Caspase & Granzyme B InhibitorsProduct Name Cat. No. Size CAS. No.Ac-DEVD-CHO B1951 1 mg, 5 mg 169332-60-9Apoptosis inhibitor 2783 5 mg, 25 mg 54135-60-3AZ10417808 2786 1 mg, 5 mg 331645-84-2Biotin-DEVD-FMK 1124 20 µl (10 mM) N/ABiotin-IETD-FMK 1121 20 µl (10 mM) N/ABiotin-VAD-FMK 1123 20 µl (10 mM) 1135688-15-1Biotin-VDVAD-FMK 1032 20 µl (10 mM) N/ABoc-D-FMK 1160 1 mg, 5 mg 187389-53-3Caspase Family Inhibitor Set K107 5 x 25 µl N/ACaspase Family Inhibitor Set II K108 7 x 25 µl N/ACaspase Family Inhibitor Set III K210 8 x 25 µl N/ACaspase Family Inhibitor Set IV K220 12 x 25 µl N/ACaspase Inhibitor Boc-D-FMK 1120 20 µl (10 mM) 187389-53-3Caspase-1 Inhibitor Z-YVAD-FMK 1012 20 µl (10 mM), 100 µl (2 mM) N/ACaspase-10 Inhibitor AEVD-FMK 1112 20 µl (10 mM), 100 µl (2 mM) 1135688-47-9Caspase-12 Inhibitor Z-ATAD-FMK 1079 20 µl (10 mM), 100 µl (2 mM) N/ACaspase-13 Inhibitor LEED-FMK 1115 20 µl (10 mM), 100 µl (2 mM) N/ACaspase-2 Inhibitor Z-VDVAD-FMK 1073 20 µl (10 mM), 100 µl (2 mM) N/ACaspase-3 Inhibitor Q-DEVD-Oph 1175 1 mg, 3 mg, 5 mg N/ACaspase-3 Inhibitor Z-DEVD-FMK 1009 20 µl (10 mM), 100 µl (2 mM) 210344-95-9Caspase-3 inhibitor, Z-DQMD-FMK 2782 1 mg, 5 mg N/ACaspase-3/7 Inhibitor 2780 1 mg, 5 mg 220509-74-0Caspase-4 Inhibitor Z-LEVD-FMK 1108 20 µl (10 mM), 100 µl (2 mM) N/ACaspase-5 Inhibitor Z-WEHD-FMK 1100 20 µl (10 mM), 100 µl (2 mM) N/ACaspase-6 Inhibitor Z-VEID-FMK 1011 20 µl (10 mM), 100 µl (2 mM) N/ACaspase-8 Inhibitor Z-IETD-FMK 1064 20 µl (10 mM), 100 µl (2 mM) N/ACaspase-8 Inhibitor, Q-IETD-Oph 1176 1 mg, 3 mg, 5 mg N/ACaspase-9 Inhibitor Z-LEHD-FMK 1074 20 µl (10 mM), 100 µl (2 mM) N/ACaspase-9 Inhibitor, Q-LEHD-Oph 1177 1 mg, 3 mg, 5 mg N/ACaspase-Family Inhibitor Z-VAD-FMK 1010 20 µl (10 mM), 100 µl (2 mM) 187389-52-2EMAP-II Inhibitor Z-ASTD-FMK 1127 20 µl (10 mM) N/AFITC-DEVD-FMK 9499 100 Assays N/AFITC-IETD-FMK 9533 100 Assays N/AFITC-LEHD-FMK 9534 100 Assays N/AFITC-VAD-FMK 9497 100 Assays N/AFITC-VDVAD-FMK 9498 100 Assays N/AFMK Negative Control 1122 20 µl (10 mM), 100 µl (2 mM) 197855-65-5Granzyme B Inhibitor Ac-IEPD-CHO 1119 1 mg N/AGranzyme B Inhibitor Z-AAD-CH2Cl 1128 20 µl (10 mM) N/AIvachtin 2788 1 mg, 5 mg 745046-84-8Pan-caspase inhibitor, Q-VD(OMe)-Oph 2787 1 mg, 5 mg N/AEZSolution™ Q-DEVD-Oph 1178 1 mg N/AEZSolution™ Q-VD-Oph 1173 1 mg 1135695-98-5Q-VD-OPh 1170 1 mg, 3 mg, 5 mg 1135695-98-5EZSolution™ Q-VD-OPh, Negative Control 1174 1 mg N/AQVD-OPh Negative Control 1171 1 mg, 3 mg, 5 mg N/AVX-765 2781 5 mg, 25 mg 273404-37-8Z-AEVD-FMK B1162 1 mg, 5 mg 1135688-47-9Z-ATAD-FMK 1152 1 mg, 5 mg N/AZ-DEVD-FMK 1143 1 mg, 5 mg 210344-95-9Z-FA-FMK 1986 1 mg, 5 mg 105637-38-5Z-IETD-FMK 1148 1 mg, 5 mg N/AZ-LEHD-FMK 1149 1 mg, 5 mg N/A

Product Name Cat. No. Size CAS. No.

DiscoveryPak™ Calpain Inhibitors Set(Containing Cat. No. 1834, 1835, 1506, 2195, 1906)

S228 1 Set

110044-82-1 136632-32-1 133410-84-1 88191-84-8 179528-45-1

MDL 28170 2195 10 mg, 50 mg 88191-84-8PD 150,606 1906 5 mg, 25 mg 179528-45-1

Product Name Cat. No. Size CAS. No.ABT-263 2467 5 mg, 25 mg 923564-51-6ABT-737 2463 5 mg, 25 mg 852808-04-9AT-101 2380 5 mg, 25 mg 90141-22-3BCl-2 Inhibitor GX15-070 2040 5 mg 803712-67-6BCl-2 Inhibitor, ABT-199 2253 1 mg, 5 mg 1257044-40-8

DiscoveryPak™ Bcl2 Inhibitors Set(Containing Cat. No. 2253, 2467, 2463, 2380, 2040)

S229 1 Set

1257044-40-8923564-51-6852808-04-990141-22-3803712-67-6

BDA366 B1827 5 mg, 25 mg 1909226-00-1BH3I-1 B1277 5 mg, 25 mg 300817-68-9CC-122 B1650 5 mg, 25 mg 1015474-32-4CID-5721353 B1275 5 mg, 25 mg 301356-95-6 HA14-1 B1832 5 mg, 25 mg 65673-63-4Pyridoclax B1817 1 mg, 5 mg 1651890-44-6 S63845 B1819 250 μg, 1 mg 1799633-27-4 TW-37 2789 5 mg, 25 mg 877877-35-5WEHI-539 B1818 5 mg, 25 mg 1431866-33-9

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Product Name Cat. No. Size CAS. No.Z-LEVD-FMK 1144 1 mg, 5 mg N/AZ-VAD-FMK 1140 1 mg, 5 mg 187389-52-2Z-VDVAD-FMK 1142 1 mg, 5 mg N/AZ-VEID-FMK 1146 1 mg, 5 mg N/AZ-YVAD-FMK 1141 1 mg, 5 mg N/A

Product Name Cat. No. Size CAS. No.Balicatib 2596 5 mg, 25 mg 354813-19-7Cathepsin B&L Inhibitor Z-Phe-Phe-FMK 1126 20 µl (10 mM) N/ACathepsin G Inhibitor 1982 1 mg 429676-93-7Odanacatib B1617 5 mg, 25 mg 603139-19-1Tanshinone IIA-Sulfonic Sodium B1902 5 mg, 25 mg 69659-80-9Z-FA-FMK 1986 1 mg, 5 mg 105637-38-5

Cathepsin Inhibitors

Product Name Cat. No. Size CAS. No.ML141 2267 5 mg, 25 mg 71203-35-5MLS-573151 1929 5 mg, 25 mg 10179-57-4ZCL278 2466 5 mg, 25 mg 587841-73-4

CDc42 Inhibitors

Product Name Cat. No. Size CAS. No.K-7174 dihydrochloride 9478 5 mg, 25 mg 191089-60-8

Cell Adhesion Inhibitors

Product Name Cat. No. Size CAS. No.EZSolution™ Anacetrapib 2531 1 mg 875446-37-0Anacetrapib 2418 1 mg, 5 mg 875446-37-0

DiscoveryPak™ CETP Inhibitors Set(Containing Cat. No. 2418, 2419, 2558, 2420)

S225 1 Set

875446-37-0 211513-37-0 1186486-62-3 262352-17-0

EZSolution ™ Dalcetrapib 2532 1 mg 211513-37-0Dalcetrapib 2419 1 mg, 5 mg 211513-37-0Evacetrapib 2558 5 mg, 25 mg 1186486-62-3Sclerotiorin 2334 250 µg, 1 mg 549-23-5EZSolution™ Torcetrapib 2533 5 mg 262352-17-0Torcetrapib 2420 5 mg, 25 mg 262352-17-0

CETP (Cholesteryl Ester Transfer Protein) Inhibitors

Product Name Cat. No. Size CAS. No.CaCCinh-A01 B2014 5 mg, 25 mg 407587-33-1CFTR Inhibitor-172 2487 1 mg, 5 mg 307510-92-5CLP-290 B1282 5 mg, 25 mg 1181083-81-7

Chloride Channel Blockers

Product Name Cat. No. Size CAS. No.Ezetimibe 9468 25 mg, 100 mg 163222-33-1U-18666A 9469 5 mg, 25 mg 3039-71-2

Cholesterol Transport Inhibitors

Product Name Cat. No. Size CAS. No.Celecoxib 1574 100 mg, 1 g 169590-42-5Cimicoxib B1984 5 mg, 25 mg 265114-23-6Deracoxib B1985 10 mg, 50 mg 169590-41-4DuP-697 B1517 5 mg, 25 mg 88149-94-4Etoricoxib B1983 10 mg, 50 mg 202409-33-4Firocoxib B1986 5 mg, 25 mg 189954-96-96-Gingerol 2507 5 mg, 25 mg 23513-14-6Loganin B1161 10 mg, 50 mg 18524-94-2Lumiracoxib B1987 5 mg, 25 mg 220991-20-8Mavacoxib B1988 5 mg, 25 mg 170569-88-7

COX (Cyclooxygenase) Inhibitors

Product Name Cat. No. Size CAS. No.Alogliptin benzoate 9656 50 mg, 250 mg 850649-62-6Diprotin A 2191 5 mg, 25 mg 90614-48-5Diprotin B 2192 5 mg, 25 mg 90614-49-6DPP IV Inhibitor, K 579 1963 1 mg, 5 mg 440100-64-1DPP IV Inhibitor, NVP DPP 728 1964 1 mg, 5 mg 247016-69-9DPPIV Inhibitor, P32/98 2571 5 mg, 25 mg 136259-20-6

DiscoveryPak™ DPP-IV Inhibitors Set(Containing Cat. No. 2240, 9528, 1757, 2798, 2188)

K890 5 Inhibitors

668270-12-0 361442-04-8 654671-77-9 1029877-94-8 274901-16-5

Linagliptin 2240 50 mg, 250 mg 668270-12-0MK-3102 9599 1 mg, 5 mg 1226781-44-7Saxagliptin 9528 50 mg, 250 mg 361442-04-8Sitagliptin Phosphate Monohydrate 1757 100 mg, 1 g 654671-77-9Teneligliptin B1932 10 mg, 50 mg 760937-92-6Trelagliptin succinate 2798 5 mg, 25 mg 1029877-94-8Vildagliptin 2188 10 mg, 50 mg 274901-16-5

DPP-4 (Dipeptidyl Peptidase-4 ) Inhibitors

Product Name Cat. No. Size CAS. No.L-189 9674 5 mg, 25 mg 64232-83-3L-67 9633 5 mg, 25 mg 325970-71-6

DNA Ligase Inhibitors

Product Name Cat. No. Size CAS. No.DUB Inhibitor, NSC-632839 2570 5 mg, 25 mg 157654-67-6DUB Inhibitor, PR-619 2302 5 mg, 25 mg 2645-32-1HBX-41108 9608 5 mg, 25 mg 924296-39-9LDN-57444 2016 5 mg, 25 mg 668467-91-2ML-323 2658 5 mg, 25 mg 1572414-83-5NSC-687852 2021 5 mg, 25 mg 1009817-63-3Spautin-1 2037 5 mg, 25 mg 1262888-28-7USP14 Inhibitor, IU1 1845 5 mg, 25 mg 314245-33-5USP7/USP47 Inhibitor, P 22077 2301 5 mg, 25 mg 1247819-59-5WP-1130 2014 5 mg, 25 mg 856243-80-6

DUBs (Deubiquitinating Enzymes) & Related Inhibitors

Product Name Cat. No. Size CAS. No.FAAH Inhibitor, PF-622 1928 5 mg, 25 mg 898235-65-9JNJ-1661010 2413 5 mg, 25 mg 681136-29-8JZL195 B1064 5 mg, 25 mg 1210004-12-8EZSolution™ MAFP 2811 5 mg 188404-10-6

FAAH (Fatty Acid Amide Hydrolase) Inhibitors

Product Name Cat. No. Size CAS. No.Cerulenin 1579 5 mg, 50 mg 17397-89-6DPVP B1243 1 mg 223386-36-5FAS Inhibitor, C75 1547 1 mg 191282-48-1GSK-2194069 B1571 5 mg, 25 mg 1332331-21-1α-Mangostin B1059 10 mg, 50 mg 6147-11-1

FAS (Fatty Acid Synthase) Inhibitors

Product Name Cat. No. Size CAS. No.Ferrostatin-1 2230 5 mg, 25 mg 347174-05-4

Ferroptosis Inhibitors

Product Name Cat. No. Size CAS. No.Nimesulide 2777 1 g, 5 g 51803-78-2Parecoxib Sodium B1989 10 mg, 50 mg 198470-85-8Robenacoxib B1990 5 mg, 25 mg 220991-32-2Rofecoxib B1982 10 mg, 50 mg 162011-90-7Valdecoxib B1991 5 mg, 25 mg 181695-72-7

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Product Name Cat. No. Size CAS. No.Andrastin A, Aspergillus fumigatus 2149 250 µg, 1 mg 174232-42-9Arglabin 9691 1 mg, 5 mg 84692-91-1FTI-277 hydrochloride 2874 5 mg, 25 mg 180977-34-8L-778123 hydrochloride 9638 10 mg, 50 mg 253863-00-2Lonafarnib B1616 5 mg, 25 mg 193275-84-2 Manumycin A 2333 1 mg, 5 mg 52665-74-4Tipifarnib, Free base 2296 1 mg, 5 mg 192185-72-1

FPT (Farnesyl Protein Transferase) Inhibitors

Product Name Cat. No. Size CAS. No.Castanospermine 2293 10 mg, 50 mg 79831-76-8Conduritol B Epoxide 9574 5 mg, 25 mg 6090-95-5Miglitol 2335 5 mg, 25 mg 72432-03-2

Glucosidase Inhibitors

Product Name Cat. No. Size CAS. No.BAY-876 B1572 5 mg, 25 mg 1799753-84-6Fasentin B1576 5 mg, 25 mg 392721-37-8Naringenin 1772 250 mg, 1 g 480-41-1Resveratrol 1758 100 mg, 500 mg 501-36-0Rubusoside B1574 5 mg, 25 mg 64849-39-4STF-31 9585 5 mg, 25 mg 724741-75-7WZB117 B1573 5 mg, 25 mg 1223397-11-2

GLUT1 (Glucose Transporter) Inhibitors

Product Name Cat. No. Size CAS. No.LY-341495 2875 1 mg, 5 mg 201943-63-7

Glutamate Receptor Antagonists

Product Name Cat. No. Size CAS. No.Evans Blue Tetrasodium 2586 1 g 314-13-6Rose bengal 2587 100 mg, 500 mg 632-69-9

Glutamate Uptake Inhibitors

Product Name Cat. No. Size CAS. No.6-Aminonicotinamide B1047 100 mg, 500 mg 329-89-53-Bromopyruvic acid B1045 100 mg, 500 mg 1113-59-32-Deoxy-D-Glucose B1048 100 mg, 500 mg 154-17-6Lonidamine B1058 10 mg, 50 mg 50264-69-2Oxythiamine Chloride Hydrochloride B1046 100 mg, 500 mg, 1 g 614-05-1Shikonin B1056 10 mg, 50 mg 517-89-5

Glycolysis Inhibitors

Product Name Cat. No. Size CAS. No.Ezatiostat 2608 5 mg, 25 mg 168682-53-9GST Inhibitor-1 (Cibacron Blue 3G-A, Sodium Salt) 1555R 1 g 84166-13-2

GST Inhibitor-2 (Ethacrynic acid)) 1556 1 g 58-54-8

GST (Glutathione S-Transferase) Inhibitors

Product Name Cat. No. Size CAS. No.BQU57 9576 5 mg, 25 mg 1637739-82-2CID-1067700 2688 5 mg, 25 mg 314042-01-8RBC8 B1136 5 mg, 25 mg 361185-42-4

GTPase Inhibitors

Product Name Cat. No. Size CAS. No.LY-83583 B1314 5 mg, 25 mg 91300-60-6

Guanylate Cyclase Inhibitors

HDAC (Histone Deacetylase) InhibitorsProduct Name Cat. No. Size CAS. No.ACY-1215 2629 5 mg, 25 mg 1316214-52-4ACY-775 B2011 5 mg, 25 mg 1375466-18-4 Apicidin 1601 1 mg 183506-66-3AR-42 (HDAC-42) 2716 1 mg, 5 mg 935881-37-1BG-45 B1866 5 mg, 25 mg 926259-99-6 BML210 B1128 5 mg, 25 mg 537034-17-6BRD-73954 9596 5 mg, 25 mg 1440209-96-0CAY10683 B1051 5 mg, 25 mg 1477949-42-0CBHA 2284 5 mg, 10 mg 174664-65-4Chidamide 2261 1 mg, 5 mg 743420-02-2CI-994 1742 10 mg, 50 mg 112522-64-2Citarinostat B1560 5 mg, 25 mg 1316215-12-9 CUDC-101 1966 5 mg, 25 mg 1012054-59-9Depudecin 2087 100 µg 139508-73-9Droxinostat 9570 5 mg, 25 mg 99873-43-5Elevenostat B1893 1 mg N/AFK228 2447 1 mg 128517-07-7HC Toxin 2728 500 µg, 1 mg 83209-65-8

DiscoveryPak™ HDAC Inhibitor Set(Containing Cat. No. 1601, 1606, 1607, 1608, 1647)

K851 6 Inhibitors

183506-66-3 58880-19-6 251456-60-7 1716-12-7 1069-66-5

DiscoveryPak™ HDAC Inhibitor Set II(Containing Cat. No. 1742, 1612, 1604, 2202, 1605, 1606, 1984)

K876 7 Inhibitors

112522-64-2 404950-80-7 149647-78-9 38937-66-5 287383-59-9 58880-19-6 537049-40-4

ITF2357 9431 1 mg, 5 mg 732302-99-7ITSA-1 2089 5 mg, 25 mg 200626-61-5JNJ-26481585 9612 5 mg, 25 mg 875320-29-9LAQ824 2634 1 mg, 5 mg 404951-53-7LMK-235 B1642 5 mg, 25 mg 1418033-25-6M344 1607 1 mg 251456-60-7MC-1568 B1085 5 mg, 25 mg 852475-26-4MGCD0103 2633 10 mg, 50 mg 726169-73-9MS-275 (Entinostat, SNDX-275) 1590 1 mg, 5 mg 209783-80-2NCH 51 B1130 5 mg, 25 mg 848354-66-5Nexturastat A 2098 1 mg 1403783-31-2NKL 22 (MDK-4154) B1133 10 mg, 50 mg 537034-15-4Nullscript 2186 1 mg, 5 mg 300816-11-9Oxamflatin 2250 1 mg, 5 mg 151720-43-3Panobinostat (LBH589) 1612 1 mg, 5 mg, 25 mg 404950-80-7PCI 34051 2251 5 mg, 25 mg 950762-95-5PXD101 2480 5 mg, 25 mg 414864-00-9Pyroxamide 2189 5 mg, 25 mg 382180-17-8RGFP966 2818 5 mg, 25 mg 1396841-57-8SAHA 1604 1 mg, 5 mg 149647-78-9SB 939 2285 1 mg, 5 mg 929016-96-6SBHA 2202 50 mg, 250 mg 38937-66-54SC-202 B1230 5 mg, 25 mg 1186222-89-8Scriptaid 1605 1 mg 287383-59-9Sodium butyrate 1609 1 g 156-54-7Sodium 4-phenylbutyrate 1608 100 mg, 1 g 1716-12-7Splitomicin 1610 5 mg 5690-03-9TC-H 106 B1148 10 mg, 50 mg 937039-45-7

Product Name Cat. No. Size CAS. No.Anacardic Acid 1849 5 mg, 25 mg 16611-84-0C646, p300/CBP Inhibitor 1948 1 mg, 5 mg 328968-36-1Curcumin, Curcuma longa (High Purity) 1850 10 mg, 50 mg 458-37-7EML-425 B1882 5 mg, 25 mg 1675821-32-5

HAT (Histone Acetyltransferase) Inhibitors

Product Name Cat. No. Size CAS. No.(-)-Epigallocatechin gallate 1841 50 mg 989-51-5Garcinol 2088 5 mg, 25 mg 78824-30-3Plumbagin 2290 50 mg, 250 mg 481-42-5Remodelin 9411 5 mg, 25 mg 949912-58-7

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Product Name Cat. No. Size CAS. No.BAY 87-2243 B1878 5 mg, 25 mg 1227158-85-1Chetomin 2180 1 mg 1403-36-7Emetine dihydrochloride 1970 50 mg, 250 mg 316-42-7KC7F2 9641 10 mg, 50 mg 927822-86-4PT-2385 B1920 5 mg, 25 mg 1672665-49-4PX 12 2217 5 mg, 25 mg 141400-58-0PX-478 hydrochloride B1033 5 mg, 25 mg 685898-44-6

HIF (Hypoxia-Inducible Factor) Inhibitors

Product Name Cat. No. Size CAS. No.BAY 85-3934 9597 5 mg, 25 mg 1154028-82-6DMOG 2216 5 mg, 25 mg 89464-63-1FG-4592 9681 5 mg, 25 mg 808118-40-3GSK1278863 B1107 1 mg, 5 mg 960539-70-2IOX2 9451 5 mg, 25 mg 931398-72-0JNJ-42041935 B1072 5 mg, 25 mg 1193383-09-3

HIF-PH (Hypoxia-Inducible Factor Prolyl Hydroxylase) Inhibitors

Product Name Cat. No. Size CAS. No.TMP-195 B1860 5 mg, 25 mg 1314891-22-9 TMP269 2679 5 mg, 25 mg 1314890-29-3EZSolution™ Trichostatin A 2271 1 mg 58880-19-6Trichostatin A 1606 1 mg 58880-19-6Tubacin 1984 250 µg, 1 mg 537049-40-4Tubastatin A 1724 1 mg, 5 mg 1239262-52-2UF 010 B1146 10 mg, 50 mg 537672-41-6Valproic Acid, Sodium Salt 1647 200 mg 1069-66-5

Product Name Cat. No. Size CAS. No.Elvitegravir 9465 5 mg, 25 mg 697761-98-1GSK1349572 2288 5 mg, 25 mg 1051375-16-6

HIV Integrase Inhibitors

Product Name Cat. No. Size CAS. No.Atorvastatin 2278 10 mg, 50 mg 134523-00-5(R,R)-Hymeglusin B1244 500 µg, 1 mg 29066-42-0Lovastatin 1692 50 mg, 250 mg 75330-75-5Mevastatin 1694 50 mg, 250 mg 73573-88-3EZSolution™ Rosuvastatin 2806 5 mg 287714-41-4Rosuvastatin 1955 5 mg, 25 mg 287714-41-4Simvastatin 1693 50 mg, 250 mg 79902-63-9

HMG-CoA (3-Hydroxy-3-Methylglutaryl Coenzyme A) Inhibitors

Product Name Cat. No. Size CAS. No.BMS-986205 B1839 5 mg, 25 mg 1923833-60-6IDO Pathway inhibitor 2746 50 mg, 250 mg 110117-83-4IDO1 Inhibitor I 2745 5 mg, 25 mg 914471-09-3INCB-024360 9477 5 mg, 25 mg 1204669-58-8Menadione 2747 500 mg, 1 g 58-27-5NLG919 9407 5 mg, 25 mg 1402836-58-1

IDO (Indoleamine 2,3-Dioxygenase) Inhibitors

Product Name Cat. No. Size CAS. No.JM6 1913 5 mg, 25 mg 1008119-83-2Ro 61-8048 1912 5 mg, 25 mg 199666-03-0

KMO (Kynurenine 3-Monoxygenase) Inhibitors

Product Name Cat. No. Size CAS. No.Galloflavin 2672 5 mg, 25 mg 568-80-9(±)-Gossypol 2579 50 mg, 250 mg 303-45-7Sodium Oxamate 2580 1 g, 5 g 565-73-1

LDH (Lactate Dehydrogenase) Inhibitors

Product Name Cat. No. Size CAS. No.Orlistat B1020 50 mg, 250 mg 96829-58-2XEN445 2681 5 mg, 25 mg 1515856-92-4

Lipase Inhibitors

Product Name Cat. No. Size CAS. No.NDGA 2581 100 mg, 500 mg 500-38-9

LO (Lipoxygenase) Inhibitors

Product Name Cat. No. Size CAS. No.EZSolution™ 17-AAG 9495 1 mg 75747-14-717-AAG 1774 1 mg, 5 mg 75747-14-717-DMAG hydrochloride 1776 1 mg, 5 mg 467214-21-7AT-13387 B1961 5 mg, 25 mg 912999-49-6BIIB 021 2291 5 mg, 25 mg 848695-25-0CUDC-305 9653 1 mg, 5 mg 1061318-81-7Ganetespib (STA-9090) 9459 5 mg, 25 mg 888216-25-9Geldanamycin 1564 1 mg, 5 mg 30562-34-6KRIBB11 B1567 5 mg, 25 mg 342639-96-7 Novobiocin Sodium Salt B1526 1 g, 5 g 1476-53-5NVP-AUY922 1591 1 mg, 5 mg 747412-49-3PU-H71 (Not Available for Sale in the U.S.) 9649 10 mg, 50 mg 873436-91-0PU-WS13 9442 5 mg, 25 mg 1454619-14-7Radicicol B1533 1 mg, 5 mg 12772-57-5Sulfamethoxazole B1534 5 g, 25 g 723-46-6XL888 2654 1 mg, 5 mg 1149705-71-4

Hsp (Heat Shock Protein) InhibitorsProduct Name Cat. No. Size CAS. No.BMS-833923 9547 5 mg, 25 mg 1059734-66-5BODIPY-Cyclopamine 2160 50 µg, 250 µg 334658-24-1CUR-61414 2743 5 mg, 25 mg 334998-36-6EZSolution™ Cyclopamine 2545 5 mg 4449-51-8Cyclopamine 1578 5 mg 4449-51-8Cyclopamine tartrate 2518 1 mg, 5 mg 1178510-81-0Cyclopamine-KAAD 1910 50 µg 306387-90-6GANT58 1812 5 mg, 25 mg 64048-12-0GANT61 1892 5 mg 500579-04-4EZSolution™ GDC-0449 2539 5 mg 879085-55-9GDC-0449 1890 5 mg, 25 mg 879085-55-9Hh Signaling Pathway Antagonist 1659 1 mg 330796-24-2HPI-1 2410 5 mg, 25 mg 599150-20-6Itraconazole 1987 50 mg, 100 mg, 500 mg, 1 g 84625-61-6Jervine 2357 1 mg, 5 mg 469-59-0JK 184 1726 1 mg 315703-52-7LDE-225 2892 5 mg, 25 mg 956697-53-3LDE-225 diphosphate 2893 5 mg, 25 mg 1218778-77-8LY-2940680 9604 5 mg, 25 mg 1258861-20-9MK-4101 B1255 5 mg, 25 mg 935273-79-3 Robotnikinin 1923 1 mg 1132653-79-2SANT-1 1978 1 mg, 5 mg 304909-07-7SANT-2 1976 1 mg, 5 mg 329196-48-7Smo Antagonist, SA1 2154 2 mg, 5 mg N/ASmo Antagonist, SA10 2159 2 mg, 5 mg N/ASmo Antagonist, SA9 2155 2 mg, 5 mg N/ATomatidine hydrochloride 1893 25 mg 6192-62-7

Hh (Hedgehog) Signaling Pathway Antagonists

Product Name Cat. No. Size CAS. No.Clorgyline hydrochloride 2622 10 mg, 50 mg 17780-75-5Harmine 2561 50 mg, 250 mg 442-51-3Moclobemide 9561 10 mg, 50 mg 71320-77-9Pargyline hydrochloride 2618 500 mg, 1 g 306-07-0Rasagiline mesylate 2237 50 mg, 250 mg 161735-79-1

MAO (Monoamine oxidase) Inhibitors

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Product Name Cat. No. Size CAS. No.Elacridar 2792 5 mg, 25 mg 143664-11-3HM-30181 B1285 5 mg, 25 mg 849675-66-7KS-176 B1272 5 mg, 25 mg 1253452-78-6MK-571 2691 5 mg, 25 mg 115104-28-4MK-571 sodium 2692 5 mg, 25 mg 115103-85-0NSC-23925 2686 5 mg, 25 mg 858474-14-3Tariquidar 2853 10 mg, 50 mg 206873-63-4Verapamil hydrochloride 2861 1 g, 5 g 152-11-4Zosuquidar trihydrochloride 9488 5 mg, 25 mg 167465-36-3

Product Name Cat. No. Size CAS. No.AMG-232 9556 1 mg, 5 mg 1352066-68-2CGM097 B1820 1 mg, 5 mg 1313363-54-0JNJ-26854165 2479 5 mg, 25 mg 881202-45-5MI-773 9610 1 mg, 5 mg 1303607-60-4MX69 B1568 5 mg, 25 mg 1005264-47-0 Nutlin-3 1842 1 mg, 5 mg 548472-68-0Nutlin-3b B1227 1 mg, 5 mg 675576-97-3EZSolution™ RG7388 B1504 1 mg 1229705-06-9RG7388 2577 1 mg, 5 mg 1229705-06-9RO8994 B1830 5 mg, 25 mg 1309684-94-3 YH239-EE B1229 5 mg, 25 mg 1364488-67-4

MDM2 (Murine Double Minute 2) Inhibitors

Methyltransferase InhibitorsProduct Name Cat. No. Size CAS. No.A-366 2859 1 mg, 5 mg 1527503-11-2AMI-1 1943 5 mg, 25 mg 20324-87-2AMI-5 2300 50 mg, 250 mg 17372-87-15-Aza-2'-deoxycytidine 1754 10 mg, 50 mg 2353-33-5AZ-505 ditrifluoroacetate B1883 1 mg, 5 mg 1035227-44-1EZSolution™ BIX 01294 2661 5 mg 935693-62-2BIX 01294 1678 5 mg, 25 mg 935693-62-2BRD4770 9525 5 mg, 25 mg 1374601-40-7Bromodomain Inhibitor, (+)-JQ1 2070 1 mg, 5 mg 1268524-70-4C7280948 B1153 10 mg, 50 mg 587850-67-7Chaetocin 2283 500 µg 28097-03-2EZSolution™ 3-Deazaneplanocin A 2409 1 mg 102052-95-93-Deazaneplanocin A 2060 250 µg, 1 mg 102052-95-93-Deazaneplanocin A hydrochloride 2444 250 µg, 1 mg 120964-45-62'-Deoxy-5-fluorocytidine 2387 50 mg, 250 mg 10356-76-05’-Deoxy-5’-methylthioadenosine BA1053 10 mg, 50 mg 2457-80-9DNA methylation inhibitor, Dichlone 2860 500 mg, 1 g 117-80-6EED-226 B1845 5 mg, 25 mg 2083627-02-3 Ellagic Acid B1154 100 mg, 500 mg 476-66-4EPZ004777 2381 1 mg, 5 mg 1338466-77-5EZSolution™ EPZ005687 2375 2 mg 1396772-26-1EPZ011989 B1221 5 mg, 25 mg 1598383-40-4EPZ-015666 9410 1 mg, 5 mg 1616391-65-1EPZ015866 (GSK591) B1216 5 mg, 25 mg 1616391-87-7EZSolution™ EPZ-5676 2427 1 mg 1380288-87-8EPZ-5676 2382 1 mg, 5 mg 1380288-87-8EZSolution™ EPZ-6438 2428 5 mg 1403254-99-8EPZ-6438 2383 5 mg, 25 mg 1403254-99-8EZH2 Inhibitor, EPZ005687 2364 2 mg, 10 mg 1396772-26-1EZSolution™ GSK126 2366 1 mg 1346574-57-9GSK126 2282 1 mg, 5 mg 1346574-57-9EZSolution™ GSK343 2365 1 mg N/AGSK343 2281 1 mg, 5 mg 1346704-33-3GSK-503 9538 5 mg, 25 mg 1346572-63-1HLCL-61 hydrochloride B1209 5 mg, 25 mg 586395-74-6EZSolution™ (+)-JQ1 2091 1 mg 1268524-70-4

MDR (Multidrug Resistance) Inhibitors

Product Name Cat. No. Size CAS. No.LLY-507 B1111 1 mg, 5 mg 1793053-37-8Lomeguatrib 2224 5 mg, 25 mg 192441-08-0MAK-683 B1972 5 mg, 25 mg 1951408-58-4MI-2 B1835 5 mg, 25 mg 1271738-62-5MI-3 B1834 5 mg, 25 mg 1271738-59-0Nanaomycin A 2790 1 mg, 5 mg 52934-83-5OICR-9429 B1256 5 mg, 25 mg 1801787-56-3 PFI-2 B1259 5 mg, 25 mg 1627676-59-8RG 108 1679 10 mg, 30 mg 48208-26-0Ryuvidine B1808 1 mg, 5 mg 265312-55-8SGC0946 2448 5 mg, 25 mg 1561178-17-3SGI-1027 2726 5 mg, 25 mg 1020149-73-8TC-E 5003 B1177 10 mg, 50 mg 17328-16-4UNC0379 9588 5 mg, 25 mg 1620401-82-2UNC0631 2605 5 mg, 25 mg 1320288-19-4UNC0638 1933 1 mg, 5 mg 1255580-76-7UNC0642 2862 5 mg, 25 mg 1481677-78-4UNC0646 2606 5 mg, 25 mg 1320288-17-2UNC1999 2449 5 mg, 25 mg 1431612-23-5WDR5 0103 B1125 10 mg, 50 mg 890190-22-4Zebularine 2225 1 mg, 5 mg 3690-10-6

Product Name Cat. No. Size CAS. No.ABT751 2836 5 mg, 25 mg 141430-65-1Colchicine 1519 1 g 64-86-8Combretastatin A4 2239 10 mg, 50 mg 117048-59-6CW069 9507 10 mg, 50 mg 1594094-64-0Cytochalasin D B1176 1 mg, 5 mg 22144-77-0D-64131 B1066 10 mg, 50 mg 74588-78-6Docetaxel 2232 10 mg, 50 mg 114977-28-5ELR-510444 9433 5 mg, 25 mg 1233948-35-0Epothilone B 2012 1 mg, 5 mg 152044-54-7Epothilone D 9559 1 mg, 5 mg 189453-10-9Maytansinol B2015 5 mg, 25 mg 57103-68-1EZSolution™ Nocodazole B1874 5 mg 31430-18-9Nocodazole 2185 10 mg, 50 mg 31430-18-9Paclitaxel 1567 25 mg 33069-62-4

Podophyllotoxin 2767 50 mg, 250 mg 518-28-5, 4354-76-1

Pseudolaric Acid B 2512 1 mg, 5 mg 82508-31-4Thiocolchicine 2213 5 mg, 25 mg 2730-71-4Vinblastine Sulfate 1959 5 mg, 25 mg 143-67-9Vinorelbine Tartrate 1957 5 mg, 25 mg 125317-39-7

Microtubule Inhibitors

Product Name Cat. No. Size CAS. No.MIF-Antagonist, ISO-1 1895 5 mg 478336-92-4MIF antagonist, p425 2158 1 g 2610-05-1

MIF (Migration Inhibitory Factor) Antagonists

Product Name Cat. No. Size CAS. No.Mdivi -1 2441 5 mg, 25 mg 338967-87-6

Mitochondrial Division Inhibitors

Product Name Cat. No. Size CAS. No.Antimycin A 2247 10 mg, 50 mg 1397-94-0Atpenin A5 (Synthetic) 2210 250 µg, 1 mg 119509-24-9Cyantraniliprole B1648 5 mg, 25 mg 736994-63-1Phenformin hydrochloride 1889 100 mg, 1 g 834-28-6Rotenone 2248 250 mg, 1 g 83-79-4

Mitochondrial Electron Transport Chain Inhibitors

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Product Name Cat. No. Size CAS. No.Myeloperoxidase Inhibitor 1977 100 mg, 500 mg 5351-17-7

MPO (Myeloperoxidase) Inhibitors

Product Name Cat. No. Size CAS. No.NAALDase Inhibitor, PMPA 2478 5 mg, 25 mg 173039-10-6

NAALADase (N-Acetylated-Alpha-Linked-Acidic Dipeptidase) Inhibitors

Product Name Cat. No. Size CAS. No.CHS-828 2044 5 mg, 25 mg 200484-11-3FK-866 1914 1 mg, 5 mg 658084-64-1Nampt-IN-1 B1171 5 mg, 25 mg 1698878-14-6STF-118804 9552 5 mg, 25 mg 894187-61-2STF-31 9585 5 mg, 25 mg 724741-75-7

Nampt (Nicotinamide Phosphoribosyltransferase) Inhibitors

Product Name Cat. No. Size CAS. No.EZSolution™ Nec-1s 2535 1 mg N/ANec-1s 2263 1 mg, 5 mg 852391-15-2Necrosis Inhibitor, Necrox-2 2228 1 mg, 5 mg N/ANecrosis Inhibitor, Necrox-5 2229 1 mg, 5 mg 1383718-29-3Necrostatin-1 1864 5 mg, 25 mg 4311-88-0Necrostatin-5 1865 5 mg, 25 mg 337349-54-9Necrostatin-7 1866 5 mg, 25 mg 351062-08-3EZSolution™ Necrosulfonamide, Sterile-Filtered B1220 10 mg 1360614-48-7

Necrosulfonamide 9635 10 mg, 50 mg 1360614-48-7

Necroptosis and Necrosis Inhibitors

Product Name Cat. No. Size CAS. No.Arglabin 9691 1 mg, 5 mg 84692-91-1Isoliquiritigenin 2528 5 mg, 25 mg 961-29-5MCC950 (Free base) B1031 1 mg, 5 mg 210826-40-7MCC950 sodium 9686 1 mg, 5 mg 256373-96-3

Product Name Cat. No. Size CAS. No.Andrographolide 2389 50 mg, 250 mg 5508-58-7BAY 11-7082 1867 10 mg, 50 mg 19542-67-7Berbamine dihydrochloride 2520 100 mg, 500 mg 6078-17-7BMS-345541 (Free base) B1907 1 mg, 5 mg 445430-58-0Celastrol 1940 5 mg, 25 mg 34157-83-0CHS-828 2044 5 mg, 25 mg 200484-11-3Dimethyl Fumarate 9660 100 mg, 500 mg 624-49-7Honokiol 1762 10 mg, 50 mg 35354-74-64'-Hydroxychalcone B1921 250 mg, 1 g 2657-25-2IKK16 B1087 5 mg, 25 mg 1186195-62-9ML130 1974 5 mg, 25 mg 799264-47-4

NF-KB (Nuclear Factor-kappa B) Pathway Inhibitors

Product Name Cat. No. Size CAS. No.Bakuchiol 2494 1 mg, 5 mg 10309-37-2Bardoxolone B1170 5 mg, 25 mg 218600-44-33-Bromo-7-nitroindazole 2361 10 mg, 50 mg 74209-34-0Curvularin 9694 1 mg, 5 mg 10140-70-2Diphenyleneiodonium chloride 2358 5 mg 4673-26-1L-NAME hydrochloride 2356 100 mg, 500 mg, 1 g 51298-62-5L-NMMA acetate 2348 5 mg, 25 mg, 100 mg 53308-83-17-Nitroindazole 2360 50 mg, 250 mg 2942-42-91400W dihydrochloride 2055 5 mg, 25 mg 214358-33-5

NOS (Nitric Oxide Synthase) Inhibitors

Product Name Cat. No. Size CAS. No.EZSolution™ Leptomycin B 1814 25 µg 87081-35-4

Nuclear Export Inhibitors

NLRP3 (NOD-Like Receptor Pyrin domain-containing protein 3) Inflammasome Inhibitors

Product Name Cat. No. Size CAS. No.Apremilast 2352 5 mg, 25 mg 608141-41-9Cilostamide 2560 5 mg, 25 mg 68550-75-4Cilostazol 2393 5 mg, 25 mg 73963-72-1EHNA hydrochloride 2265 5 mg, 25 mg 58337-38-5GSK-356278 B1292 5 mg, 25 mg 720704-34-7IBMX 1714 100 mg 28822-58-4Ibudilast B1327 5 mg, 25 mg 50847-11-5Milrinone 2163 5 mg, 25 mg 78415-72-2PF-04447943 B1264 5 mg, 25 mg 1082744-20-4Pimobendan 9676 50 mg, 250 mg 74150-27-9RO 20-1724 2042 50 mg, 250 mg 29925-17-5Roflumilast 2675 10 mg, 50 mg 162401-32-3(R,S)-Rolipram 2010 5 mg 61413-54-5

PDE (Phosphodiesterase) Inhibitors

Product Name Cat. No. Size CAS. No.SBC-110736 B1304 5 mg, 25 mg 1629166-02-4

PCSK9 (Proprotein Convertase Subtilisin Kexin 9) Inhibitors

Product Name Cat. No. Size CAS. No.Atpenin A5 (Synthetic) 2210 250 µg 119509-24-9EZSolution™ Batimastat 2540 1 mg 130370-60-4Batimastat (MMP Inhibitor) 1704 1 mg, 5 mg 130370-60-4Disulfiram 2308 50 mg, 250 mg 97-77-8Doxycycline hyclate 2209 100 mg, 500 mg 24390-14-5GM 6001 1799 1 mg 142880-36-2Marimastat 1790 1 mg, 5 mg 154039-60-8Minocycline Hydrochloride B1525 50 mg, 250 mg 13614-98-7MMP-13 inhibitor 2392 5 mg, 25 mg 307002-71-7MMP-9 Inhibitor 1981 500 µg 1177749-58-4MMP-III Inhibitor, NNGH 2569 5 mg, 25 mg 161314-17-6NSC 405020 2682 5 mg, 25 mg 7497-07-6TAPI-0 2067 1 mg 143457-40-3EZSolution™ TAPI-1 2537 1 mg 171235-71-5TAPI-1 2068 1 mg 171235-71-5TAPI-2 2069 1 mg 187034-31-7WAY-170523 9607 1 mg, 5 mg 307002-73-9

MMP (Matrix Metalloproteinase) Inhibitors

Product Name Cat. No. Size CAS. No.GSK-106 hydrochloride B1036 500 µg, 1 mg 1652591-82-6GSK-121 trifluoroacetate B1034 500 µg, 1 mg 1652591-80-4GSK-199 hydrochloride B1037 500 µg, 1 mg 1549811-53-1GSK-484 hydrochloride B1035 500 µg, 1 mg 1652591-81-5

PAD (Protein Arginine Deiminase) Inhibitors

Product Name Cat. No. Size CAS. No.MRT67307 B1604 5 mg, 25 mg 1190378-57-4NF-κB Inhibitor, SN50 2506 500 µg, 1 mg 213546-53-3Parthenolide 1868 10 mg, 50 mg 20554-84-1PDTC 1676 100 mg 5108-96-3PS-1145 9671 5 mg, 25 mg 431898-65-6Rocaglamide 1863 100 µg 84573-16-0Sauchinone 2312 1 mg, 5 mg 177931-17-8SC-514 2442 5 mg, 25 mg 354812-17-2STO-609 B1609 5 mg, 25 mg 52029-86-4 TPCA-1 2431 5 mg, 25 mg 507475-17-4Triptolide 1761 1 mg, 5 mg 38748-32-2

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Product Name Cat. No. Size CAS. No.NSC 66811 2009 5 mg 6964-62-1

p53 Inhibitors

Product Name Cat. No. Size CAS. No.Bakuchiol 2494 1 mg, 5 mg 10309-37-2bpV(phen) 1793 5 mg 42494-73-5bpV(pic) 1794 5 mg 148556-27-8BVT948 B1810 1 mg, 5 mg 39674-97-0Calyculin A 1562 25 µg 101932-71-2Cantharidin 2510 10 mg, 50 mg 56-25-7Cyclosporine A 1522 100 mg, 1 g 59865-13-3Cytostatin sodium B1240 250 µg 457070-06-3 FK-506 1563 1 mg, 10 mg 104987-11-3Fostriecin sodium B1241 10 µg 87860-39-7GSK2830371 2578 1 mg, 5 mg 1404456-53-6IQ-1 1663 1 mg 331001-62-8Microcystin-LR 1840 100 µg, 500 µg 101043-37-2Nodularin 2094 50 µg 118399-22-7NSC-663284 B1809 1 mg, 5 mg 383907-43-5NSC-87877 2687 10 mg, 50 mg 56990-57-9Okadaic acid 1543 25 µg, 100 µg 78111-17-8Okadaic acid, Ammonium Salt 1766 25 µg, 100 µg 155716-06-6Okadaic acid, Potassium Salt 1765 25 µg, 100 µg 155751-72-7Okadaic acid, Sodium Salt 1764 25 µg, 100 µg 209266-80-8(-)-p-Bromotetramisole oxalate 1901 5 mg, 25 mg 62284-79-1EZBlock™ Phosphatase Inhibitor Cocktail I (50X) K273 1 ml, Set (5 x 1 ml) N/A

EZBlock™ Phosphatase Inhibitor Cocktail II K275 1 ml, Set (5 x 1 ml) N/AEZBlock™ Phosphatase Inhibitor Cocktail III K276 1 ml, Set (5 x 1 ml) N/A

EZBlock™ Phosphatase Inhibitor Cocktail IV K282 1 ml, Set (5 x 1 ml) N/A

EZBlock™ Phosphatase Inhibitor Cocktail XI K298 1 vial, Set (5 x 1 vial) N/A

PRL-3 Inhibitor B1825 5 mg, 25 mg 893449-38-2Rubratoxin A B1239 250 µg , 500 µg 22467-31-8SHP099 hydrochloride B1308 5 mg, 25 mg 1801747-11-4Sodium orthovanadate 9470 1 g, 5 g 13721-39-6Sodium orthovanadate, Activated 9471 5 ml 13721-39-6Tautomycin B1237 10 µg, 50 µg 109946-35-2EZBlock™ Universal Protease and \Phosphatase Inhibitor Cocktail K283 2 vials, 10 vials N/A

EZBlock™ Universal Protease and Phosphatase Inhibitor Cocktail , EDTA-Free K284 1 ml, Set (5 x 1 ml) N/A

Phosphatase Inhibitors

Product Name Cat. No. Size CAS. No.Darapladib B1265 5 mg, 25 mg 356057-34-6 FIPI 9593 5 mg, 25 mg 939055-18-2LY315920 2666 1 mg, 5 mg 172732-68-2U-73122 B1887 5 mg, 25 mg 112648-68-7U-73343 B1888 5 mg, 25 mg 142878-12-4

Phospholipase Inhibitors

Product Name Cat. No. Size CAS. No.ABT-888 1620 1 mg, 5 mg 912445-05-7AG-014699 phosphate 2890 1 mg, 5 mg 459868-92-9BMN-673 B1861 1 mg, 5 mg 1207456-01-6EZSolution™ DPQ 2866 5 mg 129075-73-6DPQ 1899 1 mg, 5 mg 129075-73-6DR2313 1771 1 mg, 5 mg 284028-90-6Iniparib 1968 5 mg, 25 mg 160003-66-71,5-Isoquinolinediol 2415 10 mg, 50 mg 5154-02-9ME-0328 2751 5 mg, 25 mg 1445251-22-8MK-4827 9462 5 mg, 25 mg 1038915-60-4MK-4827 (Tosylate) B2003 5 mg, 25 mg 1038915-73-9NU 1025 2351 1 mg, 5 mg 90417-38-2Olaparib 1952 5 mg, 25 mg 763113-22-0Phenformin hydrochloride 1889 100 mg, 1 g 834-28-6PJ-34 hydrochloride 2319 1 mg, 5 mg 344458-15-7

Poly (ADP-ribose) Polymerase (PARP) Inhibitors

Product Name Cat. No. Size CAS. No.Astaxanthin 9698 5 mg, 25 mg 472-61-7GSK-0660 2897 5 mg, 25 mg 1014691-61-2GSK-3787 2400 5 mg, 25 mg 188591-46-0GW 9662 1697 5 mg 22978-25-2GW-6471 9453 1 mg, 5 mg 880635-03-0EZSolution™ GW 9662 9651 5 mg 22978-25-2PPARγ Antagonist, G3335 1979 10 mg, 25 mg 36099-95-3SR1664 9432 1 mg, 5 mg 1338259-05-4T0070907 2095 5 mg 313516-66-4

PPAR (Peroxisome Proliferator-Activated Receptor) Antagonists

Product Name Cat. No. Size CAS. No.β-Glycyrrhetinic acid 9586 1 g 471-53-4SW-033291 9584 5 mg, 25 mg 459147-39-8

15-PGDH (15-hydroxy Prostaglandin Dehydrogenase) Inhibitors

PPI (Protein-Protein Interaction) Inhibitors Product Name Cat. No. Size CAS. No.ABT-263 2467 5 mg, 25 mg 923564-51-6AT-406 B1829 5 mg, 25 mg 1071992-99-8BCl-2 Inhibitor, ABT-199 2253 1 mg, 5 mg 1257044-40-8Birinapant 2597 1 mg, 5 mg 1260251-31-7Bromodomain Inhibitor, (+)-JQ1 2070 1 mg, 5 mg 1268524-70-4CPI-203 9404 1 mg, 5 mg 1446144-04-2GDC-0152 B1602 5 mg, 25 mg 873652-48-3GDC-0917 B1918 1 mg, 5 mg 1446182-94-0I-BET151 2220 1 mg, 5 mg 1300031-49-5I-BET726 B1569 5 mg, 25 mg 1300031-52-0I-BET762 2628 1 mg, 5 mg 1260907-17-2EZSolution™ (+)-JQ1 2091 1 mg 1268524-70-4(-)-JQ1 2384 1 mg 1268524-71-5LCL161 B1601 5 mg, 25 mg 1005342-46-0Lifitegrast B1917 5 mg, 25 mg 1025967-78-5MS436 2680 5 mg, 25 mg 1395084-25-9OTX015 2651 1 mg, 5 mg 202590-98-5PFI-1 2203 1 mg, 5 mg 1403764-72-6RG-7112 B1919 1 mg, 5 mg 939981-39-2EZSolution™ RG7388 B1504 1 mg 1229705-06-9RG7388 2577 1 mg, 5 mg 1229705-06-9RVX-208 9408 1 mg, 5 mg 1044870-39-4

Product Name Cat. No. Size CAS. No.Sildenafil citrate 2872 10 mg, 50 mg 171599-83-0TAK-063 B1067 10 mg, 50 mg 1238697-26-1Vesnarinone B2008 5 mg, 25 mg 81840-15-5 Zaprinast 1715 25 mg 37762-06-4

Product Name Cat. No. Size CAS. No.Pifithrin-α, Cyclic, hydrobromide 2270 5 mg 511296-88-1Pifithrin-α 1554 10 mg 63208-82-2

Product Name Cat. No. Size CAS. No.Abametapir 9665 100 mg, 500 mg 1762-34-1

Protease Inhibitors

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Product Name Cat. No. Size CAS. No.EZSolution™ A83-01, Sterile-Filtered 1989 1 ml 909910-43-6A 83-01 1725 1 mg 909910-43-6ASP-3026 B1296 5 mg, 25 mg 1097917-15-1AZD-3463 2371 5 mg, 25 mg 1356962-20-3Belizatinib (TSR-011) B2028 5 mg, 25 mg 1357920-84-3Brigatinib (AP26113) 9675 5 mg, 25 mg 1197953-54-0Brigatinib analog B2025 5 mg, 25 mg 1197958-12-5CH5424802 2867 5 mg, 25 mg 1256580-46-7Crizotinib 1934 5 mg, 25 mg 877399-52-5Ensartinib B1946 5 mg, 25 mg 1365267-27-1Entrectinib B1324 5 mg, 25 mg 1108743-60-7GSK-1838705A B2026 1 mg, 5 mg 1116235-97-2 LDK-378 B1928 5 mg, 25 mg 1032900-25-6NVP-TAE684 1683 5 mg 761439-42-3PF-06463922 B1169 10 mg, 50 mg 1454846-35-5SU-5416 9491 5 mg, 25 mg 204005-46-9TPX-0005 B2027 5 mg, 25 mg 2058227-19-1

Product Name Cat. No. Size CAS. No.AEBSF.HCl 1644 200 mg, 1 g 30827-99-7Alvelestat B1653 5 mg, 25 mg 848141-11-7Antipain dihydrochloride 2834 5 mg, 25 mg 37682-72-7Aprotinin 4690 5 mg, 100 mg, 1 g 9087-70-1 Argatroban 9670 10 mg, 50 mg 141396-28-3Batimastat (MMP Inhibitor) 1704 1 mg, 5 mg 130370-60-4Bestatin 1733 25 mg, 100 mg 58970-76-6Bestatin hydrochloride 9630 5 mg, 25 mg 65391-42-6Clasto-Lactacystin β-lactone 1710 100 µg 154226-60-5E-64 1739 5 mg, 25 mg 66701-25-5Elastase Inhibitor 1922 5 mg 111682-13-4Elastase Inhibitor, SPCK 1921 5 mg 65144-34-5Elastatinal 9629 5 mg, 25 mg 51798-45-9Enfuvirtide Acetate 2440 1 mg 914454-00-5GGACK Dihydrochloride 1847 5 mg N/ALactacystin (Synthetic) 1709 200 µg 133343-34-7Leupeptin, hemisulfate (Microbial) 1648 25 mg, 50 mg, 100 mg 103476-89-7Lopinavir 2241 50 mg, 250 mg 192725-17-0EZSolution™ MG-132 1791 5 mg 133407-82-6MG-132 1703 5 mg, 25 mg 133407-82-6Nafamostat Mesylate 1760 10 mg, 50 mg 82956-11-4Pepstatin A 1732 25 mg, 100 mg 26305-03-3PMSF 1548 5 g, 25 g 329-98-6PPACK Dihydrochloride 1848 5 mg N/AEZBlock™ Protease Inhibitor Cocktail, EDTA-Free K272 1 ml, 5 ml, Set (5 x 1 ml) N/A

EZBlock™ Protease Inhibitor Cocktail II K277 Set (5 x 1 vial) N/AEZBlock™ Protease Inhibitor Cocktail II, Animal-Free K394 1 vial, Set (5 x 1 vial) N/A

EZBlock™ Protease Inhibitor Cocktail III K278 Set (1 vial of lyophilized cocktail + 1 ml DMSO) N/A

EZBlock™ Protease Inhibitor Cocktail IV K279 1 ml, Set (5 x 1 ml) N/AEZBlock™ Protease Inhibitor Cocktail IX K294 1 ml, Set (5 x 1 ml) N/AEZBlock™ Protease Inhibitor Cocktail V, EDTA-Free K290 1 vial, Set (5 x 1 vial) N/A

EZBlock™ Protease Inhibitor Cocktail VI, General Use K291 1 vial, Set (5 x 1 vial) N/A

EZBlock™ Protease Inhibitor Cocktail VII K292 1 ml, Set (5 x 1 ml) N/AEZBlock™ Protease Inhibitor Cocktail VIII K293 1 ml, Set (5 x 1 ml) N/AEZBlock™ Protease Inhibitor Cocktail VIII, DMSO-Free K395 1 vial, Set (5 x 1 vial) N/A

EZBlock™ Protease Inhibitor Cocktail X, EDTA-Free K297 1 vial, Set (5 x 1 vial) N/A

EZBlock™ Protease Inhibitor Cocktail XII, EDTA-free, Animal-free K221 1 vial, Set (5 x 1 vial) N/A

EZBlock™ Protease Inhibitor Cocktail XIII, EDTA & Animal-Free K222 1 vial, Set (5 x 1 vial) N/A

EZBlock™ Protease Inhibitor Cocktail XIV K223 1 vial, Set (5 x 1 vial) N/AEZBlock™ Protease Inhibitor Cocktail XV K393 1 vial, Set (5 x 1 vial) N/AProtease Inhibitor Cocktail K271 1 Kit N/ASimeprevir B1173 5 mg, 25 mg 923604-59-5EZBlock™ Universal Protease and Phosphatase Inhibitor Cocktail K283 2 vials, 10 vials N/A

EZBlock™ Universal Protease and Phosphatase Inhibitor Cocktail , EDTA-Free K284 1 ml, Set (5 x 1 ml) N/A

Vicriviroc Malate 1599 1 mg, 5 mg 541503-81-5

Product Name Cat. No. Size CAS. No.Aclacinomycin A hydrochloride B1905 1 mg, 5 mg 75443-99-1Calpain Inhibitor I, ALLN 1834 5 mg, 25 mg 110044-82-1Calpain Inhibitor II, ALLM 1835 5 mg, 25 mg 136632-32-1Carfilzomib 2385 5 mg, 25 mg 868540-17-4Celastrol 1940 5 mg, 25 mg 34157-83-0CEP-18770 2433 5 mg, 25 mg 847499-27-8Clasto-Lactacystin β-lactone 1710 100 µg 154226-60-5Clioquinol 2454 1 g, 5 g 130-26-7

Proteasome Inhibitors

Product Name Cat. No. Size CAS. No.Afuresertib hydrochloride B1848 5 mg, 25 mg 1047645-82-8Akt Inhibitor (10-NCP) 2338 1 mg, 5 mg 925681-41-0Akt Inhibitor, Isozyme-Selective 1708 1 mg 612847-09-3Akt-I-1 B1610 1 mg, 5 mg 473382-39-7Cordycepin 2078 10 mg, 50 mg 73-03-0GDC-0068 2667 1 mg, 5 mg 1001264-89-6GSK-2110183 B1089 1 mg, 5 mg 1047644-62-1GSK-690693 2272 5 mg, 25 mg 937174-76-0Miransertib B1931 5 mg, 25 mg 1313881-70-7MK-2206 1888 500 µg, 1 mg 1032350-13-2Perifosine (KRX-0401) 1592 5 mg, 25 mg 157716-52-4

DiscoveryPak™ PI 3-Kinase Inhibitor Set(Containing Cat. No. 1661, 1667, 1728, 1780, 1781)

K856 5 Inhibitors

371242-69-2 154447-36-6 371935-74-9 648450-29-7 663619-89-4

PHT-427 2465 10 mg, 50 mg 1191951-57-1SC66 1870 10 mg, 50 mg 871361-88-5SH-5 1818 500 µg 701976-54-7SH-6 1819 500 µg 701976-54-7Triciribine 1707 1 mg 35943-35-2

Protein Kinase InhibitorsAkt (thymoma viral proto-oncogene 1) Inhibitors

ALK (Anaplastic Lymphoma Kinase) Inhibitors

Product Name Cat. No. Size CAS. No.EZSolution™ Dorsomorphin 2547 5 mg 866405-64-3

AMPK (AMP-activated protein Kinase) Inhibitors

Product Name Cat. No. Size CAS. No.(-)-Epigallocatechin gallate 1841 50 mg 989-51-5Epoxomicin 2190 50 µg, 250 µg 134381-21-8Fenbendazole 2157 100 mg, 500 mg 43210-67-9Lactacystin (Natural) 2434 200 µg 133343-34-7Lactacystin (Synthetic) 1709 200 µg 133343-34-7EZSolution™ MG-115 2144 1 mg N/AMG-115 1831 1 mg, 5 mg N/AEZSolution™ MG-132 1791 5 mg 133407-82-6MG-132 1703 5 mg, 25 mg 133407-82-6ONX-0914 2555 5 mg, 25 mg 960374-59-8Oprozomib 2386 5 mg, 25 mg 935888-69-0P5091 2277 5 mg, 25 mg 882257-11-6EZSolution™ PS-341 2145 1 mg 179324-69-7PS-341 1846 1 mg, 5 mg 179324-69-7VR23 B1515 5 mg, 25 mg 1624602-30-7

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Product Name Cat. No. Size CAS. No.ATM Kinase Inhibitor, KU-55933 1685 5 mg 587871-26-9AZD-0156 B1305 5 mg, 25 mg 1821428-35-6Ku-60019 9572 5 mg, 25 mg 925701-49-1

ATM (Ataxia Telangiectasia Mutated ) Kinase Inhibitors

Product Name Cat. No. Size CAS. No.AZ20 B1724 1 mg, 5 mg 1233339-22-4AZD-6738 B1167 5 mg, 25 mg 1352226-88-0BAY-1895344 hydrochloride B1962 5 mg, 25 mg 1876467-74-1CGK733 B1725 5 mg, 25 mg 905973-89-9ETP-46464 2457 5 mg, 25 mg 1345675-02-6VE-821 B1723 5 mg, 25 mg 1232410-49-9VE-822 2840 5 mg, 25 mg 1232416-25-9

ATR (Ataxia Telangiectasia & Rad3-related) Inhibitors

Product Name Cat. No. Size CAS. No.656820-32-5 B1638 5 mg, 25 mg 160098-96-4AMG-900 B1343 5 mg, 25 mg 945595-80-2AT9283 2432 5 mg, 25 mg 896466-04-9Aurora Kinase B Inhibitor (AZD1152-HQPA) 1583 5 mg, 25 mg 722544-51-6CCT-129202 B1934 1 mg, 5 mg 942947-93-5CCT-137690 B195 5 mg, 25 mg 1095382-05-0CYC-116 B1936 5 mg, 25 mg 693228-63-6Danusertib B1937 5 mg, 25 mg 827318-97-8ENMD-2076 B1938 5 mg, 25 mg 934353-76-1GSK-1070916 B1939 5 mg, 25 mg 942918-07-2Hesperadin B1940 5 mg, 25 mg 422513-13-1JNJ-7706621 B1941 1 mg, 5 mg 443797-96-4MK-5108 B1344 5 mg, 25 mg 1010085-13-8MK-8745 B1942 5 mg, 25 mg 885325-71-3MLN-8054 B1943 5 mg, 25 mg 869363-13-3MLN8237 2718 5 mg, 25 mg 1028486-01-2PF-03814735 B1257 5 mg, 25 mg 942487-16-3PHA-680632 B1944 5 mg, 25 mg 398493-79-3Reversine 1851 1 mg, 5 mg 656820-32-5SNS-314 2446 5 mg, 25 mg 1057249-41-8TAK-901 B1945 5 mg, 25 mg 934541-31-8TC-S 7010 B1203 5 mg, 25 mg 1158838-45-9EZSolution™ Tozasertib 1803 25 mg 639089-54-6Tozasertib (VX-680, MK-0457, VX6) 1595 25 mg, 100 mg 639089-54-6Tripolin A 2307 1 mg, 5 mg 1148118-92-6ZM 447439 2018 1 mg, 5 mg 331771-20-1

Aurora Kinase Inhibitors

Product Name Cat. No. Size CAS. No.BMS-777607 2455 5 mg, 25 mg 1025720-94-8R428 9591 5 mg, 25 mg 1037624-75-1SGI-7079 B1202 5 mg, 25 mg 1239875-86-5TP-0903 9590 5 mg, 25 mg 1341200-45-0

Axl Receptor Tyrosine Kinase Inhibitors

BTK (Bruton’s Tyrosine Kinase) InhibitorsProduct Name Cat. No. Size CAS. No.Acalabrutinib B1193 5 mg, 25 mg 1420477-60-6AVL-292 (Spebrutinib) 9413 5 mg, 25 mg 1202757-89-8BTK Inhibitor, CNX-774 2600 5 mg, 25 mg 1202759-32-7BTK Inhibitor, PCI-32765 2298 5 mg, 25 mg 936563-96-1CGI-1746 9647 5 mg, 25 mg 910232-84-7LFM-A13 2414 5 mg, 25 mg 244240-24-2ONO-4059 B1283 5 mg, 25 mg 1351636-18-4

CaM (Ca2+/calmodulin-dependent) Kinase InhibitorsProduct Name Cat. No. Size CAS. No.Berbamine dihydrochloride 2520 100 mg, 500 mg 6078-17-7K252a 2013 500 µg, 1 mg 99533-80-9KN-62 2495 1 mg, 5 mg 127191-97-3KN-92 hydrochloride B1643 5 mg, 25 mg 1431698-47-3KN-92 phosphate B1644 5 mg, 25 mg 1135280-28-2KN-93 2524 250 µg, 1 mg 139298-40-1KN-93, Water-Soluble 1909 1 mg, 5 mg 1188890-41-6STO-609 B1609 5 mg, 25 mg 52029-86-4

CDC7 (Cell Division Cycle 7 Homolog) InhibitorsProduct Name Cat. No. Size CAS. No.BMS-863233 hydrochloride 2598 5 mg, 25 mg 1169562-71-3PHA-767491(HCl) B1639 5 mg, 25 mg 845714-00-3

CDK (Cyclin-Dependent Kinases) InhibitorsProduct Name Cat. No. Size CAS. No.Alsterpaullone 1897 1 mg, 5 mg 237430-03-4AMG-925 B1959 5 mg, 25 mg 1401033-86-0Aminopurvalanol A 2205 1 mg, 5 mg 220792-57-4AT-7519 hydrochloride 2816 5 mg, 25 mg 902135-91-5Bohemine B1040 10 mg, 50 mg 189232-42-6Butyrolactone I 1690 200 µg 87414-49-1CVT-313 B1137 5 mg, 25 mg 199986-75-9Dinaciclib 9537 5 mg, 25 mg 779353-01-4Flavopiridol 2090 1 mg, 5 mg 146426-40-6Kenpaullone 1904 1 mg 142273-20-9LY-2835219 B1039 10 mg, 50 mg 1231930-82-7MSC-2530818 B1975 1 mg, 5 mg 1883423-59-3 NG52 9420 5 mg, 25 mg 212779-48-1NU6102 2313 1 mg, 5 mg 444722-95-6ON-013100 B1276 5 mg, 25 mg 865783-95-5 PD-0332991 2843 5 mg, 25 mg 571190-30-2PD-0332991 isethionate 9480 5 mg, 25 mg 827022-33-3RGB-286638, free base 2886 5 mg, 25 mg 784210-88-4Ribociclib (LEE011) 9481 5 mg, 25 mg 1211441-98-3(R)-Perharidine-1 2615 1 mg, 5 mg 1133437-80-5RO-3306 2039 1 mg, 5 mg 872573-93-8Roscovitine 1950 1 mg, 5 mg 186692-46-6SNS-032 9490 5 mg, 25 mg 345627-80-7TG003 1905 5 mg, 25 mg 300801-52-9THZ1 (Free base) 9664 5 mg, 25 mg 1604810-83-4THZ1 hydrochloride 9544 5 mg, 25 mg 1604810-83-410Z-Hymenialdisine 2212 250 µg, 1 mg 82005-12-7

Product Name Cat. No. Size CAS. No.Dorsmorphin dihydrochloride 2835 5 mg, 25 mg 1219168-18-9Dorsomorphin 1686 5 mg 866405-64-3

Product Name Cat. No. Size CAS. No.ONO-4059 analog B1897 5 mg, 25 mg 1351635-67-0RN486 9678 1 mg, 5 mg 1242156-23-5TP-0903 9590 5 mg, 25 mg 1341200-45-0

Chk (Checkpoint Kinase) Kinase InhibitorProduct Name Cat. No. Size CAS. No.AZD-7762 9414 5 mg, 25 mg 860352-01-8CCT244747 9575 5 mg, 25 mg 1404095-34-6Chk2 Inhibitor 1702 1 mg 516480-79-8

CK (Casein kinase) InhibitorsProduct Name Cat. No. Size CAS. No.Apigenin 2508 25 mg, 100 mg 520-36-5BMS-582949 B1704 1 mg, 5 mg 623152-17-0CX-4945 2459 5 mg, 25 mg 1009820-21-6D4476 1770 1 mg, 5 mg 301836-43-1IC261 9669 5 mg, 25 mg 186611-52-9LH-846 9423 10 mg, 50 mg 639052-78-1

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Product Name Cat. No. Size CAS. No.Altiratinib 9563 5 mg, 25 mg 1345847-93-9AMG-208 2553 5 mg, 25 mg 1002304-34-8BMS-777607 2455 5 mg, 25 mg 1025720-94-8Crizotinib 1934 5 mg, 25 mg 877399-52-5Carbozantinib 1935 5 mg, 25 mg 849217-68-1SU 11274 1938 5 mg, 25 mg 658084-23-2Foretinib 9476 5 mg, 25 mg 849217-64-7Golvatinib 2655 5 mg, 25 mg 928037-13-2JNJ-38877605 B2063 5 mg, 25 mg 943540-75-8PF-04217903 B2062 5 mg, 25 mg 956905-27-4PHA-665752 B2057 5 mg, 25 mg 477575-56-7Tivantinib B1546 5 mg, 25 mg 905854-02-6

DNA-PK (DNA-dependent Protein Kinase) InhibitorsProduct Name Cat. No. Size CAS. No.Compound 401 1657 5 mg 168425-64-7KU-0060648 B1115 5 mg, 25 mg 881375-00-4EZSolution™ NU-7441 B1875 5 mg 503468-95-9NU-7441 B1117 5 mg, 25 mg 503468-95-9

DYRK (Dual-specificity Tyrosine Phosphorylation-regulated Kinase) Inhibitors

FAK (Focal Adhesion Kinase) Inhibitors

Product Name Cat. No. Size CAS. No.Leucettine L41 2617 1 mg, 5 mg 1112978-84-3

Product Name Cat. No. Size CAS. No.PF-562271 besylate B1253 5 mg, 25 mg 939791-38-5Y15 B1252 10 mg, 50 mg 4506-66-5

GSK (Glycogen Synthase Kinases) InhibitorsProduct Name Cat. No. Size CAS. No.Alsterpaullone 1897 1 mg, 5 mg 237430-03-41-Azakenpaullone 1944 1 mg, 5 mg 676596-65-9Bikinin 2034 10 mg, 50 mg 188011-69-0BIO 1673 1 mg 667463-62-9Bisindolylmaleimide I 1945 1 mg, 5 mg 133052-90-1Bisindolylmaleimide I hydrochloride 1947 1 mg, 5 mg 176504-36-2Ezsolution™ CHIR-98014 2639 1 mg 556813-39-9CHIR-98014 2595 1 mg, 5 mg 556813-39-9CHIR 99021 1677 5 mg, 25 mg 252917-06-9EZSolution™ CHIR99021 1748 5 mg 252917-06-9EZSolution™ CHIR99021 trihydrochloride, Sterile-Filtered B1219 1 ml 1782235-14-6

CHIR 99021 trihydrochloride B1199 5 mg, 25 mg 1782235-14-6CP21R7 B1563 5 mg, 25 mg 125314-13-8 EZSolution™ CHIR99021, Sterile-Filtered 1991 1 ml 252917-06-9EZSolution™ Necrosulfonamide, Sterile-Filtered B1220 10 mg 1360614-48-7

GSK-3 Inhibitor, AR-A014418 1953 2 mg, 5 mg 487021-52-3

DiscoveryPak™ GSK-3 Inhibitors Set(Containing Cat. No. 1897, 2034, 1677, 2595, 1953, 1655, B1043, 9601)

S237 8 Inhibitors

237430-03-4 188011-69-0 252917-06-9 556813-39-9 487021-52-3 601514-19-6 603288-22-8 865854-05-3

JAK (Janus Kinases) InhibitorsProduct Name Cat. No. Size CAS. No.ABT-494 B1947 5 mg, 25 mg 1310726-60-3AZD1480 2315 1 mg, 5 mg 935666-88-9Baricitinib 2842 10 mg, 50 mg 1187594-09-7Baricitinib phosphate 2841 10 mg, 50 mg 1187595-84-1BMS-911543 2630 1 mg, 5 mg 1271022-90-2Cedrulatinib 2803 5 mg, 25 mg 1198300-79-6CP-690550 1622 5 mg, 25 mg 477600-75-2CP-690550 citrate 9428 5 mg, 25 mg 540737-29-9Cyt387 2316 1 mg, 5 mg 1056634-68-4Decernotinib (VX-509) B1260 5 mg, 25 mg 944842-54-0Filgotinib 2871 10 mg, 50 mg 1206161-97-8GLPG0634 Analog B1836 5 mg, 25 mg 1206101-20-3 INCB39110 B1894 5 mg, 25 mg 1334298-90-6

DiscoveryPak™ JAK Inhibitors Set(Containing Cat. No. 2315, 2842, 2630, 1622, 2316, 2871, 2139, 1853, 1809)

S236 9 Inhibitors

935666-88-91187594-09-71271022-90-2477600-75-21056634-68-41206161-97-8941678-49-5202475-60-3857064-38-1

PathwayReady™ JAK/STAT Signaling Inhibitor Panel(Containing Cat. No. 1570, 1622, 1805, 1792, 1775, 1809, 1887, 1778)

K864 8 Inhibitors

133550-30-8 477600-75-2 111358-88-4 1260247-42-4 501919-59-1 857064-38-1 2062-78-4N/A

LY-2784544 B1914 5 mg, 25 mg 1229236-86-5MS-1020 1911 1 mg 1255516-86-9PF-03394197 2883 5 mg, 25 mg 1208319-26-9Ruxolitinib, Free base 2139 5 mg, 25 mg 941678-49-5SAR-20347 B1290 5 mg, 25 mg 1450881-55-6TG101348 2314 1 mg, 5 mg 936091-26-8Tyrphostin AG 490 1570 5 mg 133550-30-8WHI-P131 1853 5 mg, 25 mg 202475-60-3WHI-P154 2659 5 mg, 25 mg 211555-04-3WP1066 1809 5 mg, 25 mg 857064-38-1

JNK (c-Jun N-terminal Kinase) InhibitorsProduct Name Cat. No. Size CAS. No.AS 602801 B1687 5 mg, 25 mg 848344-36-5AS601245 2162 1 mg, 5 mg 345987-15-7BI-78D3 B1686 5 mg, 25 mg 883065-90-5DB07268 B1134 10 mg, 50 mg 929007-72-7IQ-1S B1279 5 mg, 25 mg 1421610-21-0JNK-IN-7 B1695 1 mg, 5 mg 1408064-71-0JNK-IN-8 2729 5 mg, 25 mg 1410880-22-6L-JNK Peptide Inhibitor I 7011 50 µl N/AEZSolution™ SP600125 9541 5 mg 129-56-6SP600125 1669 5 mg 129-56-6

C-Met (Mesenchymal-Epithelial Transition Factor) Kinase Inhibitors

Product Name Cat. No. Size CAS. No.OSI-930 B1712 5 mg, 25 mg 728033-96-3Pexmetinib B1711 5 mg, 25 mg 945614-12-0PH-797804 B1707 5 mg, 25 mg 586379-66-0SB239063 B1699 5 mg, 25 mg 193551-21-2TA-01 B1214 5 mg, 25 mg 1784751-18-3TA-02 B1215 5 mg, 25 mg 1784751-19-4

Product Name Cat. No. Size CAS. No.GSK-3β Inhibitor, TWS119 1655 2 mg, 5 mg 601514-19-6IM-12 2822 5 mg, 25 mg 1129669-05-1Kenpaullone 1904 1 mg 142273-20-9Leucettine L41 2617 1 mg, 5 mg 1112978-84-3LY-2090314 B1043 5 mg, 25 mg 603288-22-8PKC-9 B1755 5 mg N/ARo 31-8220 methanesulfonate 1946 1 mg, 5 mg 138489-18-6SB 216763 1769 1 mg, 5 mg 280744-09-4SB-415286 B1954 5 mg, 25 mg 264218-23-7TDZD-8 2854 5 mg, 25 mg 327036-89-5Tideglusib 9601 5 mg, 25 mg 865854-05-3

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LRRK2 (Leucine-Rich Repeat Kinase 2) InhibitorsProduct Name Cat. No. Size CAS. No.CZC-54252 hydrochloride 9567 10 mg, 50 mg 1191911-27-9GSK2578215A 2845 5 mg, 25 mg 1285515-21-0HG-10-012-01 2604 5 mg, 25 mg 1351758-81-0JH-II-127 9632 5 mg, 25 mg 1700693-08-8PF-06447475 9447 5 mg, 25 mg 1527473-33-1

Product Name Cat. No. Size CAS. No.APS-2-79 B1696 5 mg, 25 mg 2002381-31-7AZD6244 2234 5 mg, 25 mg 606143-52-6AZD8330 B1693 5 mg, 25 mg 869357-68-6BAY 43-9006 1594 25 mg, 100 mg 475207-59-1BI-847325 B1589 5 mg, 25 mg 1207293-36-4 BIX02189 2670 1 mg, 5 mg 1094614-85-3Cobimetinib B1689 5 mg, 25 mg 934660-93-2DEL-22379 B1680 5 mg, 25 mg 181223-80-3Doramapimod 1954 5 mg, 25 mg 285983-48-4FR180204 B1683 5 mg, 25 mg 865362-74-9GDC-0623 B1690 5 mg, 25 mg 1168091-68-6GSK-1120212 1960 1 mg, 5 mg 871700-17-3LY2228820 B1702 5 mg, 25 mg 862507-23-1

PathwayReady™ MAP Kinase Signaling Inhibitor Panel(Containing Cat. No. 1585, 1666, 1712, 1594, 1669, 1789, 1669)

K862 7 Inhibitors

212631-79-3 167869-21-8 152121-47-6 475207-59-1 109511-58-2 208260-29-1 129-56-6

MEK-162 2254 5 mg, 25 mg 606143-89-9Pamapimod B1700 1 mg, 5 mg 449811-01-2PD 169316 B1703 5 mg, 25 mg 152121-53-4EZSolution™ PD 98059 1783 5 mg 167869-21-8PD 98059 1666 5 mg 167869-21-8EZSolution™ PD-0325901, Sterile-Filtered 1990 1 ml 391210-10-9PD-0325901 1643 2 mg, 5 mg, 25 mg 391210-10-9EZSolution™ PD184352 1871 1 mg 212631-79-3PD184352 1585 1 mg, 5 mg, 25 mg 212631-79-3PD318088 B1697 1 mg, 5 mg 391210-00-7Pimasertib B1698 5 mg, 25 mg 1236699-92-5Refametinib B1889 5 mg, 25 mg 923032-37-5SB 202190 2493 5 mg, 25 mg 152121-30-7EZSolution™ SB 203580 1786 1 mg 152121-47-6SB 203580 1712 1 mg, 5 mg 152121-47-6SCH772984 B1682 5 mg, 25 mg 942183-80-4Skepinone-L B1110 1 mg, 5 mg 1221485-83-1SKF-86002 2894 5 mg, 25 mg 72873-74-6SL327 B1694 5 mg, 25 mg 305350-87-2TAK-715 B1701 5 mg, 25 mg 303162-79-0TAK-733 2460 5 mg, 25 mg 1035555-63-57,3',4'-Trihydroxyisoflavone 1886 25 mg, 100 mg 485-63-2U0126 1668 5 mg 109511-58-2VRT752271 B1679 5 mg, 25 mg 869886-67-9VX-11e B1681 5 mg, 25 mg 896720-20-0VX-702 1598 1 mg, 5 mg 745833-23-2VX-745 2812 5 mg, 25 mg 209410-46-8XMD17-109 B1685 5 mg, 25 mg 1435488-37-1XMD8-92 B1684 5 mg, 25 mg 1234480-50-210Z-Hymenialdisine 2212 250 µg, 1 mg 82005-12-7

MAP (Mitogen-Activated Protein) Kinase-MEK Inhibitors

MLK (Mixed Lineage Kinase) InhibitorsProduct Name Cat. No. Size CAS. No.GNE-3511 B1341 5 mg, 25 mg 1496581-76-0LY364947 2646 1 mg, 5 mg 396129-53-6URMC-099 9443 5 mg, 25 mg 1229582-33-5

mTOR (mammalian Target Of Rapamycin) InhibitorsProduct Name Cat. No. Size CAS. No.A-674563 B1761 5 mg, 25 mg 552325-73-2AZD-2014 9449 5 mg, 25 mg 1009298-59-2AZD-5363 B1762 5 mg, 25 mg 1143532-39-1AZD8055 2340 1 mg, 5 mg 1009298-09-2BEZ235 (NVP-BEZ235) 1626 5 mg, 25 mg 915019-65-7BI-D1870 1924 1 mg, 5 mg 501437-28-1BX-517 B1764 5 mg, 25 mg 850717-64-5BX795 B1766 5 mg, 25 mg 702675-74-9BX-912 B1765 5 mg, 25 mg 702674-56-4CCT128930 B1763 1 mg, 5 mg 885499-61-6Deforolimus 1587 5 mg, 25 mg 572924-54-0Everolimus 1917 5 mg, 25 mg 159351-69-6GDC-0084 B1656 5 mg, 25 mg 1382979-44-3GSK-2126458 1961 1 mg, 5 mg 1086062-66-9INK-128 9527 5 mg, 25 mg 1224844-38-5LY 303511 B1734 1 mg, 5 mg 154447-38-8LY3023414 B1759 5 mg, 25 mg 1386874-06-1mTOR Inhibitor, Ku-0063794 1779 1 mg, 5 mg 938440-64-3mTOR Inhibitor, WYE-132 2256 500 µg, 1 mg 1144068-46-1mTOR Inhibitor, WYE-23 2257 500 µg, 1 mg 1062169-46-3mTOR Inhibitor, WYE-28 2255 500 µg, 1 mg 1062172-60-4OSI-027 2372 5 mg, 25 mg 936890-98-1OXA-01 2695 5 mg, 25 mg 936889-68-8

DiscoveryPak™ PI 3-Kinase Inhibitor Set(Containing Cat. No. 1661, 1667, 1728, 1780, 1781)

K856 5 Inhibitors

371242-69-2 154447-36-6 371935-74-9 648450-29-7 663619-89-4

PP242 1658 1 mg 1092351-67-1Prodigiosin 2311 250 µg, 1 mg 82-89-3EZSolution™ Rapamycin 1746 5 mg 53123-88-9Rapamycin 1568 5 mg, 50 mg 53123-88-9Temsirolimus (CCI-779, Torisel) 1600 5 mg, 25 mg 162635-04-3EZSolution™ Torin 1 2353 5 mg 1222998-36-8Torin 1 2273 5 mg, 25 mg 1222998-36-8EZSolution™ Torin 2 2354 5 mg 1223001-51-1Torin 2 2274 5 mg, 25 mg 1223001-51-1Uprosertib B1760 5 mg, 25 mg 1047634-65-0VPS34 inhibitor B1754 5 mg 1383716-40-2WAY-600 B1731 1 mg, 5 mg 1062159-35-6WYE-354 B1732 5 mg, 25 mg 1062169-56-5WYE-687 B1730 5 mg, 25 mg 1062161-90-3XL388 B1733 1 mg, 5 mg 1251156-08-7

MLCK (Myosin Light Chain Kinase) InhibitorsProduct Name Cat. No. Size CAS. No.ML-7 hydrochloride B2000 10 mg, 50 mg 110448-33-4

Product Name Cat. No. Size CAS. No.TCS JNK 5a B1688 5 mg, 25 mg 312917-14-9

PDK1 (Phosphoinositide-Dependent Kinase 1) InhibitorsProduct Name Cat. No. Size CAS. No.GSK-2334470 B1555 5 mg, 25 mg 1227911-45-6OSU-03012 2295 5 mg, 25 mg 742112-33-0SGK-1 inhibitor B1757 5 mg N/A

PI 3-Kinase (Phosphoinositide 3-Kinase) InhibitorsProduct Name Cat. No. Size CAS. No.A66 B1654 5 mg, 25 mg 1166227-08-2Acalisib B1666 5 mg, 25 mg 870281-34-8

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Product Name Cat. No. Size CAS. No.Alpelisib B1271 5 mg, 25 mg 1217486-61-7 AMG319 B1663 5 mg, 25 mg 1608125-21-8APY-0201 9564 5 mg, 25 mg 1232221-74-7AS 604850 2339 1 mg, 5 mg 648449-76-7AS-041164 B1870 5 mg, 25 mg 6318-41-8AZD-6482 B1143 5 mg, 25 mg 1173900-33-8AZD-8186 B1027 5 mg, 25 mg 1627494-13-6AZD8835 B1661 5 mg, 25 mg 1620576-64-8BAG 956 2456 5 mg, 25 mg 853910-02-8BAY 80-6946 B1267 5 mg, 25 mg 1032568-63-0BEZ235 (NVP-BEZ235) 1626 5 mg, 25 mg 915019-65-7CAL-101 (GS-1101) 2613 5 mg, 25 mg 870281-82-6CH5132799 B1669 5 mg, 25 mg 1007207-67-1CNX-1351 B1673 5 mg, 25 mg 1276105-89-5CUDC-907 B1675 5 mg, 25 mg 1339928-25-4CZC24832 B1676 5 mg, 25 mg 1159824-67-5GDC-0032 9573 5 mg, 25 mg 1282512-48-4GDC-0326 B1655 5 mg, 25 mg 1282514-88-8GDC-0941 1623 1 mg, 5 mg 957054-30-7GSK-1059615 9450 5 mg, 25 mg 958852-01-2GSK-2126458 1961 1 mg, 5 mg 1086062-66-9GSK2292767 B1660 5 mg, 25 mg 1254036-66-2GSK2636771 2793 5 mg, 25 mg 1372540-25-4IC87114 1661 1 mg 371242-69-2IPI-145 2445 5 mg, 25 mg 1201438-56-3IPI-549 B1971 5 mg, 25 mg 1693758-51-8EZSolution™ LY294002 1747 5 mg 154447-36-6LY 294002 1667 5 mg, 25 mg 154447-36-6MTX-211 B1968 5 mg, 25 mg 1952236-05-3NVP-BKM120 2619 5 mg, 25 mg 944396-07-0PI-103 1728 1 mg, 5 mg 371935-74-9PI-3065 B1674 5 mg, 25 mg 955977-50-1PI3K-α Inhibitor B1869 5 mg, 25 mg 371943-05-4PI3-Kγ Inhibitor, AS-605240 1780 1 mg, 5 mg 648450-29-7

PathwayReady™ PI3-K/Akt/mTOR Signaling Inhibitor Panel(Containing Cat. No. 1708, 1626, 1667, 1779, 1728, 1780, 1658, 1568, 1781, 1707, 1670)

K857 11 Inhibitors

612847-09-3 915019-65-7 154447-36-6 938440-64-3 371935-74-9 648450-29-7 1092351-67-1 53123-88-9 663619-89-4 35943-35-2 19545-26-7

DiscoveryPak™ PI 3-Kinase Inhibitor Set(Containing Cat. No. 1661, 1667, 1728, 1780, 1781)

K856 5 Inhibitors

371242-69-2 154447-36-6 371935-74-9 648450-29-7 663619-89-4

PIK-293 B1658 5 mg, 25 mg 900185-01-5PIK-294 2614 5 mg, 25 mg 900185-02-6PIK75 B1668 5 mg, 25 mg 372196-77-5PIK-90 B1671 5 mg, 25 mg 677338-12-4PIK-93 B1670 5 mg, 25 mg 593960-11-3PX-866 1965 1 mg, 5 mg 502632-66-8SAR-260301 B1263 5 mg, 25 mg 1260612-13-2Serabelisib B1930 5 mg, 25 mg 1268454-23-4 SF-2523 B1858 1 mg, 5 mg 1174428-47-7 TG100-115 B1667 5 mg, 25 mg 677297-51-7TGR-1202 B1284 5 mg, 25 mg 1532533-67-7 TGX-115 1660 1 mg 351071-62-0TGX-221 1781 1 mg, 5 mg 663619-89-4Wortmannin, Penicillium funiculosum 1670 1 mg 19545-26-7XL-147 9401 5 mg, 25 mg 956958-53-5YM201636 2045 1 mg, 5 mg 371942-69-7

Product Name Cat. No. Size CAS. No.AZD1208 2719 1 mg, 5 mg 1204144-28-4CX-6258 2851 5 mg, 25 mg 1202916-90-2Quercetin, Dihydrate 1773 250 mg, 1 g 6151-25-3SGI-1776 2554 5 mg, 25 mg 1025065-69-3SMI-4a 2211 5 mg 327033-36-3TCS PIM-1 1 2848 10 mg, 50 mg 491871-58-0XL765 2551 5 mg, 25 mg 934493-76-2

PI3K-mTOR (Phosphoinositide 3Kinase-mTOR) InhibitorsProduct Name Cat. No. Size CAS. No.AS-252424 B1611 5 mg, 25 mg 900515-16-4BEZ235 (NVP-BEZ235) 1626 5 mg, 25 mg 915019-65-7BGT226 B1719 1 mg, 5 mg 1245537-68-1CP-466722 B1722 1 mg, 5 mg 1080622-86-1CZ415 B1726 5 mg, 25 mg 1429639-50-8GDC-0349 B1729 1 mg, 5 mg 1207360-89-1GDC-0941 Dimethanesulfonate 9618 10 mg, 50 mg 957054-33-0GDC-0980 2668 1 mg, 5 mg 1032754-93-0GNE 477 B1657 5 mg, 25 mg 1032754-81-6GNE-317 B1716 5 mg, 25 mg 1394076-92-6HS-173 B1627 5 mg, 25 mg 1276110-06-5 P529 2462 5 mg, 25 mg 914913-88-5PF-04691502 2289 5 mg, 25 mg 1013101-36-4PF-05212384 9461 10 mg, 50 mg 1197160-78-3PF-4989216 B1659 5 mg, 25 mg 1276553-09-3PKI-402 B1727 1 mg, 5 mg 1173204-81-3PKI-402 B1715 1 mg, 5 mg 173204-81-3PQR-309 B1300 5 mg, 25 mg 1225037-39-7TG100713 B1717 5 mg, 25 mg 925705-73-3VS-5584 9603 1 mg, 5 mg 1246560-33-7XL765 2551 5 mg, 25 mg 934493-76-2

PIM (Proto-oncogene proviral Integration site for Moloney murine leukemia virus) Kinase Inhibitors

PLK (Polo Like Kinase) InhibitorsProduct Name Cat. No. Size CAS. No.BI-2536 2370 5 mg, 25 mg 755038-02-9BI 6727 2222 1 mg, 5 mg 755038-65-4CFI-400945 B1287 5 mg, 25 mg 1338806-76-0GSK461364 2287 5 mg, 25 mg 929095-18-1HMN-214 B1646 5 mg, 25 mg 173529-46-9Rigosertib 9482 5 mg, 25 mg 1225497-78-8Ro3280 B1175 5 mg, 25 mg 1062243-51-9SBE13 hydrochloride 2847 10 mg, 50 mg 1052532-15-6Wortmannin, Penicillium funiculosum 1670 1 mg 19545-26-7

PKD (Protein Kinase D) InhibitorsProduct Name Cat. No. Size CAS. No.CID-2011756 2607 5 mg, 25 mg 638156-11-3CID-755673 2660 5 mg, 25 mg 521937-07-5CRT0066101 B1847 1 mg, 5 mg 1883545-60-5kb NB 142-70 9566 5 mg, 25 mg 1233533-04-4

PKG (Protein Kinase G) InhibitorsProduct Name Cat. No. Size CAS. No.H-7 dihydrochloride 9543 5 mg, 25 mg 108930-17-2KT5823 2164 50 µg, 250 µg 126643-37-6

Protein Kinase C InhibitorsProduct Name Cat. No. Size CAS. No.Bisindolylmaleimide I 1945 1 mg, 5 mg 133052-90-1

Product Name Cat. No. Size CAS. No.ZSTK474 1597 25 mg, 100 mg 475110-96-4

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Protein Tyrosine Kinase InhibitorsProduct Name Cat. No. Size CAS. No.EZSolution™ A83-01, Sterile-Filtered 1989 1 ml 909910-43-6A 83-01 1725 1 mg 909910-43-6AAL-993 2740 2 mg, 10 mg 269390-77-4ABL-001 B1949 1 mg, 5 mg 1492952-76-7ABT-869 1615 1 mg, 5 mg 796967-16-3AC710 2884 5 mg, 25 mg 1351522-04-7ACTB-1003 B2016 5 mg, 25 mg 939805-30-8AEE-788 9658 1 mg, 5 mg 497839-62-0AG 1478 1800 5 mg, 25 mg 175178-82-2AG-1296 2376 5 mg 146535-11-7Altenusin, Penicillium sp. 2146 1 mg, 5 mg 31186-12-6Altiratinib 9563 5 mg, 25 mg 1345847-93-9AMG-208 2553 5 mg, 25 mg 1002304-34-8AMG-47a 2825 5 mg, 25 mg 882663-88-9AMG-925 B1959 5 mg, 25 mg 1401033-86-0AMG-Tie2 B1612 5 mg, 25 mg 870223-96-4Amuvatinib 9458 5 mg, 25 mg 850879-09-3ANA-12 2878 10 mg, 50 mg 219766-25-3Anomalin A 2151 1 mg 548740-86-9Apatinib (Free base) B1613 5 mg, 25 mg 811803-05-1Apatinib mesylate B1608 5 mg, 25 mg 1218779-75-9ASP-3026 B1296 5 mg, 25 mg 1097917-15-1AT9283 2432 5 mg, 25 mg 896466-04-9AVL-292 (Spebrutinib) 9413 5 mg, 25 mg 1202757-89-8Axitinib (AG-013736) 1581 5 mg, 25 mg 319460-85-0AZ-5104 9441 10 mg, 50 mg 1421373-98-9AZD-3463 2371 5 mg, 25 mg 1356962-20-3AZD-3759 9609 5 mg, 25 mg 1626387-80-1AZD-4547 9403 5 mg, 25 mg 1035270-39-3AZD-8931 9659 5 mg, 25 mg 848942-61-0AZD-9291 2674 5 mg, 25 mg 1421373-65-0AZD-9291 mesylate B1899 5 mg, 25 mg 1421373-66-1Bafetinib B1172 5 mg, 25 mg 859212-16-1EZSolution™ BAY 43-9006 2031 25 mg 475207-59-1BAY 43-9006 1594 25 mg, 100 mg 475207-59-1BAY 43-9006, Free base 2142 25 mg, 100 mg 284461-73-0Bay 61-3606 Hydrochloride 1796 1 mg, 5 mg 732983-37-8BIBF1120 2167 5 mg, 25 mg 928326-83-4

Product Name Cat. No. Size CAS. No.BIBW2992 (Tovok) 1616 1 mg, 5 mg 439081-18-2BIBX-1382 9463 5 mg, 25 mg 196612-93-8BLU9931 9639 5 mg, 25 mg 1538604-68-0BLZ-945 B1651 5 mg, 25 mg 953769-46-5BMS-536924 B1908 1 mg, 5 mg 468740-43-4BMS-599626 1614 1 mg, 5 mg 873837-23-1BMS-754807 2631 1 mg, 5 mg 1001350-96-4BMS-777607 2455 5 mg, 25 mg 1025720-94-8BMX-IN-1 B1330 5 mg, 25 mg 1431525-23-3Bosutinib (SKI-606) 1584 5 mg, 25 mg 380843-75-4Brigatinib (AP26113) 9675 5 mg, 25 mg 1197953-54-0Brivanib B1325 1 mg, 5 mg 649735-46-6Brivanib Alaninate B1326 1 mg, 5 mg 649735-63-7BTK Inhibitor, CNX-774 2600 5 mg, 25 mg 1202759-32-7BTK Inhibitor, PCI-32765 2298 5 mg, 25 mg 936563-96-1Canertinib (CI-1033, PD-183805) 1617 5 mg, 50 mg 289499-45-2Carbozantinib 1935 5 mg, 25 mg 849217-68-1Cediranib (AZD2171) 1613 1 mg, 5 mg 288383-20-0CGI-1746 9647 5 mg, 25 mg 910232-84-7CH5183284 B1649 5 mg, 25 mg 1265229-25-1CH5424802 2867 5 mg, 25 mg 1256580-46-7CL-387785 2826 10 mg, 50 mg 194423-06-8CO-1686 (Rociletinib) 2794 5 mg, 25 mg 1374640-70-6CP-673451 B1337 1 mg, 5 mg 343787-29-1CP-690550 1622 5 mg, 25 mg 477600-75-2CP-724714 B1333 5 mg, 25 mg 537705-08-1Crenolanib 9679 5 mg, 25 mg 670220-88-9Crizotinib 1934 5 mg, 25 mg 877399-52-5CTx-0294885 9435 5 mg, 25 mg 1439934-41-4CUDC-101 1966 5 mg, 25 mg 1012054-59-9CZC-8004 B1868 5 mg, 25 mg 916603-07-1Damnacanthal B1094 1 mg, 5 mg 477-84-9EZSolution™ Dasatinib 2029 25 mg 302962-49-8Dasatinib (BMS-354825, Sprycel) 1586 25 mg, 100 mg 302962-49-8DDR1-IN-1 B1331 5 mg, 25 mg 1449685-96-4 Dovitinib B1614 5 mg, 25 mg 405169-16-6Dovitinib lactate B1615 5 mg, 25 mg 915769-50-5EAI-045 B1247 5 mg, 25 mg 1942114-09-1

PathwayReady™ EGFR Signaling Inhibitor Panel(Containing Cat. No. 1570, 1708, 1617, 1589, 1624, 1667, 1666, 1767, 1712, 1594, 1775, 1789, 1568)

K863 14 Inhibitors

133550-30-8 612847-09-3 289499-45-2 184475-35-2 388082-78-8 154447-36-6 167869-21-8 172889-27-9 152121-47-6 475207-59-1 501919-59-1 208260-29-1 53123-88-9 129-56-6

DiscoveryPak™ EGFR Tyrosine Kinase Inhibitor Set(Containing Cat. No. 1617, 1588, 1589, 1624, 1656)

K858 5 Inhibitors

289499-45-2 183319-69-9 184475-35-2 388082-78-8 153436-54-5

EMD-1214063 B1297 5 mg, 25 mg 1100598-32-0Emodin 1875 25 mg, 100 mg 518-82-1Ensartinib B1946 5 mg, 25 mg 1365267-27-1Entrectinib B1324 5 mg, 25 mg 1108743-60-7Erlotinib, Free Base 2048 100 mg, 1 g 183321-74-6EW-7197 B1191 1 mg, 5 mg 1352608-82-2 FIIN-2 9577 5 mg, 25 mg 1633044-56-0Foretinib 9476 5 mg, 25 mg 849217-64-7Fostamatinib Disodium 1936 1 mg, 5 mg 1025687-58-4

Product Name Cat. No. Size CAS. No.Bisindolylmaleimide I hydrochloride 1947 1 mg, 5 mg 176504-36-2Calphostin C 2611 50 µg, 100 µg 121263-19-2Cercosporin 9684 250 µg, 1 mg 35082-49-6Chelerythrine chloride 2064 5 mg 3895-92-9D-erythro-Sphingosine 2425 5 mg, 25 mg 123-78-4Enzastaurin (LY317615) 1619 1 mg, 5 mg 170364-57-5EZSolution™ Gö 6976 1785 500 µg 136194-77-9Gö 6976 1711 500 µg 136194-77-9EZSolution™ Gö 6983 9540 1 mg 133053-19-7Gö 6983 9539 1 mg, 5 mg 133053-19-7H-7 dihydrochloride 9543 5 mg, 25 mg 108930-17-2Hypericin 2526 1 mg, 5 mg 548-04-9K252a 2013 500 µg, 1 mg 99533-80-9LY-333,531 hydrochloride 2156 250 µg, 1 mg 169939-93-9PKC412 2052 1 mg, 5 mg 120685-11-2PKC-9 B1755 5 mg N/ARo 31-8220 methanesulfonate 1946 1 mg, 5 mg 138489-18-6EZSolution™ Staurosporine 1745 100 µg 62996-74-1Staurosporine 1048 100 µg, 1 mg 62996-74-1Tamoxifen citrate 1551 1 g 54965-24-1

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Product Name Cat. No. Size CAS. No.Fruquintinib B1979 5 mg, 25 mg 1194506-26-7EZSolution™ Gefitinib 2030 5 mg 184475-35-2Gefitinib 1589 5 mg, 25 mg 184475-35-2Genistein 1533 10 mg, 100 mg 446-72-0Genistin 1535 10 mg 529-59-9Gilteritinib B1294 5 mg, 25 mg 1254053-43-4 GNF-2 2470 5 mg, 25 mg 778270-11-4GNF-5 B1329 5 mg, 25 mg 778277-15-9Golvatinib 2655 5 mg, 25 mg 928037-13-2GS-9973 2669 1 mg, 5 mg 1229208-44-9GSK1904529A 2286 5 mg, 25 mg 1089283-49-7GSK2256098 B1224 5 mg, 25 mg 1224887-10-8 EZSolution™ GW2580 2549 5 mg 870483-87-7GW2580 1740 5 mg, 25 mg 870483-87-7GW-786034 1916 5 mg, 25 mg 444731-52-6GW788388 2820 10 mg, 50 mg 452342-67-5GZD824 2795 5 mg, 25 mg 1257628-77-5H3B-6527 B1647 5 mg, 25 mg 1702259-66-2Harmine 2561 50 mg, 250 mg 442-51-3Herbimycin A 2748 100 µg, 1 mg 70563-58-5Hypericin 2526 1 mg, 5 mg 548-04-9Imatinib Mesylate (CGP-57148B, STI-571) 1625 100 mg, 1 g 220127-57-1Imatinib, Free base 2141 100 mg, 1 g 152459-95-5IPI-549 B1971 5 mg, 25 mg 1693758-51-8ITD-1 2879 10 mg, 50 mg 1099644-42-4JAK Inhibitor, Pyridone 6 2534 500 µg, 1 mg 457081-03-7

PathwayReady™ JAK/STAT Signaling Inhibitor Panel(Containing Cat. No. 1570, 1622, 1805, 1792, 1775, 1809, 1887)

K864 8 Inhibitors

133550-30-8 477600-75-2 111358-88-4 1260247-42-4 501919-59-1 857064-38-1 2062-78-4

JNJ-10198409 B1078 5 mg, 25 mg 627518-40-5Ki 8751 2677 5 mg, 25 mg 228559-41-9KRN-633 2839 5 mg, 25 mg 286370-15-8KW-2449 hydrochloride B1208 5 mg, 25 mg 1000669-72-6Lapatinib Ditosylate (Tykerb, Tyverb, GW-572016) 1624 25 mg, 100 mg 388082-78-8

EZSolution™ Lapatinib Ditosylate 2807 10 mg 388082-78-8Lapatinib, Free base 2138 25 mg, 100 mg 231277-92-2Lenvatinib B1157 5 mg, 25 mg 417716-92-8LFM-A13 2414 5 mg, 25 mg 244240-24-2Linsitinib, Free base 2294 5 mg, 25 mg 867160-71-2LY-2109761 9605 5 mg, 25 mg 700874-71-1LY-2157299 9475 5 mg, 25 mg 700874-72-2LY-2874455 9532 5 mg, 25 mg 1254473-64-7LY364947 2646 1 mg, 5 mg 396129-53-6Masitinib 2007 5 mg, 25 mg 790299-79-5meta-Topolin B1298 50 mg, 250 mg 75737-38-1MK-1775 2373 5 mg, 25 mg 955365-80-7Motesanib 2022 5 mg, 25 mg 453562-69-1MTX-211 B1968 5 mg, 25 mg 1952236-05-3Naquotinib B1317 5 mg, 25 mg 448232-80-1 Neratinib 2023 5 mg, 25 mg 698387-09-6Nilotinib 1750 25 mg, 100 mg 641571-10-0NVP-AEW541 B1335 5 mg, 25 mg 475489-16-8NVP-BGJ398 2855 5 mg, 25 mg 872511-34-7NVP-BHG712 2464 5 mg, 25 mg 940310-85-0NVP-TAE684 1683 5 mg 761439-42-3Olmutinib B1218 5 mg, 25 mg 1353550-13-6PD 153035 Hydrochloride 1656 2 mg 153436-54-5PD 173074 1675 1 mg 219580-11-7

Product Name Cat. No. Size CAS. No.Pelitinib (EKB-569) 2676 5 mg, 25 mg 257933-82-7PF-04554878 2888 5 mg, 25 mg 1073154-85-4PF-06463922 B1169 10 mg, 50 mg 1454846-35-5PF299804 2678 5 mg, 25 mg 1110813-31-4PF-431396 2844 5 mg, 25 mg 717906-29-1PF-573228 2819 10 mg, 50 mg 869288-64-2Piceatannol 2072 5 mg, 25 mg 10083-24-6Picropodophyllotoxin 2765 1 mg, 5 mg 477-47-4PLX-3397 9617 10 mg, 50 mg 1029044-16-3PND-1186 2823 5 mg, 25 mg 1061353-68-1Ponatinib 2712 10 mg, 50 mg 943319-70-8Poziotinib 9519 10 mg, 50 mg 1092364-38-9PP1 1927 1 mg, 5 mg 172889-26-8PP2 1767 1 mg, 5 mg 172889-27-9PP3 1797 10 mg, 50 mg 5334-30-5Quizartinib 2008 1 mg, 5 mg 950769-58-1R428 9591 5 mg, 25 mg 1037624-75-1Radotinib 9613 10 mg, 50 mg 926037-48-1Rebastinib (DCC-2036) B1619 5 mg, 25 mg 1020172-07-9

DiscoveryPak™ Receptor Tyrosine Kinase (RTK) Inhibitor Set(Containing Cat. No. 1581, 1617, 1589, 1740, 1624, 1675, 1674, 1611)

K859 8 Inhibitors

319460-85-0 289499-45-2 184475-35-2 870483-87-7 388082-78-8 219580-11-7 301836-41-9 341031-54-7

Regorafenib 2891 5 mg, 25 mg 755037-03-7Regorafenib monohydrate B1621 5 mg, 25 mg 1019206-88-2EZSolution™ RepSox 2641 5 mg 446859-33-2RN486 9678 1 mg, 5 mg 1242156-23-5Saracatinib (AZD0530) 1582 5 mg, 25 mg 379231-04-6SB1518 (Pacritinib) 2450 1 mg, 5 mg 937272-79-2EZSolution™ SB-431542 1872 1 mg 301836-41-9EZSolution™ SB-431542, Sterile-Filtered 1992 1 ml 301836-41-9SB-431542 1674 1 mg, 5 mg 301836-41-9EZSolution™ SB-525334 2881 5 mg 356559-20-1SB-525334 2880 5 mg, 25 mg 356559-20-1SD208 2885 5 mg, 25 mg 627536-09-8SSR128129E B1165 5 mg, 25 mg 848318-25-2STK-321130 B2006 5 mg, 25 mg 923562-23-6 SU 11274 1938 5 mg, 25 mg 658084-23-2SU 1498 1836 1 mg, 5 mg 168835-82-3SU 16f B1081 5 mg, 25 mg 251356-45-3SU 6668 1931 5 mg, 25 mg 252916-29-3SU-5214 B1307 5 mg, 25 mg 186611-04-1EZSolution™ SU-5402 2017 500 µg 215543-92-3SU-5402 1645 500 µg, 1 mg 215543-92-3EZSolution™ SU-5416 9492 5 mg 204005-46-9SU-5416 9491 5 mg, 25 mg 204005-46-9SU-5614 9643 5 mg, 25 mg 1055412-47-9EZSolution™ Sunitinib Malate 1804 25 mg 341031-54-7Sunitinib Malate (Sutent) 1611 25 mg, 100 mg, 1 g 341031-54-7Sunitinib, Free base 2097 25 mg, 100 mg, 1 g 557795-19-4Syk Inhibitor 1983 1 mg, 5 mg 622387-85-3TAE-226 9436 5 mg, 25 mg 761437-28-9TAK 165 1951 5 mg, 25 mg 366017-09-6Tandutinib 2024 5 mg, 25 mg 387867-13-2Tie2 Kinase Inhibitor B1338 5 mg, 25 mg 948557-43-5Tivantinib B1546 5 mg, 25 mg 905854-02-6Tivozanib B1545 5 mg, 25 mg 475108-18-0 Toceranib B1542 5 mg, 25 mg 356068-94-5TP-0903 9590 5 mg, 25 mg 1341200-45-0

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Product Name Cat. No. Size CAS. No.TX1-85-1 B1313 5 mg, 25 mg 1603845-32-4Tyrphostin AG 1295 1571 5 mg 71897-07-9Tyrphostin AG 490 1570 5 mg 133550-30-8UNC-2025 B1262 5 mg, 25 mg 1429881-91-3UNC2881 2837 5 mg, 25 mg 1493764-08-1Vandetanib 1751 25 mg, 100 mg 443913-73-3Varlitinib 2656 5 mg, 25 mg 845272-21-1Vatalanib Dihydrochloride 2025 5 mg, 25 mg 212141-51-0Vatalanib, Free Base 2026 5 mg, 25 mg 212141-54-3WH-4-023 2827 10 mg, 50 mg 837422-57-8WHI-P131 1853 5 mg, 25 mg 202475-60-3EZSolution™ WP1066 2546 5 mg 857064-38-1WZ4002 2461 5 mg, 25 mg 1213269-23-8XL019 2609 5 mg, 25 mg 945755-56-6XL-228 2632 1 mg, 5 mg 898280-07-4

Raf Kinase InhibitorsProduct Name Cat. No. Size CAS. No.AZ 628 B1713 5 mg, 25 mg 878739-06-1B-Raf Inhibitor 1 2599 5 mg, 25 mg 1093100-40-3CCT196969 B1752 5 mg 1163719-56-9CCT241161 B1753 5 mg 1163719-91-2CEP-32496 9615 5 mg, 25 mg 1188910-76-0DP-4978 B1288 5 mg, 25 mg 1454682-72-4GDC0879 B1340 5 mg, 25 mg 905281-76-7GDC0994 B1629 5 mg, 25 mg 1453848-26-4Gossypin 2374 50 mg, 250 mg 652-78-8GSK-2118436 mesylate 2800 5 mg, 25 mg 1195768-06-9GW-5074 2412 5 mg, 25 mg 220904-83-6L-779450 B1709 5 mg, 25 mg 303727-31-3MLN2480 B1706 5 mg, 25 mg 1096708-71-2

PLX-4032 2235 5 mg, 25 mg 1029872-54-5, 918504-65-1

PLX-4720 2813 5 mg, 25 mg 918505-84-7PLX-7904 B1249 5 mg, 25 mg 1393465-84-3 RAF265 2856 5 mg, 25 mg 927880-90-8RO5126766 B1705 5 mg, 25 mg 946128-88-7SB-590885 B1708 5 mg, 25 mg 405554-55-4TAK-632 2473 5 mg, 25 mg 1228591-30-7ZM 336372 1789 1 mg, 5 mg 208260-29-1

ROCK (Rho-associated protein Kinase) InhibitorsProduct Name Cat. No. Size CAS. No.Fasudil, Monohydrochloride 1787 10 mg, 50 mg 105628-07-7GSK-269962 9654 5 mg, 25 mg 850664-21-0EZSolution™ GSK429286A 2640 1 mg 864082-47-3GSK429286A 2637 1 mg, 5 mg 864082-47-3Hydroxyfasudil Hydrochloride B1559 5 mg, 25 mg 155558-32-0RKI-1313 B1092 5 mg, 25 mg 1342276-76-9RKI-1447 2472 5 mg, 25 mg 1342278-01-6ROCK Inhibitor (Rockout) 2342 5 mg, 25 mg 7272-84-6(S)-H-1152 dihydrochloride B1106 1 mg, 5 mg 451462-58-1EZSolution™ Thiazovivin 1736 1 mg 1226056-71-8EZSolution™ Thiazovivin, Sterile-Filtered 1993 1 ml 1226056-71-8Thiazovivin 1681 1 mg, 5 mg 1226056-71-8EZSolution™ Y-27632 1784 5 mg 146986-50-7EZSolution™ Y-27632, Sterile-Filtered 1994 1 ml 146986-50-7Y-27632, dihydrochloride 1596 1 mg, 5 mg, 50 mg 146986-50-7ZINC00881524 B1840 5 mg, 25 mg 557782-81-7

Product Name Cat. No. Size CAS. No.SRPIN340 2458 5 mg, 25 mg 218156-96-8

SRPK (Serine-arginine-Rich Protein Kinase) Inhibitors

Syk (Spleen Tyrosine Kinase) InhibitorsProduct Name Cat. No. Size CAS. No.Bay 61-3606 Hydrochloride 1796 1 mg, 5 mg 732983-37-8Cedrulatinib 2803 5 mg, 25 mg 1198300-79-6Fostamatinib Disodium 1936 1 mg, 5 mg 1025687-58-4GS-9973 2669 1 mg, 5 mg 1229208-44-9

P505-15 9583 5 mg, 25 mg 1370261-96-3, 1370261-97-4

Piceatannol 2072 5 mg, 25 mg 10083-24-6PRT-060318 B1911 5 mg, 25 mg 1194961-19-7Syk Inhibitor 1983 1 mg, 5 mg 622387-85-3SYK Inhibitor, R406 9682 5 mg, 25 mg 841290-80-0

Other Protein Kinase InhibitorsProduct Name Cat. No. Size CAS. No.APY29 2591 5 mg, 25 mg 1216665-49-4AS-2444697 Hydrochloride B1585 5 mg, 25 mg 1287665-60-4AT-13148 B1144 5 mg, 25 mg 1056901-62-2AZ-3146 B1145 5 mg, 25 mg 1124329-14-1BAY-1217389 B1295 5 mg, 25 mg 1554458-53-5 Cercosporamide 9662 100 µg, 500 µg 131436-22-1CGP-57380 9661 1 mg, 5 mg 522629-08-9Compound 43 B1758 5 mg N/ACPD5 B1750 5 mg N/ACZC-54252 hydrochloride 9567 10 mg, 50 mg 1191911-27-9FRAX597 B1890 1 mg, 5 mg 1286739-19-2GNE-7915 B1342 5 mg, 50 mg 1351761-44-8GNF-5837 B1339 5 mg, 25 mg 1033769-28-6GNF-7 B1139 5 mg, 25 mg 839706-07-9GSK180736A B1628 5 mg, 25 mg 817194-38-0GSK2578215A 2845 5 mg, 25 mg 1285515-21-0GSK-2606414 9467 5 mg, 25 mg 1337531-36-8GSK-2656157 9466 5 mg, 25 mg 1337532-29-2GSK-583 B1301 5 mg, 25 mg 1346547-00-9 EZSolution™ GSK'872 B1501 5 mg 1346546-69-7GSK'872 2673 5 mg, 25 mg 1346546-69-7GW-441756 B1147 5 mg, 25 mg 504433-23-2HG-10-012-01 2604 5 mg, 25 mg 1351758-81-0HG-9-91-01 B1849 1 mg, 5 mg 1456858-58-4HTH-01-015 2887 5 mg, 25 mg 1613724-42-7IPA-3 2647 5 mg, 25 mg 42521-82-4IRAK-1/4 Inhibitor 9578 5 mg, 25 mg 509093-47-4Kobe0065 B1714 5 mg, 25 mg 436133-68-5Kobe2602 B1710 5 mg, 25 mg 454453-49-7LDK-378 B1928 5 mg, 25 mg 1032900-25-6LIMKi 3 B1095 5 mg, 25 mg 1338247-35-0LJH685 B1232 5 mg, 25 mg 1627710-50-2LJI-308 B1233 5 mg, 25 mg 1627709-94-7LY-2584702 9445 5 mg, 25 mg 1082949-68-5MPI-0479605 9589 5 mg, 25 mg 1246529-32-7Mps1-IN-1 B1603 5 mg, 25 mg 1125593-20-5NQDI-1 9645 10 mg, 50 mg 175026-96-7OTS-964 B1964 5 mg, 25 mg 1338545-07-5OTSSP167 B1065 5 mg, 25 mg 1431697-89-0PF-06447475 9447 5 mg, 25 mg 1527473-33-1PF-06650833 B1558 5 mg, 25 mg 1817626-54-2 PF-4708671 9460 10 mg, 50 mg 1255517-76-0SBI-0206965 9580 5 mg, 25 mg N/ASelonsertib B1312 5 mg, 25 mg 1448428-04-3SL0101 B1895 5 mg, 25 mg 77307-50-7SR7826 B1096 1 mg, 5 mg 1219728-20-7T5601640 B1097 1 mg, 5 mg 924473-59-6TGR5-Receptor-Agonist B1635 5 mg, 25 mg 1197300-24-5

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PTEN (Phosphatase & Tensin Homolog) InhibitorsProduct Name Cat. No. Size CAS. No.bpV(phen) 1793 5 mg 42494-73-5bpV(pic) 1794 5 mg 148556-27-8SF1670 2774 1 mg, 5 mg 345630-40-2VO-OHpic, Trihydrate 1801 5 mg, 25 mg 476310-60-8

Rac1 InhibitorsProduct Name Cat. No. Size CAS. No.EHop-016 9595 5 mg, 25 mg 1380432-32-5NSC 23766 1941 1 mg, 5 mg 733767-34-5

Renin InhibitorsProduct Name Cat. No. Size CAS. No.Rat renin inhibitor peptide 2557 1 mg, 5 mg N/ARenin Inhibitor 2084 5 mg, 25 mg 173334-58-2

SAH (S-Adenosyl-l-Homocysteine) hydrolase InhibitorsProduct Name Cat. No. Size CAS. No.3-Deazaadenosine 2771 1 mg, 5 mg 6736-58-9EZSolution™ 3-Deazaneplanocin A 2409 1 mg 102052-95-93-Deazaneplanocin A 2060 250 µg, 1 mg 102052-95-93-Deazaneplanocin A hydrochloride 2444 250 µg, 1 mg 120964-45-6

SCD1 (Stearoyl-CoA Desaturase 1) InhibitorsProduct Name Cat. No. Size CAS. No.MF-438 B1178 5 mg, 25 mg 921605-87-0PluriSIn 1 2471 10 mg, 50 mg 91396-88-2EZSolution™ SCD1 Inhibitor 2548 1 mg N/ASCD1 Inhibitor 1716 1 mg, 5 mg 103229-33-6

Secretase InhibitorsProduct Name Cat. No. Size CAS. No.Beta-Secretase Inhibitor I 7501 1 mg N/ABeta-Secretase Inhibitor II 7502 1 mg N/ABMS-299897 9606 5 mg, 25 mg 290315-45-6BMS-708163 B1622 5 mg, 25 mg 1146699-66-2Compound 34 1898 200 µg, 1 mg N/ACompound E 1949 250 µg, 1 mg 209986-17-4Compound W 2208 50 mg, 250 mg 173550-33-9EZSolution™ DAPT 2663 5 mg 208255-80-5DAPT 1855 5 mg 208255-80-5DBZ 1649 1 mg, 5 mg 209984-56-5IMR-1 B1131 5 mg, 25 mg 310456-65-6L-685, 458 1713 250 µg 292632-98-5LY-411575 2648 1 mg, 5 mg 209984-57-6LY2811376 B1606 5 mg, 25 mg 1194044-20-6LY2886721 2299 5 mg, 25 mg 1262036-50-9MK-0752 B1980 1 mg, 5 mg 471905-41-6MK-8931 B1315 1 mg, 5 mg 1286770-55-5RO4929097 2011 1 mg, 5 mg 847925-91-1Semagacestat 2430 1 mg, 5 mg 425386-60-3

SGLT-2 (Sodium Glucose Co-Transporter 2) InhibitorsProduct Name Cat. No. Size CAS. No.Bexgliflozin (EGT1442) B1929 1 mg, 5 mg 1118567-05-7Canagliflogin B1597 10 mg, 50 mg 842133-18-0 Dapagliflozin 9452 10 mg, 50 mg 461432-26-8Empagliflozin 2877 10 mg, 50 mg 864070-44-0Ertugliflozin B1896 5 mg, 25 mg 1210344-57-2Ipragliflozin B1926 5 mg, 25 mg 761423-87-4LX-4211 9623 5 mg, 25 mg 1018899-04-1

SIRT (Sirtuin) InhibitorsProduct Name Cat. No. Size CAS. No.Cambinol 1653 10 mg 14513-15-64-Hydroxynonenal 2083 1 mg, 5 mg 75899-68-2Hyperforin. DCHA 2153 500 µg, 1 mg 238074-03-8Inauhzin 9555 5 mg, 25 mg 309271-94-1Salermide 1873 5 mg, 25 mg 1105698-15-4SIRT1 Inhibitor, EX-527 1652 10 mg 49843-98-3SIRT2 Inhibitor 1857 5 mg, 25 mg 420831-40-9SIRT2 Inhibitor, AGK2 1651 10 mg 304896-28-4SIRT2 Inhibitor, B2 2085 5 mg 115687-05-3Sirtinol 2062 1 mg, 5 mg 410536-97-9Suramin Hexasodium Salt 1874 50 mg, 250 mg 129-46-4Tenovin-1 9400 5 mg, 25 mg 380315-80-0

Smad InhibitorsProduct Name Cat. No. Size CAS. No.Smad3 Inhibitor, SIS3 2227 1 mg, 5 mg 521984-48-5

SK (Sphingosine Kinase) InhibitorsProduct Name Cat. No. Size CAS. No.ABC294640 B1231 5 mg, 25 mg 915385-81-8Sphingosine Kinase Inhibitor, SKI-I 2046 5 mg, 25 mg 306301-68-8Sphingosine Kinase Inhibitor, SKI-II 2047 5 mg, 25 mg 312636-16-1

SREBP (Sterol Regulatory Element-Binding Proteins) Activation InhibitorsProduct Name Cat. No. Size CAS. No.Betulin 1942 5 mg, 25 mg 473-98-3Fatostatin 2035 5 mg, 25 mg 298197-04-3Xanthohumol 2258 5 mg, 25 mg 6754-58-1

Sodium Channel ModulatorsProduct Name Cat. No. Size CAS. No.Aconitine 2423 10 mg, 50 mg 302-27-2Ambroxol hydrochloride 9688 100 mg, 500 mg 23828-92-4Veratridine 2422 5 mg, 25 mg 71-62-5

Stat InhibitorsProduct Name Cat. No. Size CAS. No.Cryptotanshinone 2429 5 mg, 25 mg 35825-57-1Galiellactone 2623 100 µg, 500 µg 133613-71-5

PathwayReady™ JAK/STAT Signaling Inhibitor Panel(Containing Cat. No. 1570, 1622, 1805, 1732, 1887, 1775, 1778, 1809)

K864 8 Inhibitors

133550-30-8477600-75-2111358-88-426305-03-32062-78-4501919-59-1N/A857064-38-1

Lestaurtinib 1805 500 µg, 1 mg 111358-88-4LLL12 1792 5 mg, 25 mg N/AMS-1020 1911 1 mg 1255516-86-9Niclosamide 1826 100 mg, 500 mg 50-65-7Pimozide 1887 50 mg, 250 mg 2062-78-4Resveratrol 1758 100 mg, 500 mg 501-36-0SH-4-54 B1637 5 mg, 25 mg 1456632-40-8STA-21 2626 250 µg, 1 mg 28882-53-3Stat3 Activation Inhibitor, SPI 1813 2 mg N/AEZSolution™ Stat3 Inhibitor I, S3I-201 2541 5 mg 501919-59-1Stat3 Inhibitor I, S3I-201 1775 5 mg, 25 mg 501919-59-1

Product Name Cat. No. Size CAS. No.

DiscoveryPak™ SGLT-2 Inhibitors Set(Containing Cat. No. B1597, 9452, 2877, B1896)

S235 4 Inhibitors

842133-18-0461432-26-8864070-44-01210344-57-2

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SUMOYlation InhibitorsProduct Name Cat. No. Size CAS. No.Anacardic Acid 1849 5 mg, 25 mg 16611-84-0Ginkgolic acid C15:1 9523 5 mg, 25 mg 22910-60-7

TACE InhibitorsProduct Name Cat. No. Size CAS. No.TAPI-0 2067 1 mg 143457-40-3TAPI-1 2068 1 mg 171235-71-5TAPI-2 2069 1 mg 187034-31-7

Tankyrase InhibitorsProduct Name Cat. No. Size CAS. No.AZ-6102 B1200 5 mg, 25 mg 1645286-75-4JW55 2612 5 mg, 25 mg 664993-53-7MN64 B1127 10 mg, 50 mg 92831-11-3XAV939 1727 1 mg 284028-89-3

Thioredoxin inhibitorsProduct Name Cat. No. Size CAS. No.Auranofin 2219 10 mg, 50 mg 34031-32-8PX 12 2217 5 mg, 25 mg 141400-58-0

Topoisomerase InhibitorsProduct Name Cat. No. Size CAS. No.Camptothecin 1039 1 ml, 50 mg, 500 mg 7689-03-4Doxorubicin.HCl 1527 5 mg 25316-40-9Ellipticine 9579 5 mg, 25 mg 519-23-3Epirubicin Hydrochloride 1753 5 mg, 25 mg 56390-09-1Etoposide 1043 10 µl, 25 mg, 250 mg 33419-42-0Etoposide phosphate 2896 10 mg, 50 mg 117091-64-210-Hydroxycamptothecin B1995 25 mg, 100 mg 19685-09-7Irinotecan Hydrochloride 1752 50 mg, 250 mg 100286-90-6β-Lapachone 2262 5 mg, 25 mg 4707-32-8Mitoxantrone 1885 50 mg, 250 mg 65271-80-9Pixantrone maleate 1958 5 mg, 25 mg 144675-97-8

Podophyllotoxin 2767 50 mg, 250 mg 518-28-5, 4354-76-1

SW-044248 B1135 5 mg, 25 mg 522650-83-5TAS-103 B1841 5 mg, 25 mg 174634-08-3Topotecan hydrochloride B2050 10 mg, 50 mg 119413-54-6

Ubiquitin Activating Enzyme E1 InhibitorProduct Name Cat. No. Size CAS. No.PYR-41 1925 5 mg, 25 mg 418805-02-4

Ubiquitin Ligase (E3) InhibitorsProduct Name Cat. No. Size CAS. No.NSC 146109 hydrochloride 1907 5 mg 59474-01-0NSC 66811 2009 5 mg 6964-62-1NSC-687852 2021 5 mg, 25 mg 1009817-63-3PRT4165 B1054 5 mg, 25 mg 31083-55-3SKPin C1 2343 5 mg, 25 mg 432001-69-9SMER-3 2514 5 mg, 25 mg 67200-34-4(±)-Thalidomide 2020 10 mg, 50 mg 50-35-1TCID 2204 5 mg, 25 mg 30675-13-9

Ubiquitin Proteasome Pathway InhibitorsProduct Name Cat. No. Size CAS. No.Calpain Inhibitor I, ALLN 1834 5 mg, 25 mg 110044-82-1

Product Name Cat. No. Size CAS. No.Stat3 Peptide Inhibitor, Cell-Permeable 1778 1 mg, 5 mg N/AStat5 Inhibitor 9484 1 mg, 5 mg 285986-31-4Stattic 2625 5 mg, 25 mg 19983-44-9

Product Name Cat. No. Size CAS. No.Calpain Inhibitor II, ALLM 1835 5 mg, 25 mg 136632-32-1Carfilzomib 2385 5 mg, 25 mg 868540-17-4Celastrol 1940 5 mg, 25 mg 34157-83-0CEP-18770 2433 5 mg, 25 mg 847499-27-8Clasto-Lactacystin β-lactone 1710 100 µg 154226-60-5Clioquinol 2454 1 g, 5 g 130-26-7DBeQ 1858 5 mg, 25 mg 177355-84-9DUB Inhibitor, NSC-632839 2570 5 mg, 25 mg 157654-67-6Eeyarestatin I 9602 5 mg, 25 mg 412960-54-4(-)-Epigallocatechin gallate 1841 50 mg 989-51-5Fenbendazole 2157 100 mg, 500 mg 43210-67-9Ginkgolic acid C15:1 9523 5 mg, 25 mg 22910-60-7HBX-41108 9608 5 mg, 25 mg 924296-39-9Lactacystin (Synthetic) 1709 200 µg 133343-34-7LDN-57444 2016 5 mg, 25 mg 668467-91-2MDBN 2033 10 mg, 50 mg 1485-00-3MG-115 1831 1 mg, 5 mg 133407-86-0MG-132 1703 5 mg, 25 mg 133407-82-6MLN-4924 2566 500 µg 905579-51-3NMS-873 9600 5 mg, 25 mg 1418013-75-8NSC-687852 2021 5 mg, 25 mg 1009817-63-3NSC-697923 B1091 5 mg, 25 mg 343351-67-7ONX-0914 2555 5 mg, 25 mg 960374-59-8Oprozomib 2386 5 mg, 25 mg 935888-69-0P5091 2277 5 mg, 25 mg 882257-11-6PS-341 1846 1 mg, 5 mg 179324-69-7PYR-41 1925 5 mg, 25 mg 418805-02-4SMER-3 2514 5 mg, 25 mg 67200-34-4Spautin-1 2037 5 mg, 25 mg 1262888-28-7(±)-Thalidomide 2020 10 mg, 50 mg 50-35-1TAME Hydrochloride 2050 100 mg, 500 mg, 1 g 1784-03-8TCID 2204 5 mg, 25 mg 30675-13-9USP14 Inhibitor, IU1 1845 5 mg, 25 mg 314245-33-5VR23 B1515 5 mg, 25 mg 1624602-30-7WP-1130 2014 5 mg, 25 mg 856243-80-6

VCP-p97 (Valosin-Containing Protein-p97) InhibitorsProduct Name Cat. No. Size CAS. No.CB5083 B1032 5 mg, 25 mg 1542705-92-9DBeQ 1858 5 mg, 25 mg 177355-84-9Eeyarestatin I 9602 5 mg, 25 mg 412960-54-4MDBN 2033 10 mg, 50 mg 1485-00-3ML-240 B1142 5 mg, 25 mg 1346527-98-7NMS-873 9600 5 mg, 25 mg 1418013-75-8

Wnt (Wingless Phenotype in Drosophila) Signaling InhibitorsProduct Name Cat. No. Size CAS. No.CRT Inhibitor, iCRT5 1896 5 mg, 25 mg N/AFH535 2657 5 mg, 25 mg 108409-83-2ICG-001 2275 5 mg, 25 mg 847591-62-2IQ-1 1663 1 mg 331001-62-8IWP-2 1962 5 mg, 25 mg 686770-61-6IWP-3 2349 1 mg, 5 mg 687561-60-0IWP-4 2650 1 mg, 5 mg 686772-17-8JW55 2612 5 mg, 25 mg 664993-53-7KY02111 2264 5 mg, 25 mg 1118807-13-8LGK974 2645 1 mg, 5 mg 1243244-14-5PNU-74654 B1837 5 mg, 25 mg 113906-27-7QS11 1680 5 mg 944328-88-5

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Cancer Stem cell InhibitorsOther Inhibitors

Product Name Cat. No. Size CAS. No.A37 B1577 5 mg, 25 mg 896795-60-1BRD7116 B1578 5 mg, 25 mg 329059-55-4Cancer Cell Stemness Inhibitor I 2476 5 mg, 25 mg 83280-65-3Emetine dihydrochloride 1970 50 mg, 250 mg 316-42-7Galiellactone 2623 100 µg, 500 µg 133613-71-5GDC-0084 B1656 5 mg, 25 mg 1382979-44-3GNE 477 B1657 5 mg, 25 mg 1032754-81-6ITE B1579 5 mg, 25 mg 448906-42-1ML239 2696 5 mg, 25 mg 1378872-36-6ML243 2515 5 mg, 25 mg 1426576-80-8PF-4989216 B1659 5 mg, 25 mg 1276553-09-3PND-1186 2823 5 mg, 25 mg 1061353-68-1Pyrvinium Pamaote B1593 5 mg, 25 mg 3546-41-6Salinomycin Sodium B1584 25 mg, 100 mg 55721-31-8SC-26196 B1580 5 mg, 25 mg 218136-59-5Thioridazine Hydrochloride B1581 1 g, 5 g 130-61-0TY-52156 B1582 5 mg, 25 mg 934369-14-9Verteporfin B1583 5 mg, 25 mg 129497-78-5VS-5584 9603 1 mg, 5 mg 1246560-33-7

Protein Synthesis InhibitorsProduct Name Cat. No. Size CAS. No.Anisomycin 1549 10 mg 22862-76-6Aurodox 2317 1 mg 12704-90-4(-)-6-Azauridine 2’, 3’,5’-triacetate B1025 50 mg, 250 mg 2169-64-46-Azauridine B1024 100 mg, 500 mg 54-25-1Blasticidin S Hydrochloride 1859 25 mg, 100 mg 3513-03-9Clindamycin hydrochloride 2627 10 mg, 50 mg 21462-39-5Cycloheximide 1041 1 ml, 1 g, 5 g 66-81-9Emetine dihydrochloride 1970 50 mg, 250 mg 316-42-7Erythromycin 9619 5 g , 25 g 114-07-8G418 Sulfate 1557 1 g, 5 g, 25 g 108321-42-2Kanamycin Sulfate, USP 2498 5 g, 25 g 25389-94-0Kirromycin B1236 1 mg, 5 mg 50935-71-2Neomycin sulfate 9620 25 g, 100 g 1405-10-3Nourseothricin sulfate 2882 50 mg, 100 mg, 500 mg, 1 g 96736-11-7Paromomycin Sulfate B1528 1 g, 5 g 1263-89-4EZSolution™ Puromycin Dihydrochloride 1861 100 mg 58-58-2

Puromycin Dihydrochloride 1860 25 mg, 100 mg, 250 mg, 500 mg, 1 g 58-58-2

Roxithromycin 9621 1 g, 5 g 80214-83-1Streptomycin Sulfate 2517 50 g, 100 g, 500 g 3810-74-0Tetracycline Hydrochloride B1535 10 g, 50 g 64-75-5Thiostrepton 9677 50 mg, 250 mg 1393-48-2Tildipirosin 9673 1 mg, 5 mg 328898-40-4

Protein Transport InhibitorsProduct Name Cat. No. Size CAS. No.EZCell™ Protein Transport Inhibitor Cocktail (500X)(Containing Cat. No. 1560, 1808)

K932 500 µl 20350-15-628636-21-7

Other InhibitorsProduct Name Cat. No. Size CAS. No.A-803467 2559 5 mg, 25 mg 944261-74-9Acivicin B1028 1 mg, 5 mg 42228-92-2

Product Name Cat. No. Size CAS. No.WIKI-4 B1630 5 mg, 25 mg 838818-26-1EZSolution™ Wnt Antagonist, C59 9493 1 mg 1243243-89-1Wnt Antagonist, C59 2063 1 mg, 5 mg 1243243-89-1XAV939 1727 1 mg 284028-89-3

Product Name Cat. No. Size CAS. No.Agistatin B B1021 1 mg, 5 mg 144096-46-8Agistatin D B1022 1 mg, 5 mg 144096-47-9Agistatin E B1023 1 mg, 5 mg 144096-48-0AHU-377 9520 5 mg, 25 mg 149709-62-6AM-095 9581 5 mg, 25 mg 1228690-36-5AM-095 Sodium B1225 5 mg, 25 mg 1345614-59-6Amidepsine A, Humcola sp. 2147 500 µg, 1 mg 169181-28-6Amidepsine D, Humcola sp. 2148 500 µg, 1 mg 79786-34-8Andrastin A, Aspergillus fumigatus 2149 250 µg, 1 mg 174232-42-9Apilimod mesylate B1129 5 mg, 25 mg 870087-36-8 Apixaban B1855 10 mg, 50 mg 503612-47-3Aprepitant 9531 10 mg, 50 mg 170729-80-3Aripiprazole B1186 10 mg, 50 mg 129722-12-9AT 56 2592 5 mg, 25 mg 162640-98-4AT-406 B1829 5 mg, 25 mg 1071992-99-8Atazanavir B1901 5 mg, 25 mg 198904-31-3Atglistatin B1864 5 mg, 25 mg 1469924-27-3Aurantimycin A 9692 1 mg, 5 mg 162478-50-4Avibactam sodium 9569 5 mg, 25 mg 1192491-61-4AX-024 hydrochloride B2013 5 mg, 25 mg 1704801-24-0AZD-1283 2838 5 mg, 25 mg 919351-41-0AZD-1981 9611 5 mg, 25 mg 802904-66-1AZD-4635 B2012 5 mg, 25 mg 1321514-06-0AZD-5069 B2053 5 mg, 25 mg 878385-84-3Azeliragon B1152 5 mg, 25 mg 603148-36-3BAY 57-1293 2556 5 mg, 25 mg 348086-71-5BD 1047 dihydrobromide B1069 10 mg, 50 mg 138356-21-5Bedaquiline 9598 5 mg, 25 mg 843663-66-1Bempedoic acid B1913 5 mg, 25 mg 738606-46-7 Betulin 1942 5 mg, 25 mg 473-98-3Birinapant 2597 1 mg, 5 mg 1260251-31-7BMS-303141 2821 10 mg, 50 mg 943962-47-8Bongkrekic Acid, Triammonium Salt 1820 100 µg 11076-19-0Bosentan B1857 1 mg, 5 mg 147536-97-8BQ-123 Sodium Salt B1552 1 mg, 5 mg 136553-81-6BQ-610 B1553 1 mg, 5 mg 141595-53-1BQ-788 Sodium Salt B1554 500 μg, 1 mg 156161-89-6BTZ043 B1206 5 mg, 25 mg 1161233-85-7BV6 B1332 5 mg, 25 mg 1001600-56-1680C91 2292 5 mg, 25 mg 163239-22-3Capsaicin 2521 50 mg, 250 mg 404-86-4Catharanthine 1749 100 mg, 1 g 2468-21-5CB-839 B1179 5 mg, 25 mg 1439399-58-2CBL0137 B2036 5 mg, 25 mg 1197996-80-7CCF-642 B2009 5 mg, 25 mg 346640-08-29434 5 mg, 25 mg 5 mg, 25 mg 285986-88-1Ceralifimod B1289 5 mg, 25 mg 891859-12-4CFTR Inhibitor, GlyH-101 2863 5 mg, 25 mg 328541-79-3CH-223191 2723 5 mg, 25 mg 301326-22-7CHD-5 2693 5 mg, 25 mg 289494-16-2Chetomin 2180 1 mg 1403-36-7CHIR-090 B1852 5 mg, 25 mg 728865-23-4Chloroquine Diphosphate 1825 100 mg, 500 mg 50-63-5Chlorpromazine Hydrochloride B1992 100 mg, 500 mg 69-09-0CHR2797 2720 5 mg, 25 mg 238750-77-1CHS-828 2044 5 mg, 25 mg 200484-11-3CID 2745687 1969 5 mg, 25 mg 264233-05-8CID-5951923 2690 5 mg, 25 mg 749872-43-3Cladribine B2037 5 mg, 25 mg 4291-63-8Congo Red 2588 100 mg, 500 mg 573-68-0CPI-444 B1970 5 mg, 25 mg 1202402-40-1

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Product Name Cat. No. Size CAS. No.CPI-613 9464 10 mg, 50 mg 95809-78-2CT-2584 B1182 5 mg, 25 mg 166981-13-1Curcubitacin E B1592 1 mg, 5 mg 18444-66-1CWHM-12 B1251 5 mg, 25 mg 1564286-55-0DiscoveryPak™ Cytochlor-THU Set(Containing Cat. No. 2833, 1671) K955 2 Radiosensitizers 32387-56-7

18771-50-1Cytochlor 2833 5 mg, 25 mg 32387-56-7DBeQ 1858 5 mg, 25 mg 177355-84-9Decylubiquinone 2099 1 mg, 10 mg 55486-00-5DG051 B1105 1 mg, 5 mg 929916-05-2DHEA 2172 100 mg, 500 mg 53-43-0DMOG 2216 5 mg, 25 mg 89464-63-1Dofetilide B1189 5 mg, 25 mg 115256-11-6Dynasore 1900 5 mg, 25 mg 304448-55-3E-7046 B1966 5 mg, 25 mg 1369489-71-3Edoxaban Tosylate 2714 5 mg, 25 mg 480449-71-6Eliglustat B1217 5 mg, 25 mg 491833-29-5Embelin B1600 5 mg, 25 mg 550-24-3Entacapone B1190 10 mg, 50 mg 130929-57-6Epalrestat 2397 5 mg, 25 mg 82159-09-9Eptifibatide 2439 1 mg 188627-80-7Ethynylcytidine B1266 5 mg, 25 mg 180300-43-0(R)-(+)-Etomoxir B1104 1 mg, 5 mg 124083-20-1Evans Blue Tetrasodium 2586 1 g 314-13-6Ezatiostat 2608 5 mg, 25 mg 168682-53-910058-F4 2739 5 mg, 25 mg 403811-55-2Fatostatin 2035 5 mg, 25 mg 298197-04-3FCCP 2398 5 mg, 25 mg 370-86-5Felbamate B2004 10 mg, 50 mg 25451-15-4Fevipiprant B1588 5 mg, 25 mg 872365-14-5Fidaxomicin 2832 1 mg, 5 mg 873857-62-6FITM B1859 1 mg, 5 mg 932737-65-0 FK-866 1914 1 mg, 5 mg 658084-64-1FLI-06 2603 5 mg, 25 mg 313967-18-9Fosaprepitant 9529 10 mg, 50 mg 172673-20-0FPS-ZM1 B1933 5 mg, 25 mg 945714-67-0Fulvestrant B1863 5 mg, 25 mg 129453-61-8Fusicoccin B1625 1 mg, 2 mg 20108-30-9FX1 B2010 5 mg, 25 mg 1426138-42-2Ganciclovir 1918 50 mg, 250 mg, 1 g 82410-32-0GBR-12935 B1998 10 mg, 50 mg 76778-22-8GDC-0152 B1602 5 mg, 25 mg 873652-48-3DiscoveryPak™ Gemcitabine-THU Set(Containing Cat. No. 1759, 1671) K841 2 Modulators 122111-03-9

18771-50-1Geodin 9685 1 mg, 5 mg 427-63-4GIBH-130 B2071 5 mg, 25 mg 1252608-59-5GKT-137831 9444 5 mg, 25 mg 1218942-37-0GLPG-1690 B1850 5 mg, 25 mg 1628260-79-6Glutaminase C-IN-1 (968) B1198 5 mg, 25 mg 311795-38-7GSK-961081 B1590 5 mg, 25 mg 743461-65-6GSK1325756 B1103 1 mg, 5 mg 954126-98-8GSK2190915 B1891 1 mg, 5 mg 936350-00-4GSK2330672 B1102 1 mg, 5 mg 1345982-69-5GW 4869 dihydrocloride 2417 1 mg, 5 mg 6823-69-4GYY 4137 1908 5 mg, 25 mg 106740-09-4HA 130 B1192 5 mg, 25 mg 1229652-21-4Heptelidic Acid 2215 250 µg, 1 mg 74310-84-2Itaconic acid 2576 1 g, 5 g 97-65-4Ivabradine Hydrochloride B1595 10 mg, 50 mg 148849-67-6JNJ-31020028 9648 5 mg, 25 mg 1094873-14-9K858 B1073 10 mg, 50 mg 72926-24-0Ki 16425 9545 5 mg, 25 mg 355025-24-0

Product Name Cat. No. Size CAS. No.L-67 9633 5 mg, 25 mg 325970-71-6L-DON B1955 5 mg, 25 mg 157-03-9Lamotrigine B1234 10 mg, 50 mg 84057-84-1Lasofoxifene tartrate 9680 5 mg, 25 mg 190791-29-8LCL161 B1601 5 mg, 25 mg 1005342-46-0Leelamine hydrochloride 2717 5 mg, 25 mg 16496-99-4Lomitapide 2876 5 mg, 25 mg 182431-12-5LY404187 2698 5 mg, 25 mg 211311-95-4Macitentan B1856 5 mg, 25 mg 441798-33-0Madrasin B1278 5 mg, 25 mg 374913-63-0Mambalgin-1 2421 50 µg, 100 µg N/AMaraviroc B2044 5 mg, 25 mg 376348-65-16-Mercaptopurine (monohydrate) B2039 50 mg, 250 mg 50-44-2MDV-3100 9479 10 mg, 50 mg 915087-33-1Mifepristone 1561 50 mg 84371-65-3Mirin B1075 10 mg, 50 mg 1198097-97-0 MK-1439 B1250 5 mg, 25 mg 1338225-97-0 ML-354 9415 5 mg, 25 mg 89159-60-4ML161 2689 5 mg, 25 mg 423735-93-7MPEP hydrochloride B1151 10 mg, 50 mg 219911-35-03-Nitropropionic acid 2093 50 mg, 250 mg 504-88-12-Nitro-5-thiothiocyanatobenzoic acid B1316 50 mg, 250 mg 30211-77-9NS-3763 B1814 5 mg, 25 mg 70553-45-6NS6180 B1640 5 mg, 25 mg 353262-04-1NSC-207895 B1228 5 mg, 25 mg 58131-57-0NSC-348884 B1204 5 mg, 25 mg 81624-55-7NVS-SM1 B1844 5 mg, 25 mg 1562338-42-4ODQ 2051 10 mg, 50 mg 41443-28-1ONO 1078 B1099 5 mg, 25 mg 103177-37-3OSMI-1 B1916 5 mg, 25 mg 1681056-61-0Ozanimod B1196 5 mg, 25 mg 1306760-87-1PBTZ169 B1205 5 mg, 25 mg 1377239-83-2PD-1/PD-L1 Inhibitor 1 B1213 5 mg, 25 mg 1675201-83-8PD-1/PD-L1 Inhibitor 2 B1050 5 mg, 25 mg 1675203-84-5PD-123319 ditrifluoroacetate 9640 5 mg, 25 mg 130663-39-7Pellitorine 2053 1 mg, 5 mg 18836-52-7Pemetrexed B1862 50 mg, 250 mg 137281-23-3Pentostatin B2038 5 mg, 25 mg 53910-25-1Perampanel B2066 5 mg, 25 mg 380917-97-5PF-04418948 B1168 5 mg, 25 mg 1078166-57-0PF-06291874 B2001 5 mg, 25 mg 1393124-08-7 PF-3274167 B1026 5 mg, 25 mg 900510-03-4PF-8380 B1927 1 mg, 5 mg 1144035-53-9Phloretin 9625 100 mg, 500 mg 60-82-2Pimecrolimus 1593 5 mg, 25 mg 137071-32-0PK 11195 2054 10 mg, 50 mg 85532-75-83PO B2018 10 mg, 50 mg 13309-08-5Posaconazole 9526 10 mg, 50 mg 171228-49-2Prasugrel 9472 10 mg, 50 mg 150322-43-3PSI-7977 2715 5 mg, 25 mg 1190307-88-0PTC-124 9421 10 mg, 50 mg 775304-57-9PTC-209 B1055 5 mg, 25 mg 315704-66-6QNZ46 B2007 5 mg, 25 mg 1237744-13-6R162 B1180 5 mg, 25 mg 64302-87-0RAD140 B1211 10 mg, 50 mg 1182367-47-0Retro-2 2516 5 mg, 25 mg 1429192-00-6RI-1 B1823 5 mg, 25 mg 415713-60-9Rivaroxaban B1854 10 mg, 50 mg 366789-02-8RK-33 B1273 5 mg, 25 mg 1070773-09-9Ro 48-8071 fumarate B1042 10 mg, 50 mg 189197-69-1RQ-002303078 9636 10 mg, 50 mg 1254205-52-1

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For complete list of products please visit www.BioVision.com.

Product Name Cat. No. Size CAS. No.RSV-604 B1846 5 mg, 25 mg 676128-63-5 S0859 9425 5 mg, 25 mg 1019331-10-2Salubrinal 1980 5 mg 405060-95-9SB-715992 2468 5 mg, 25 mg 336113-53-2SB-742457 9568 5 mg, 25 mg 607742-69-8SM-164 B1816 250 μg, 1 mg 957135-43-2Suplatast tosylate 2624 10 mg, 50 mg 94055-76-2Suvorexant B1321 5 mg, 25 mg 1030377-33-3Syrosingopine B1323 1 mg, 5 mg 84-36-6T-5224 9546 5 mg, 25 mg 530141-72-1TAS-301 9644 10 mg, 50 mg 193620-69-8TCS OX2 29 B1838 5 mg, 25 mg 372523-75-6Tenofovir disoproxil fumarate 1920 5 mg, 25 mg 202138-50-9EZSolution™ Tetrahydrouridine 2355 25 mg 18771-50-1Tetrahydrouridine 1671 10 mg, 25 mg 18771-50-1TG6-10-1 9646 5 mg, 25 mg 1415716-58-3Thapsigargin 1558 1 mg 67526-95-8Thiabendazole 2161 1 g 148-79-8Tiplaxtinin B1634 5 mg, 25 mg 393105-53-8TM-5275 Sodium salt B1884 5 mg, 25 mg 1103926-82-4Tranilast 1876 10 mg, 50 mg 53902-12-8

Product Name Cat. No. Size CAS. No.trans-ISRIB B1906 5 mg, 25 mg 1597403-47-8EZSolution™ Triacsin C 9683 100 µg, 500 µg 76896-80-5Triapine B1174 10 mg, 50 mg 143621-35-6Triclopidine hydrochloride B1141 50 mg, 250 mg 53885-35-1Trifluorothymidine B1126 10 mg, 50 mg 70-00-8Triflupromazine hydrochloride B1993 100 mg, 500 mg 1098-60-8Troviridine B1212 10 mg, 50 mg 149488-17-5Tunicamycin 2802 5 mg, 25 mg 11089-65-9U-104 9631 5 mg, 25 mg 178606-66-1U-93631 B1851 5 mg, 25 mg 152273-12-6UK-371804 B1843 5 mg, 25 mg 256477-09-5UK-5099 B1952 5 mg, 25 mg 56396-35-1UMI-77 B1108 5 mg, 25 mg 518303-20-3XAV939 1727 1 mg 284028-89-3YK-4-279 2846 5 mg, 25 mg 1037184-44-3YM-90709 B1074 10 mg, 50 mg 163769-88-8YM155 2310 5 mg, 25 mg 781661-94-7(Z)-4-Hydroxytamoxifen B1114 5 mg, 25 mg 68047-06-3Z-VRPR-FMK B1238 250 µg, 1 mg 1381885-28-4Zanamivir B1900 10 mg, 50 mg 139110-80-8

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