10 cloranfenicol. dra. raquel
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CLASIFICACIÓN DE ANTIMICROBIANOS
III. ACTÚAN EN EL CITOPLASMA: A. INHIBIDORES DE SÍNTESIS DE PROTEÍNAS.
1. IRREVERSIBLES: AMINOGLICÓSIDOS.
2. REVERSIBLES:a) MACRÓLIDOS
b) CETÓLIDO
c) LINCOSAMIDASd) TETRACICLINAS
e) CICLILGLICINA
f) CLORANFENICOL
g) OXAZOLIDINONASh) ESTREPTOGRAMINAS
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Streptomyces venezuelae
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Gram +
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UAC
pMET
Fen
5’ ^^^^^^ AUG ^^^^ UUU ^^^^ AAG ^^^^ CGG ^^^^ 3’ UAC
pMETFen
5’ ^^^^^^ AUG ^^^^ UUU ^^^^ AAG ^^^^ CGG ^^^^ 3’ AAA AAA
ELONGACIÓN
(PEPTIDIL TRANSFERASA)
Peptidil transferasaCL
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ANAEROBIOSAntimicrobiano (s)Recomendado (s)
Alternativa (s) También efectivo (s)
Peptostreptococo Pen-G Clindamicina CARB, VANCO o TEICODOXI, ERITRO
Clostridiumperfringes
Pen-G +/-Clindamicina
DOXI TIC o PIP, Cefoxitina
CARB, CLOR, ERITRO
Clostridium tetani Pen-GMetronidazol
DOXI CARB
Clostridiumdifficile
Metronidazol (oral) VANCO (oral) Bacitracina (oral)
Fusobacterium
nucleatum
Pen-G
Clindamicina
Metronidazol CARB, Cefoxitina,
DOXI, CLOR,ERITRO/AZITRO
Prevotellamelaninogénicus
CARBMetronidazol
TC-CLClindamicina
AM-SB, PIP-TZ
Bacteroides fragilis Metronidazol Clindamicina AM-SB, TC-CL
PIP-TZ, CARB,Cefoxitina
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- Via de administración Oral y E.V.
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