tudományos munkásság: i. publikációk és független idézettségük · tudományos...

Tudományos munkásság: I. Publikációk és független idézettségük 1. G. Bernáth, Z. Szakonyi, F. Fülöp, P. Sohár: Synthesis of tert-butylcyclopentane-fused 1,3-oxazines and 1,3-thiazines Heterocycles 37, 1687-94 (1994) I.f.: 0,989

1. Rodd’s Chemistry of Carbon Compounds, Ed.: M. Sainsbury, Elsevier Science, Amsterdam, 1998, Vol. IV, Part H, p. 436

2. Bernáth G., Szakonyi Zs., Fülöp F., Sohár P.: terc-Butil-ciklopentánnal kondenzált 1,3-oxazinok és 1,3-tiazinok szintézise Acta Pharm. Hung. 64, 153-157 (1994)

1. J. E. Thirkettle, C. J. Schofield, M. W. Walter, Amino Acids, Peptides, and Proteins 28, 281-333 (1997)

2. Rodd’s Chemistry of Carbon Compounds, Ed.: M. Sainsbury, Elsevier Science, Amsterdam, 1998, Vol. IV, Part H, p. 436

3. N. De Kimpe, M. Boeykens, L. Lázár, Z. Szakonyi, A. Kemme, G. Duburs: Rearrangement and cyclization of β-mesyloxy ketones. Synthesis of δ-sultones Bull. Soc. Chim. Belg. 103, 299-302 (1994) I.f.: 0,354

1. P. Metz: J. Prak. Chem-Chem. Ztg. 340, 1 (1998) 4. Z. Szakonyi, F. Fülöp, G. Bernáth, P. Sohár: Synthesis of tert-butylcyclopentane-fused pyrimidin-4-ones Heterocycles 42, 625-34 (1996) I.f.: 0,976

1. M. P. Groziak: Progress in Heterocyclic Chemistry 9 249-267 (1997) 5. Szakonyi Zs., Fülöp F., Bernáth G., Sohár P.:

terc-Butil-ciklopentánnal kondenzált pirimidin-4-onok Magyar Kémiai Folyóirat, 104, 17-24 (1998) I.f.: 0,262

1. M. G. A. Shvekhgeimer: Khim. Geterotsikl. 483-529 (2003) 2. M. G. Shvekhgeimer: Chemistry of Heterocyclic Compounds, 39(4), 405-448

(2003)

6. N. De Kimpe, D. De Smaele, Z. Szakonyi: A new synthesis of 2-methyleneaziridines J. Org. Chem., 62, 2448-2452, (1997) I.f.: 3,476

1. J. Ince, M. Shipman, D. S. Ennis: Tetrahedron Lett. 38, 5887 (1997) 2. S.S. Murphree, A. Padwa: Progress in Heterocyclic Chemistry 10 49-69 (1998) 3. M. Shipman, T. M. Ross, A.M.Z. Slawin: Tetrahedron Lett. 40, 6091 (1999) 4. D.S. Ennis, J. Ince, S. Rahman et al.: J. Chem Soc. Perk. Trans. 1 2047 (2000) 5. M. Karpf, R. Trussardi: J. Org. Chem. 66, 2044 (2001) 6. J.F. Hayes, M. Shipman, H. Twin: J. Org. Chem. 67 (3), 935-942 (2002)

7. N. Prevost, M. Shipman: Tetrahedron 58 (35), 7165-7175 (2002) 8. B. H. Oh, I. Nakamura, Y. Yamamoto: Tetrahedron Lett. 43 (52) 9625-9628

(2002) 9. B. H. Oh, I. Nakamura, Y. Yamamoto: ARKIVOC 2003 (xiii) 67-78. 10. Y. H. Oh, I. Nakamura , Y. Yamamoto: J. Org. Chem. 69(8), 2856-2858

(2004) 11. M. Karikomi, T. Takayama, K. Haga, K. Hiratani: Tetrahedron Lett. 46 (38)

6541-6544 (2005) 12. C. Montagne, N. Prevost, J. J. Shiers, G. Prie, S. Rahman, J. F. Hayes, M.

Shipman: Tetrahedron 62 (36) 8447-8457 (2006) 13. M. Shipman: SYNLETT (19) 3205-3217 (2006) 14. K. K. A. D. S. Kathriarachchi, A. I. Siriwardana, I. Nakamura, Y.

Yamamoto: Tetrahedron Lett. 48 (13) 2267-2270 (2007) 15.Comprehensive Heterocyclic Chemistry III., Ed.: A. R. Katritzky, C. A.

Ramsden, R. J. K. Taylor, E. F. V. Scriven, Elsevier Ltd. Oxford, 2008, Vol. 1.01, p82.

16. K. Higashiyama, M. Matsumura, H. Kojima, T. Yamauchi: Heterocycles, 78(2), 471-485 (2009)

17. J. Magano: Chem. Rev., 109, 4398-4438 (2009) 7. F. Fülöp, Z. Szakonyi, G. Bernáth, P. Sohár: Synthesis of 2,4-dioxo and 4-oxo-2-thioxo derivatives of octahydro-

cyclopenta[d]pyrimidines J. Heterocyclic Chem., 34, 1211-1217 (1997) I.f.: 0,669

1. Progress in Heterocyclic Chemistry (Eds: G. W. Gribble, T. L. Gilchrist), 1997, p. 256

2. M. P. Groziak: Progress in Heterocyclic Chemistry, 10, 251-274 (1998) 3. E. Atay, I.B. Blagoeva, F.L. Chubb, et al.: Can. J. Chem. 78, 84-94 (2000)

8. Z. Szakonyi, F. Fülöp, G. Bernáth, F. Evanics, F. G. Riddell: Synthesis and characterisation of angularly substituted cycloalkane-fused tetrahydro-1,3-oxazines Tetrahedron, 54, 1013-1020, (1998) I.f.: 2,16

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3. A. Star, B. Fuchs: J. Org. Chem. 64, 1166 (1999) 4. J. P. Tam, Z. Miao: J. Am. Chem. Soc. 121, 9013-9022 (1999) 5. P. Tähtinen, A. Bagno, K. D. Klika, K. Pihlaja: J. Am. Chem. Soc. 125 (15):

4609-4618 (2003) 6. J. H. Ye, Y. Huang, R. Y. Chen: Org. Prep. Proced. Int. 35(4) 429-432 (2003) 7. A. W. Murray: Organic Reaction Mechanisms 487-615 (2003) 8. A. A. Fuller, B. Chen, A. R. Minter, A. K. Mappet, J. Am. Chem. Soc. 127

(15), 5376-5383 (2005) 9. S. Pérez, C. López, A. Caubet, A. Roig, E. Molins, J. Org. Chem. 70 (12),

4857-4860 (2005) 10. E. V. Bayandina, E. Y. Davydova, M. N. Dimukhametov, Dobrynin AB,

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11. M. Sathe, R. Ghorpade, M. P. Kaushik: Chemistry Letters 35(9), 1004-1005 (2006)

12. D. N. Dhar, P. Dhar: The chemistry of chlorosulfonyl isocyanate, World Scientific Publishing Co., Singapore, 2002.

13. M. Sathe, D. Thavaselvam, A. K. Srivastava, M. P. Kaushik: Molecules, 13, 432-443 (2008) 14. M. Yoshioka, M. Takenaka, Y. Shin, T. Orita, K. Shundo, M. Watari:

Japanese Journal of Chemotherapy 56(1), 1-6 (2008) 9. Z. Szakonyi, F. Fülöp, G. Bernáth, G. Török, A. Péter: Preparation of cycloalkane-fused dihydropyrimidin-4(3H)-one enantiomers Tetrahedron: Asymmetry, 9, 993-999 (1998) I.f.: 2,484

1. R. M. Alvarez, A. H. Fernandez, A. S. Vazqez, J.J.A. Maroto, M. Chioua, R. Chioua: Rapid Comm. Mass Spectrom. 13, 79-83 (1999)

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3. M. P. Groziak: Progress in Heterocyclic Chemistry 11, 256-275 (1999) 4. Herrera A, Martinez-Alvarez R, Chioua M, et al.: Magn. Reson. Chem. 40,

293-299 (2002) 5. J. A. Miller, S. T. Nguyen: Mini-Reviews in Organic Chemistry 2, 39-45

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Tetrahedron 61 (17), 4249-4260 (2005) 7. Chaturong Suparpprom, Choladda Srisuwannaket, Polkit Sangvanich, Tirayut

Vilaivan, Tetrahedron Lett. 46 (16), 2833-2837 (2005) 10. E. Forró, Z. Szakonyi, F. Fülöp:

Enzymatic resolution of (±)-2-(Nβ-t-butoxycarbonyl-Nα-methylhydrazino)-cycloalkanols Tetrahedron: Asymmetry, 10, 4619-4626 (1999) I.f.: 2,647

1. Anon: Process Biochemistry (Oxford) 36(1-2), 189-200 (2000) 2. S.M. Roberts: J. Chem. Soc., Perkin Trans. 1 1475-1499 (2001) 3. L. M. Levy, I. Lavandera, V. Gotor: Org. Biomol. Chem. 2(18) 2572-2577

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Chem. 71, 2320-2331 (2006) 5. J. Gonzalez-Sabin, I. Lavandera, F. Rebolledo, V. Gotor: Tetrahedron:

Asymmetry, 17, 1264-1274 (2006) 6. Q. Jing, R. J. Kaziauskas: Chirality 20, 724-735 (2008) 7. I. Schiffers, C. Bolm: Org. Synth. 85, 106-117 (2008)

11. Z. Szakonyi, T. Martinek, A. Hetényi, F. Fülöp:

Synthesis and transformations of enantiomeric 1,2-disubstituted monoterpene derivatives Tetrahedron: Asymmetry, 11 4571-4579 (2000) I.f.: 2,797

1. J. A. Miller, S. T. Nguyen: Mini-Reviews in Organic Chemistry 2, 39-45 (2005)

2. D. Viña, L. Santana, E. Uriarte, C. Terán : Tetrahedron 61, 473-478 (2005) 3. A. Liljeblad, L. T. Kanerva: Tetrahedron 62, 5831-5854 (2006)

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6. E. A. Koneva, K. P. Volcho, Y. V. Gatilov, D. V. Korchagina, G. E. Salnikov, N. F. Salakhutdinov: Helv. Chim. Acta 91, 1849-1856 (2008)

7. T.G. Tolstikova, E.A. Morozova, A.V. Pavlova, A.V. Bolkunov, M.P. Dolgikh, E.A. Koneva, K.P. Volcho, N.F. Salakhutdinov, G.A. Tolstikov, 2008, Doklady Akademii Nauk, 422, 490-492 (2008)

8. E. A. Koneva, K. P. Volcho, D. V. Korchagina, N. I. Komarova, A. I. Kochnev, N. F. Salakhutdinov, A. G. Tolstikov: Russian Chem. Bull. 57(1), 108–117 (2008)

12. A. Salgado, T. Huybrechts, A. Eeckhaut, J. Van der Eycken, Z. Szakonyi, F. Fülöp, A. Tkachev, N. De Kimpe: Synthesis of (1S)-1-amino-2,2-dimethylcyclopentane-1-carboxylic acid via PLE mediated hydrolysis of bis(2,2,2-trifluoroethyl)2,2-dimethylcyclopropane-1,1-dicarboxylate Tetrahedron, 57, 2781-2786 (2001) I.f.: 2,276

1. E. Bunuel, S. D. Bull, S. G. Davies, A. C. Garner, E. D. Savory, A. D. Smith, R. J. Vickers, D. J. Watkin: Org. Biomol. Chem. 1(14) 2531-2542 (2003)

2. G.F. Su, H.T. Mu, D.M. Za, L.M. Zeng, C. Cativiela, R.P. Hammer, K.B. Yu: Synth. Commun. 33(16), 2873-2884 (2003)

3. T.T. Talele, M.L. McLaughlin: Biopolymers 71(3), 182 (2003) 4. A. I. Jimemez, P. Lopez, C. Cativiela: Chirality 17(1), 22-29 (2005) 5. S. P. Bew: Comprehensive Organic Functional Group Transformations II 5,

19-125 (2005) 6. J. T. Su, G. F. Qiu, S. C. Liang, X. M. Hu Synth. Commun. 35(11), 1427-

1433 (2005) 7. H. Lebel, O. Leogane: Org. Lett. 7(19), 4107-4110 (2005) 8. S. Akai, T. Tsujino, N. Fukuda, K. Iio, Y. Takeda, K. Kawaguchi, T. Naka,

K. Higuchi, E. Akiyama, H. Fujioka, Y. Kita Chemistry-A European Journal 11(21), 6286-6297 (2005)

9. M. Pizzonero, F. Dumas, J. d'Angelo Heterocycles 66, 31-37 (2005) 10. J.T. Su, J. Xiong, S. C. Liang, G. F. Qiu, X. C. Feng, H. B. Teng, L. M. Wu,

X. M. Hu Synth. Commun. 36 (6), 693-699 (2006) 11. W. C. Chan, A. Higton, J. S. Davies Amino Acids, Peptides, and Proteins 35,

1-73 (2006) 12. P. D. de Maria, C. A. Garcia-Burgos, G. Bargeman, R. W. van Gemert

Synthesis-Stutgart 10, 1439-1452 (2007) 13. F. Brackmann, A. de Meijere : Chem. Rev., 107, 4493-4537 (2007) 14. Q. F. Zhu, Z.X. Xu, Y. B. Hao, Y. L. Xiao, W. J. Xu, X. B. Ke, H. B. Teng,

L. M. Wu, G. F. Qiu, S. C. Liang, X. M. Hu: Lett. Org. Chem. 5(6), 478-483 (2008)

15. C. Cativiela, M. Ordóñez: Tetrahedron: Asymmetry 20, 1–63 (2009) 16. Y. A. Volkova, O. A. Ivanova, E. M. Budynina, E. V. Revunov, E. B.

Averina: Tetrahedron Lett. 50, 2793-2796 (2009)

13. P. Tähtinen, J. Sinkkonen, K.D. Klika, V. Nieminen, G. Stájer, Z. Szakonyi, F. Fülöp, K. Pihlaja 1H, 13C, and 15N NMR stereochemical study of cis-fused 7a(8a)-methyl and 6-phenyl octa(hexa)hydrocyclopenta[d][1,3]oxazines and [3,1]benzoxazines Chirality, 13, 1-12 (2002) I.f.: 1,554

1. G. Puigbo, F. Diaba, J. Bonjoch: Tetrahedron 59(15), 2657-2665 (2003 ) 2. R. H. Contreras, V. Barone, J. C. Facelli, J. E. Peralta: Annual Reports on

NMR Spectroscopy 51, 167-260 (2003) 3. E. Kolehmainen: Annual Reports on NMR Spectroscopy 49, 167-260 (2003) 4. W.-D. Rudorf: Journal of Sulfur Chemistry 28 (3), 295-339 (2007) 5. L. B. Krivdin, R. Contreras: Annual Reports on NMR Spectroscopy 61, 133-

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Chem. 11(13), 1154-1205 (2007) 14. Z. Szakonyi, F. Fülöp, D. Tourwé, N. De Kimpe

Synthesis of 1,2,7,7a-tetrahydro-1aH-cyclopropa[b]quinoline-1a-carboxylic acid derivatives, doubly constrained ACC derivatives, by a remarkable cyclopropanation process. J. Org. Chem., 67, 2192-2196 (2002) I.f.: 3,28

1. M. Meusel, M. Guetschow Org. Prep. Proced. Int. 36(5) 391-443 (2004) 2. S. P. Bew: Comprehensive Organic Functional Group Transformations II 5,

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3369 (2005) 4. F. Brackmann, A. de Meijere : Chem. Rev., 107, 4493-4537 (2007) 5. W. Wan, Y. Gao, H. Jiang, J. Hao: J. Fluorine. Chem. 129, 510-514 (2008)

15. S. Gyónfalvi, Z. Szakonyi, F. Fülöp

Synthesis and transformation of novel cyclic β-amino acid derivatives from (+)-3-carene Tetrahedron: Asymmetry, 14, 3965-3972 (2003) I.f.: 2,178

1. M. I. Aguilar, G. D. Fallon, P. A. Mayes, S. Nordin, A. J. Robinson, M. L. Rose, F. Vounatsos, B. Wilman, P. Perlmutter: Letters in Peptide Science 10(5-6), 597-604 (2003)


3. F. Z. Macaev, A. V. Malkov Tetrahedron 62 9-29 (2006) 4. M. Frackowiak, K. Ochalik, A. Bialonska, Z. Ciunik, C. Wawrzenczyk, S.

Lochynski Tetrahedron: Asymmetry, 17 124-129 (2006) 5. M. Sathe, R. Ghorpade, M. P. Kaushik: Chemistry Letters 35(9), 1004-1005

(2006) 6. X.-G. Li, M. Lähitie, M. Päiviö, L.T. Kanerva: Tetrahedron: Asymmetry 18,

1567–1573 (2007) 7. B. Alcaide, P. Almendros, C. Aragoncillo: Chem. Rev., 107, 4437-4592

(2007) 8. A. Mondière, R. Peng, R. Remuson, D.J. Aitken: Tetrahedron 64, 1088-

1093 (2008)

9. M. D’hooghe, Y. Dejaegher, N. De Kimpe: Tetrahedron 64, 4575–4584 (2008)

10. M. Sathe, H. N. Karade, M. P. Kaushik: Synth. Commun. 38(9), 1375-1380 (2008)

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13. L. Zhou, H.F. Jiang, C.J. Li : Adv. Synth. Catal. 350, 2226-2230 (2008) 14. E. A. Koneva, T. M. Khomenko, S. Yu. Kurbakova, N. I. Komarova, D. V.

Korchagina, K. P. Volcho, N. F. Salakhutdinov, A. G. Tolstikov, G. A. Tolstikov: Russ. Chem. Bull., Int. Ed., 57, 1680-1685 (2008)

15. E. Forró: J. Chrom. A. 1216(6), 1025-1029 (2009) 16. K. Gajcy, T. Librowski, S. Lochynski: Lett. Org. Chem. 6(3), 186-188

(2009) 17. E. A. Koneva, K. P. Volcho, D. V. Korchagina, N. F. Salakhutdinov, A. G.

Tolstikov: Russ. J. Org. Chem. 45, 815-824 (2009) 16. G. Tóth, Z. Szakonyi, B. Kanyó, F. Fülöp, G. Jancsó, L. Pávics: Preparation of

[99mTc]TRODAT-1 involving a simple purification method J. Labelled Compd. Rad., 46, 1067-1073 (2003) I.f.: 1,207

1. Z. P. Chen, S. P. Wang, J. Tang, X. M. Li, C. Y. Liu, X. J. Xu, G. X. Cao: Journal of Radioanalytical and Nuclear Chemistry 3, 591-594 (2008), DOI: 10.1007/s10967-007-7109-z

17. Kanyó B. Árgyelán M., Dibó Gy., Szakonyi Zs., Vécsei L., Fülöp F., Láncz A.,

Forgács P., Pávics L: Dopamintranszporter-vizsgálatok egyfotonemissziós komputertomográfiával (SPECT) mozgászavarokkal járó kórképekben Clin. Neurosci./Ideggy. Szle. 56(7-8), 231-240 (2003)

1. C.S. Ming, E. Amaro Jr., H. B. Ferraz, M. Q. Hoexter, F. O. Goulart, J.

Wagner, F. L. Li, K. F. Ying, J. J. Mari, A. L. T. De Lacerda, S. Tufik, R.A. Bressan Arq. Neuro-Psiquiatr., 64 (3A) 628-634 (2006)

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3. I.H. Li, W.S. Huang, C.B. Yeh, M.H. Liao, C.C. Chen, L.H. Shen, J.C. Liu, K.H. Ma: Nuclear Medicine and Biology 36, 605–611 (2009)

4. 18. E.R. Alonso, K.A. Tehrani, M. Boelens, A.V. Tkachev, Z. Szakonyi, F. Fülöp, N. De

Kimpe Novel synthesis of functionalized 2-pyrrolidinones via unsaturated imidoyl cyanides Organic Preparations and Procedures International, 35, 215-219 (2003)

I.f.: 0,841

19. A. Hetényi, Z. Szakonyi, K. D. Klika, K. Pihlaja, and F. Fülöp Formation and characterization of a nine-component equilibrium system derived from cis- and trans-1-aminomethylcyclohexane-1,2-diol J. Org. Chem., 68, 2175-2182 (2003) I.f.: 3,297

1. H. S. El Khadem, A. J. Fatiadi Carbohydrate Chemistry and Biochemistry 59, 135-173 (2004)

2. S. Pérez, C. López, A. Caubet, A. Roig, E. Molins, J. Org. Chem. 70 (12), 4857-4860 (2005)

3. E. Frank, B. Kazi,, Z. Mucsi, K. Ludányi, G. Keglevich: Steroids 72 (5), 446-458 (2007)

20. M. D'hooghe, Z. Szakonyi, F. Fülöp, N. De Kimpe

Synthesis of N-(4-chlorobutyl)butanamide, a chlorinated amide isolated from Aloe sabaea Organic Preparations and Procedures International, 35, 501-507 (2003)

I.f.: 0,841

21. Z. Szakonyi, F. Fülöp Mild and efficient ring opening of monoterpene-fused β-lactam enantiomers. Synthesis of novel β-amino acid derivatives ARKIVOC, (xiv), 225-232 (2003) I.f.: 0,392

1. L. Liu, L.L. Zhang, G. Liu, J. X. Xu: ARKIVOC (xvi) 318-326 (2008)

22. Lázár L., Szakonyi Zs., Forró E., Palkó M., Zalán Z., Szatmári I., Fülöp F. Gyulladásgátló hatású hidrazinoalkoholok szintézise Acta Pharm. Hung., 74, 11-18 (2004)

23. F. Fülöp, L. Lázár, Z. Szakonyi, M. Pihlavisto, S. Alaranta, P. J. Vainio, A. Juhakoski, A. Marjamäki, D. J. Smith Discovery of new anti-inflammatory agents Pure Appl. Chem., 76 (5), 965–972 (2004). I.f.: 1,449

1. P. Knowles, C. Kurtis, J. Murray, C. Saysell, W. Tambyrajah, C. Wilmot, M. McPherson, S. Phillips, D. Dooley, D. Brown, M. Rogers, M. Mure: J. Neural Transmission 114(6), 743-746 (2007)

2. B. M. Strolin, K.F. Tipton, R. Whomsley: Fundamental and Clinical Pharmacology 21(5), 467–479 (2007)

3. P. Dunkel, A. Gelain, D. Barlocco, N. Haider, K. Gyires, B. Sperlágh, K. Magyar, E. Maccioni, A. Fadda, P. Mátyus, Curr. Med. Chem. 15, 1827-1839 (2008)

24. Z. Szakonyi, M. D’hooghe, I. Kanizsai, F. Fülöp, N. De Kimpe

Synthesis of bicyclic carbamates as precursors of Sedum alkaloid derivatives Tetrahedron 61, 1595-1602 (2005) I.f.: 2,61

1. J. D. Adams, C. Garcia Evidence-based complementary and alternative medicine 3 (1), 125-131 (2006)

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3. J. M. Carney, P. J. Donoghue, W. M. Wuest, O. Wiest, P. Helquist: Org. Lett. 10(17), 3903–3906 (2008)

25. Z. Szakonyi, S. Gyónfalvi, A. Hetényi, F. Forró, N. De Kimpe, F. Fülöp

Synthesis of 3- and 4-hydroxy-2-aminocyclohexanecarboxylic acids by iodocyclization Eur. J. Org. Chem. 4017–4023 (2005) I.f.: 2,548

1. G. W. Gribble, J. A. Joule, Progress in Heterocyclic Chemistry, Vol.

18, Eds.: Elsevier, 2007, p. 112. 2. B. Alcaide, P. Almendros, C. Aragoncillo: Chem. Rev., 107, 4437-4592

(2007) 3. M. Lloyd, R. Lloyd, P. Keene, A. Osborne, Journal of Chemical Technology

and Biotechnology, 82(12), 1099-1106 (2007) 4. A. Mondière, R. Peng, R. Remuson, D.J. Aitken: Tetrahedron 64, 1088-1093

(2008) 5. O. Songis, C. Didierjean, J. Martinez, M. Calmés: Tetrahedron: Asymmetry

19, 2135–2139 (2008) 6. Y. Matsushima, J. Kino: Eur. J. Org. Chem., 1619-1624 (2009)

26. Z. Szakonyi, Á. Balázs, T. A. Martinek,F. Fülöp

Enantioselective addition of diethylzinc to aldehydes catalyzed by γ-amino alcohols derived from (+)- and (-)-α-pinene Tetrahedron: Asymmetry, 17, 199-204 (2006) I.f.: 2,468

1. E. Busto, V. Gotor-Fernandez, V. Gotor: Tetrahedron: Asymmetry, 17, 1007-1016 (2006)

2. R.W. Parrott II, S. R. Hitchcock: Tetrahedron: Asymmetry, 18, 377-382 (2007)

3. A. G. Martínez, E. T.,Vilar, A. G. Fraile, S. de la Moya Cerero, P. Martínez Ruiz, C. Díaz Morillo: Tetrahedron: Asymmetry, 18, 742-749 (2007)

4. B. Alcaide, P. Almendros, C. Aragoncillo: Chem. Rev., 107, 4437-4592 (2007)

5. R.W. Parrott II, S.R. Hitchcock: Tetrahedron: Asymmetry, 19, 19-26 (2008)

6. D. Hobuß, A. Baro, S. Laschat, W. Frey: Tetrahedron, 64, 1635-1640 (2008)

7. I.V. Il'ina, K.P. Volcho, N.E. Salakhutdinov: Russian J. Org. Chem. 44(1), 1-23 (2008)

8. B. Alcaide, P. Almendros, Progress in Heterocyclic Chemistry, Vol. 19, Eds.: Elsevier, 2008, p. 92-111.

9. A.B. Terent’ev, T.T. Vasil’eva, O.V. Chahovskaya, N.E. Mysova, H.H. Hambardzumyan, K.A. Kochetkov: J. Fluorine. Chem. 129, 669-673 (2008)

10. M.I. Burguete, J. Escorihuela, S.V. Luis, A. Lledo´s, G. Ujaque: Tetrahedron, 64, 9717-9724 (2008)


12. J. Li, Y.M. Shang, C. Xiao, Z.G. Song, Y.Z. Li, H.M. Huang: Chem. Res. Chinese U. 25(1), 43–46 (2009)

13. D. Scarpi, E. G. Occhiato, A. Guarna: Tetrahedron: Asymmetry, 20, 340–350 (2009)

14. N. Ananthi, U. Balakrishnan, A. Vinu, K. Ariga, S. Velmathi: Tetrahedron: Asymmetry, 20, 1731–1735 (2009)

15. T. Noël, K. Robeyns, L. Van Meervelt, E. Van der Eycken, J. Van der Eycken: Tetrahedron: Asymmetry, 20, 1962–1968 (2009)

27. J. Magyar, B. Horváth, T. Bányász, N. Szentandrássy, P. Birinyi, A. Varró, Z.

Szakonyi, F. Fülöp, P. P. Nánási L-364,373 fails to activate the slow delayed rectifier K+ current in canine ventricular cardiomyocytes Naunyn-Schmiedeberg’s Arch. Pharmacol. 373, 85-90 (2006) I.f.: 2,779

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28. I. Kanizsai,, Z. Szakonyi, R. Sillanpää, F. Fülöp

A comparative study of the multicomponent Ugi reactions of an oxabicycloheptene-based β-amino acid in water and in methanol Tetrahedron Lett. 47, 9113–9116 (2006) I.f.: 2,509

1. R. E. Dolle, B. Le Bourdonnec, A. J. Goodman, G. A. Morales, J. M. Salvino, W. Zhang, : J. Comb. Chem., 9(6), 855-902 (2007)

2. N. Shapiro, A. Vigalok: Angew. Chem. Int. Ed. 47(15), 2849-2852 (2008) 3. B. Alcaide, P. Almendros, Progress in Heterocyclic Chemistry, Vol.

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5. A. Brandi, S. Cicchi, F. M. Cordero: Chem. Rev., 108, 3988-4035 (2008) 6. C. C. A. Cariou, G. J. Clarkson, M. Shipman: J. Org. Chem. 73 (24), 9762-

9764 (2008) 7. C. Hulme, J. Dietrich: Mol. Divers. 13, 195–207 (2009)

29. I. Kanizsai, Z. Szakonyi, M. D’hooghe, F. Fülöp, N. De Kimpe

Synthesis of chiral 1,5-disubstituted pyrrolidinones via electrophile-induced cyclization of 2-(3-butenyl)oxazolines derived from (1R,2S)- and (1S,2R)-norephedrine Tetrahedron: Asymmetry, 17, 2857–2863 (2006) I.f.: 2,468 1. M. Hiroshi, O. Fumi, Y. Kenji: Heterocycles 74, 383-396 (2007)

30. I. Kanizsai, S. Gyónfalvi, Z. Szakonyi, R. Sillanpää, F. Fülöp

Synthesis of bi- and tricyclic β-lactam libraries in aqueous medium Green Chemistry, 9, 357-360 (2007) I.f.: 4,836

1. S. Capone, S. Pedatella, A. Guaragna, M. De Nisco, G. Palumbo: Tetrahedron, 63, 12202-12206 (2007)

2. O. Sereda, R. Wilhelm: Synlett, 3032-3036 (2007) 3. M. Krasavin, V. Parchinsky: Synlett, 645-648 (2008) 4. N. Liu, S. Cao, J. Wu, J. Yu, L. Shen, X. Feng, X. Qian: Tetrahedron, 64,

3966-3974 (2008) 5. G. Vasuki, K. Kumaravel: Tetrahedron Lett. 49, 5636-5638 (2008) 6. E. Forró: J. Chrom. A. 1216(6), 1025-1029 (2009)

7. A.S. Nagarajan, B.S.R. Reddy: Synlett, 2002-2004 (2009)

31. Á. Balázs, Z. Szakonyi, F. Fülöp

Synthesis of alicyclic N-substituted 1,3-amino alcohols via 1,3-oxazines J. Heterocyclic Chem., 44, 403–406 (2007) I.f.: 0,735

32. Z. Szakonyi, T. A Martinek, R. Sillanpää, F. Fülöp

Regio- and stereoselective synthesis of the enantiomers of monoterpene-based β-amino acid derivatives Tetrahedron: Asymmetry, 18, 2442–2447 (2007) I.f.: 2,634

1. M. Sathe, D. Thavaselvam, A. K. Srivastava, M. P. Kaushik: Molecules, 13, 432-443 (2008)

33. W. J. Peláez, Z. Szakonyi, F. Fülöp, G. I. Yranzo

Flash vacuum pyrolysis (FVP) of some hexahydroquinazolin-4(1H)-ones Tetrahedron 64, 1049-1057 (2008) I.f.: 2,897

34. Z. Szakonyi, A. Hetényi, F. Fülöp

Synthesis of enantiomeric spirooxazolines and spirooxazolidines by the regioselective ring closure of monoterpene-based aminodiols ARKIVOC part (iii) , 33-42 (2008) I.f.: 1,377

1. N. Hazeri, M. T. Maghsoodlou, S. M. Habibi-Khorassani, G. Marandi: ARKIVOC (xiv) 282-288 (2008)


Synthesis and application of monoterpene-based chiral aminodiols Tetrahedron 64, 1034-1039 (2008) I.f.: 2,897 1. D. Frain, F. Kirby, P. McArdle, P. O'Leary: Synlett 1261-1264 (2009) 2. H. Mehrabi: Can. J. Chem. 87(8), 1117-1121 (2009)


Regio- and stereoselective synthesis of constrained enantiomeric β-amino acid derivatives Tetrahedron: Asymmetry, 19, 2296–2303 (2008) I.f.: 2,796

37. Anasztázia Hetényi, Zsolt Szakonyi, István M. Mándity, Éva Szolnoki, Gábor K.

Tóth, Tamás A. Martinek, Ferenc Fülöp Sculpting the β-peptide H12 helix via a designed side-chain shape Chem. Commun. 177–179 (2009) I.f.: 5,34

1. T. Beke, C. Somlai, G. Magyarfalvi, A. Perczel, G. Tarczay: J. Phys.

Chem. B, 113(22), 7918-7926 (2009) 38. Á. Balázs, A. Hetényi, Z. Szakonyi, R. Sillanpää, F. Fülöp

Solvent Enhanced diastereo- and regioselectivity in the Pd(II)-catalyzed synthesis of six- and eight-membered heterocycles via cis-aminopalladation

Chemistry - A European Journal, 15, 7376–7381 (2009) I.f.: 5,454 39. Z. Szakonyi, R. Sillanpää, F. Fülöp

Synthesis of conformationally constrained tricyclic β-lactam enantiomers through Ugi four-centre three-component reactions of a monoterpene-based β-amino acid Mol. Div. kézirat elfogadva I.f.: 2,708

Össz I.f.: 81,475 II. Szabadalmak:

1. D. J. Smith, M. Jalkanen, F. Fülöp, L. Lázár, Z. Szakonyi, G. Bernáth: Inhibitors of copper-containing amine oxidases. (Biotie Therapies Corp., Finland). PCT Int. Appl. (2002),57 pp.; CAN 136:79760.

1. P. Mátyus, B. Dajka-Halász, A. Földi, N. Haider, D. Barlocco, K. Magyar:

Current Medicinal Chemistry 11(10), 1285-1298 (2004) 2. R. Ueno, A. Nagashima, T. Inoue, M. Ohkubo, K. Yoshihara PCT Int. Appl.

(2004), 269 pp., CAN 141:350160 3. S. S. Costa, M. De Souza, T. Ibrahim, G. Oliveira de Melo, A. P. De Almeida,

C. Guette, J.-P. Ferezou, V. L. G. Koatz J. Nat. Prod. 69(5), 815-818 (2006) 4. G. Negrón-Silva, C. X. Hernández-Reyes, D. Angeles-Beltrán, L. Lomas-

Romero, E. González-Zamora: Molecules, 13, 977-985 (2008) 5. P. Dunkel, A. Gelain, D. Barlocco, N. Haider, K. Gyires, B. Sperlágh, K.

Magyar, E. Maccioni, A. Fadda, P. Mátyus, Curr. Med. Chem. 15, 1827-1839 (2008)

2. D. J. Smith, J. David, M. Jalkanen, F. Fülöp, L. Lázár, Z. Szakonyi, G. Bernáth:

Oxadiazine derivatives as inhibitors of copper-containing amine oxidases. (Biotie Therapies Corp., Finland). PCT Int. Appl. (2002), 53 pp.; CA 136:102405.



(2004), 269 pp., CAN 141:350160 3. D. J. Smith, J. David; F. Fülöp, M. Pihlavisto, L. Lázár, S. Alaranta, P. Vainio, Z.

Szakonyi: Preparation of hydrazino indanes as inhibitors of copper-containing amine oxidases (Biotie Therapies Corporation, Finland). PCT Int. Appl. (2003), 58 pp.; CA 138:106506.

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2005063261, CAN 143:109791 4. P. Dunkel, A. Gelain, D. Barlocco, N. Haider, K. Gyires, B. Sperlágh, K.


4. F. Fülöp, Z. Szakonyi: Chiral cyclic β-amino acids and their derivatives, pharmaceutical compositions contaioning them and the use of such compounds (Bioblocks Magyarország Gyógyszerkémiai és Fejlesztı Kft., Hungary) PCT Int. Appl., WO 2008/059299 A1, 36 pp.

Összes független idézettség: 173 ISI független idézettség: 133 2009. szeptember 25.

Az elmúlt 10 év munkássága és független idézettsége: 1. Z. Szakonyi, T. Martinek, A. Hetényi, F. Fülöp:

Synthesis and transformations of enantiomeric 1,2-disubstituted monoterpene derivatives Tetrahedron: Asymmetry, 11 4571-4579 (2000) I.f.: 2,386


2. D. Viña, L. Santana, E. Uriarte, C. Terán : Tetrahedron 61, 473-478 (2005) 3. A. Liljeblad, L. T. Kanerva: Tetrahedron 62, 5831-5854 (2006)

4. M. Sathe, R. Ghorpade, M. P. Kaushik: Chem. Lett. 35(9), 1004-1005 (2006)



7. T.G. Tolstikova, E.A. Morozova, A.V. Pavlova, A.V. Bolkunov, M.P. Dolgikh, E.A. Koneva, K.P. Volcho, N.F. Salakhutdinov, G.A. Tolstikov, 2008, Doklady Akademii Nauk, 422, 490-492 (2008)


2. A. Salgado, T. Huybrechts, A. Eeckhaut, J. Van der Eycken, Z. Szakonyi, F. Fülöp, A. Tkachev, N. De Kimpe: Synthesis of (1S)-1-amino-2,2-dimethylcyclopentane-1-carboxylic acid via PLE mediated hydrolysis of bis(2,2,2-trifluoroethyl)2,2-dimethylcyclopropane-1,1-dicarboxylate Tetrahedron, 57, 2781-2786 (2001) I.f.: 2,643

1. E. Bunuel, S. D. Bull, S. G. Davies, A. C. Garner, E. D. Savory, A. D. Smith, R. J. Vickers, D. J. Watkin: Org. Biomol. Chem. 1(14) 2531-2542 (2003)

2. G.F. Su, H.T. Mu, D.M. Za, L.M. Zeng, C. Cativiela, R.P. Hammer, K.B. Yu: Synth. Commun. 33(16), 2873-2884 (2003)

3. T.T. Talele, M.L. McLaughlin: Biopolymers 71(3), 182 (2003) 4. A. I. Jimemez, P. Lopez, C. Cativiela: Chirality 17(1), 22-29 (2005) 5. S. P. Bew: Comprehensive Organic Functional Group Transformations II 5,

19-125 (2005) 6. J. T. Su, G. F. Qiu, S. C. Liang, X. M. Hu Synth. Commun. 35(11), 1427-

1433 (2005) 7. H. Lebel, O. Leogane: Org. Lett. 7(19), 4107-4110 (2005) 8. S. Akai, T. Tsujino, N. Fukuda, K. Iio, Y. Takeda, K. Kawaguchi, T. Naka,

K. Higuchi, E. Akiyama, H. Fujioka, Y. Kita Chemistry-A European Journal 11(21), 6286-6297 (2005)

9. M. Pizzonero, F. Dumas, J. d'Angelo Heterocycles 66, 31-37 (2005) 10. J.T. Su, J. Xiong, S. C. Liang, G. F. Qiu, X. C. Feng, H. B. Teng, L. M. Wu,

X. M. Hu Synth. Commun. 36 (6), 693-699 (2006) 11. W. C. Chan, A. Higton, J. S. Davies Amino Acids, Peptides, and Proteins 35,

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12. P. D. de Maria, C. A. Garcia-Burgos, G. Bargeman, R. W. van Gemert Synthesis-Stutgart 10, 1439-1452 (2007)

13. F. Brackmann, A. de Meijere : Chem. Rev., 107, 4493-4537 (2007) 14. Q. F. Zhu, Z.X. Xu, Y. B. Hao, Y. L. Xiao, W. J. Xu, X. B. Ke, H. B. Teng,

L. M. Wu, G. F. Qiu, S. C. Liang, X. M. Hu: Lett. Org. Chem. 5(6), 478-483 (2008)

15. C. Cativiela, M. Ordóñez: Tetrahedron: Asymmetry 20, 1–63 (2009) 16. Y. A. Volkova, O. A. Ivanova, E. M. Budynina, E. V. Revunov, E. B.

Averina: Tetrahedron Lett. 50, 2793-2796 (2009)

3. P. Tähtinen, J. Sinkkonen, K.D. Klika, V. Nieminen, G. Stájer, Z. Szakonyi, F. Fülöp,

K. Pihlaja 1H, 13C, and 15N NMR stereochemical study of cis-fused 7a(8a)-methyl and 6-phenyl octa(hexa)hydrocyclopenta[d][1,3]oxazines and [3,1]benzoxazines Chirality, 13, 1-12 (2002) I.f.: 1,976

1. G. Puigbo, F. Diaba, J. Bonjoch: Tetrahedron 59(15), 2657-2665 (2003 ) 2. R. H. Contreras, V. Barone, J. C. Facelli, J. E. Peralta: Annual Reports on

NMR Spectroscopy 51, 167-260 (2003) 3. E. Kolehmainen: Annual Reports on NMR Spectroscopy 49, 167-260 (2003) 4. W.-D. Rudorf: Journal of Sulfur Chemistry 28 (3), 295-339 (2007) 5. L. B. Krivdin, R. Contreras: Annual Reports on NMR Spectroscopy 61, 133-

245 (2007) 6. R. Marek, A. Lycka, E. Kolehmainen, E. Sievanen, J. Tousek: Curr. Org.

Chem. 11(13), 1154-1205 (2007) 4. S. Gyónfalvi, Z. Szakonyi, F. Fülöp

Synthesis and transformation of novel cyclic β-amino acid derivatives from (+)-3-carene Tetrahedron: Asymmetry, 14, 3965-3972 (2003) I.f.: 2,386

1. M. I. Aguilar, G. D. Fallon, P. A. Mayes, S. Nordin, A. J. Robinson, M. L. Rose, F. Vounatsos, B. Wilman, P. Perlmutter: Letters in Peptide Science 10(5-6), 597-604 (2003)


3. F. Z. Macaev, A. V. Malkov Tetrahedron 62 9-29 (2006) 4. M. Frackowiak, K. Ochalik, A. Bialonska, Z. Ciunik, C. Wawrzenczyk, S.

Lochynski Tetrahedron: Asymmetry, 17 124-129 (2006) 5. M. Sathe, R. Ghorpade, M. P. Kaushik: Chemistry Letters 35(9), 1004-

1005 (2006) 6. X.-G. Li, M. Lähitie, M. Päiviö, L.T. Kanerva: Tetrahedron: Asymmetry

18, 1567–1573 (2007) 7. B. Alcaide, P. Almendros, C. Aragoncillo: Chem. Rev., 107, 4437-4592

(2007) 8. A. Mondière, R. Peng, R. Remuson, D.J. Aitken: Tetrahedron 64, 1088-

1093 (2008) 9. M. D’hooghe, Y. Dejaegher, N. De Kimpe: Tetrahedron 64, 4575–

4584 (2008) 10. M. Sathe, H. N. Karade, M. P. Kaushik: Synth. Commun. 38(9), 1375-1380

(2008)

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13. L. Zhou, H.F. Jiang, C.J. Li : Adv. Synth. Catal. 350, 2226-2230 (2008) 14. E. A. Koneva, T. M. Khomenko, S. Yu. Kurbakova, N. I. Komarova, D. V.

Korchagina, K. P. Volcho, N. F. Salakhutdinov, A. G. Tolstikov, G. A. Tolstikov: Russ. Chem. Bull., Int. Ed., 57, 1680-1685 (2008)

15. E. Forró: J. Chrom. A. 1216(6), 1025-1029 (2009) 16. K. Gajcy, T. Librowski, S. Lochynski: Lett. Org. Chem. 6(3), 186-188

(2009) 17. E. A. Koneva, K. P. Volcho, D. V. Korchagina, N. F. Salakhutdinov, A. G.

Tolstikov: Russ. J. Org. Chem. 45, 815-824 (2009) 5. G. Tóth, Z. Szakonyi, B. Kanyó, F. Fülöp, G. Jancsó, L. Pávics: Preparation of

[99mTc]TRODAT-1 involving a simple purification method J. Labelled Compd. Rad., 46, 1067-1073 (2003) I.f.: 1,207

1. Z. P. Chen, S. P. Wang, J. Tang, X. M. Li, C. Y. Liu, X. J. Xu, G. X. Cao: Journal of Radioanalytical and Nuclear Chemistry 3, 591-594 (2008), DOI: 10.1007/s10967-007-7109-z

6. Kanyó B. Árgyelán M., Dibó Gy., Szakonyi Zs., Vécsei L., Fülöp F., Láncz A.,

Forgács P., Pávics L: Dopamintranszporter-vizsgálatok egyfotonemissziós komputertomográfiával (SPECT) mozgászavarokkal járó kórképekben Clin. Neurosci./Ideggy. Szle. 56(7-8), 231-240 (2003)

1. C.S. Ming, E. Amaro Jr., H. B. Ferraz, M. Q. Hoexter, F. O. Goulart, J.

Wagner, F. L. Li, K. F. Ying, J. J. Mari, A. L. T. De Lacerda, S. Tufik, R.A. Bressan Arq. Neuro-Psiquiatr., 64 (3A) 628-634 (2006)

2. M. C. Shih, M. Q. Hoexter, L. A. F. de Andrade, R. A. Bressan Sao Paulo Med. J. 124(3) 168-175 (2006)

3. I.H. Li, W.S. Huang, C.B. Yeh, M.H. Liao, C.C. Chen, L.H. Shen, J.C. Liu, K.H. Ma: Nuclear Medicine and Biology 36, 605–611 (2009)

7. Z. Szakonyi, F. Fülöp, D. Tourwé, N. De Kimpe

Synthesis of 1,2,7,7a-tetrahydro-1aH-cyclopropa[b]quinoline-1a-carboxylic acid derivatives, doubly constrained ACC derivatives, by a remarkable cyclopropanation process. J. Org. Chem., 67, 2192-2196 (2002) I.f.: 3,462

1. M. Meusel, M. Guetschow Org. Prep. Proced. Int. 36(5) 391-443 (2004) 2. S. P. Bew: Comprehensive Organic Functional Group Transformations II 5,

19-125 (2005) 3. B. Bonnaud, P. Funes, N. Jubault, B. Vacher : Eur. J. Org. Chem. 15, 3360-

3369 (2005) 4. F. Brackmann, A. de Meijere : Chem. Rev., 107, 4493-4537 (2007) 5. W. Wan, Y. Gao, H. Jiang, J. Hao: J. Fluorine. Chem. 129, 510-514 (2008)

8. E.R. Alonso, K.A. Tehrani, M. Boelens, A.V. Tkachev, Z. Szakonyi, F. Fülöp, N. De

Kimpe

Novel synthesis of functionalized 2-pyrrolidinones via unsaturated imidoyl cyanides Organic Preparations and Procedures International, 35, 215-219 (2003)

I.f.: 0,791

9. A. Hetényi, Z. Szakonyi, K. D. Klika, K. Pihlaja, and F. Fülöp Formation and characterization of a nine-component equilibrium system derived from cis- and trans-1-aminomethylcyclohexane-1,2-diol J. Org. Chem., 68, 2175-2182 (2003) I.f.: 3,462

1. H. S. El Khadem, A. J. Fatiadi Carbohydrate Chemistry and Biochemistry 59, 135-173 (2004)

2. S. Pérez, C. López, A. Caubet, A. Roig, E. Molins, J. Org. Chem. 70 (12), 4857-4860 (2005)

3. E. Frank, B. Kazi,, Z. Mucsi, K. Ludányi, G. Keglevich: Steroids 72 (5), 446-458 (2007)

10. M. D'hooghe, Z. Szakonyi, F. Fülöp, N. De Kimpe

Synthesis of N-(4-chlorobutyl)butanamide, a chlorinated amide isolated from Aloe sabaea Organic Preparations and Procedures International, 35, 501-507 (2003)

I.f.: 0,791

11. Z. Szakonyi, F. Fülöp Mild and efficient ring opening of monoterpene-fused β-lactam enantiomers. Synthesis of novel β-amino acid derivatives ARKIVOC, (xiv), 225-232 (2003) I.f.: 0,418

1. L. Liu, L.L. Zhang, G. Liu, J. X. Xu: ARKIVOC (xvi) 318-326 (2008)

12. Lázár L., Szakonyi Zs., Forró E., Palkó M., Zalán Z., Szatmári I., Fülöp F. Gyulladásgátló hatású hidrazinoalkoholok szintézise Acta Pharm. Hung., 74, 11-18 (2004)

13. F. Fülöp, L. Lázár, Z. Szakonyi, M. Pihlavisto, S. Alaranta, P. J. Vainio, A. Juhakoski, A. Marjamäki, D. J. Smith Discovery of new anti-inflammatory agents Pure Appl. Chem., 76 (5), 965–972 (2004). I.f.: 1,449

1. P. Knowles, C. Kurtis, J. Murray, C. Saysell, W. Tambyrajah, C. Wilmot, M. McPherson, S. Phillips, D. Dooley, D. Brown, M. Rogers, M. Mure: J. Neural Transmission 114(6), 743-746 (2007)

2. B. M. Strolin, K.F. Tipton, R. Whomsley: Fundamental and Clinical Pharmacology 21(5), 467–479 (2007)

3. P. Dunkel, A. Gelain, D. Barlocco, N. Haider, K. Gyires, B. Sperlágh, K. Magyar, E. Maccioni, A. Fadda, P. Mátyus, Curr. Med. Chem. 15, 1827-1839 (2008)

14. Z. Szakonyi, M. D’hooghe, I. Kanizsai, F. Fülöp, N. De Kimpe

Synthesis of bicyclic carbamates as precursors of Sedum alkaloid derivatives Tetrahedron 61, 1595-1602 (2005) I.f.: 2,643

1. J. D. Adams, C. Garcia Evidence-based complementary and alternative medicine 3 (1), 125-131 (2006)

2. Comprehensive Heterocyclic Chemistry III., Ed.: A. R. Katritzky, C. A. Ramsden, R. J. K. Taylor, E. F. V. Scriven, Elsevier Ltd. Oxford, 2008, Vol. 12.02, p97.

3. J. M. Carney, P. J. Donoghue, W. M. Wuest, O. Wiest, P. Helquist: Org. Lett. 10(17), 3903–3906 (2008)

15. Z. Szakonyi, S. Gyónfalvi, A. Hetényi, F. Forró, N. De Kimpe, F. Fülöp

Synthesis of 3- and 4-hydroxy-2-aminocyclohexanecarboxylic acids by iodocyclization Eur. J. Org. Chem. 4017–4023 (2005) I.f.: 2,426

1. G. W. Gribble, J. A. Joule, Progress in Heterocyclic Chemistry, Vol.

18, Eds.: Elsevier, 2007, p. 112. 2. B. Alcaide, P. Almendros, C. Aragoncillo: Chem. Rev., 107, 4437-4592

(2007) 3. M. Lloyd, R. Lloyd, P. Keene, A. Osborne, Journal of Chemical Technology

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(2008) 5. O. Songis, C. Didierjean, J. Martinez, M. Calmés: Tetrahedron: Asymmetry

19, 2135–2139 (2008) 6. Y. Matsushima, J. Kino: Eur. J. Org. Chem., 1619-1624 (2009)

16. Z. Szakonyi, Á. Balázs, T. A. Martinek,F. Fülöp

Enantioselective addition of diethylzinc to aldehydes catalyzed by γ-amino alcohols derived from (+)- and (-)-α-pinene Tetrahedron: Asymmetry, 17, 199-204 (2006) I.f.: 2,386

1. E. Busto, V. Gotor-Fernandez, V. Gotor: Tetrahedron: Asymmetry, 17, 1007-1016 (2006)

2. R.W. Parrott II, S. R. Hitchcock: Tetrahedron: Asymmetry, 18, 377-382 (2007)

3. A. G. Martínez, E. T.,Vilar, A. G. Fraile, S. de la Moya Cerero, P. Martínez Ruiz, C. Díaz Morillo: Tetrahedron: Asymmetry, 18, 742-749 (2007)

4. B. Alcaide, P. Almendros, C. Aragoncillo: Chem. Rev., 107, 4437-4592 (2007)

5. R.W. Parrott II, S.R. Hitchcock: Tetrahedron: Asymmetry, 19, 19-26 (2008)

6. D. Hobuß, A. Baro, S. Laschat, W. Frey: Tetrahedron, 64, 1635-1640 (2008)

7. I.V. Il'ina, K.P. Volcho, N.E. Salakhutdinov: Russian J. Org. Chem. 44(1), 1-23 (2008)

8. B. Alcaide, P. Almendros, Progress in Heterocyclic Chemistry, Vol. 19, Eds.: Elsevier, 2008, p. 92-111.

9. A.B. Terent’ev, T.T. Vasil’eva, O.V. Chahovskaya, N.E. Mysova, H.H. Hambardzumyan, K.A. Kochetkov: J. Fluorine. Chem. 129, 669-673 (2008)

10. M.I. Burguete, J. Escorihuela, S.V. Luis, A. Lledo´s, G. Ujaque: Tetrahedron, 64, 9717-9724 (2008)


12. J. Li, Y.M. Shang, C. Xiao, Z.G. Song, Y.Z. Li, H.M. Huang: Chem. Res. Chinese U. 25(1), 43–46 (2009)

13. D. Scarpi, E. G. Occhiato, A. Guarna: Tetrahedron: Asymmetry, 20, 340–350 (2009)

17. J. Magyar, B. Horváth, T. Bányász, N. Szentandrássy, P. Birinyi, A. Varró, Z.

Szakonyi, F. Fülöp, P. P. Nánási L-364,373 fails to activate the slow delayed rectifier K+ current in canine ventricular cardiomyocytes Naunyn-Schmiedeberg’s Arch. Pharmacol. 373, 85-90 (2006) I.f.: 1,963

18. I. Kanizsai,, Z. Szakonyi, R. Sillanpää, F. Fülöp

A comparative study of the multicomponent Ugi reactions of an oxabicycloheptene-based β-amino acid in water and in methanol Tetrahedron Lett. 47, 9113–9116 (2006) I.f.: 2,509

1. R. E. Dolle, B. Le Bourdonnec, A. J. Goodman, G. A. Morales, J. M. Salvino, W. Zhang, : J. Comb. Chem., 9(6), 855-902 (2007)

2. N. Shapiro, A. Vigalok: Angew. Chem. Int. Ed. 47(15), 2849-2852 (2008) 3. B. Alcaide, P. Almendros, Progress in Heterocyclic Chemistry, Vol.

19, Eds.: Elsevier, 2008, p. 92-111. 4. Comprehensive Heterocyclic Chemistry III., Ed.: A. R. Katritzky, C. A.


5. A. Brandi, S. Cicchi, F. M. Cordero: Chem. Rev., 108, 3988-4035 (2008) 6. C. C. A. Cariou, G. J. Clarkson, M. Shipman: J. Org. Chem. 73 (24), 9762-

9764 (2008) 7. C. Hulme, J. Dietrich: Mol. Divers. 13, 195–207 (2009)

19. I. Kanizsai, Z. Szakonyi, M. D’hooghe, F. Fülöp, N. De Kimpe

Synthesis of chiral 1,5-disubstituted pyrrolidinones via electrophile-induced cyclization of 2-(3-butenyl)oxazolines derived from (1R,2S)- and (1S,2R)-norephedrine Tetrahedron: Asymmetry, 17, 2857–2863 (2006) I.f.: 2,468 1. M. Hiroshi, O. Fumi, Y. Kenji: Heterocycles 74, 383-396 (2007)

20. I. Kanizsai, S. Gyónfalvi, Z. Szakonyi, R. Sillanpää, F. Fülöp

Synthesis of bi- and tricyclic β-lactam libraries in aqueous medium Green Chemistry, 9, 357-360 (2007) I.f.: 4,836

1. S. Capone, S. Pedatella, A. Guaragna, M. De Nisco, G. Palumbo: Tetrahedron, 63, 12202-12206 (2007)

2. O. Sereda, R. Wilhelm: Synlett, 3032-3036 (2007) 3. M. Krasavin, V. Parchinsky: Synlett, 645-648 (2008) 4. N. Liu, S. Cao, J. Wu, J. Yu, L. Shen, X. Feng, X. Qian: Tetrahedron, 64,

3966-3974 (2008)

5. G. Vasuki, K. Kumaravel: Tetrahedron Lett. 49, 5636-5638 (2008) 6. E. Forró: J. Chrom. A. 1216(6), 1025-1029 (2009)

21. Á. Balázs, Z. Szakonyi, F. Fülöp

Synthesis of alicyclic N-substituted 1,3-amino alcohols via 1,3-oxazines J. Heterocyclic Chem., 44, 403–406 (2007) I.f.: 0,735


Regio- and stereoselective synthesis of the enantiomers of monoterpene-based β-amino acid derivatives Tetrahedron: Asymmetry, 18, 2442–2447 (2007) I.f.: 2,634

1. M. Sathe, D. Thavaselvam, A. K. Srivastava, M. P. Kaushik: Molecules, 13, 432-443 (2008)

23. W. J. Peláez, Z. Szakonyi, F. Fülöp, G. I. Yranzo

Flash vacuum pyrolysis (FVP) of some hexahydroquinazolin-4(1H)-ones Tetrahedron 64, 1049-1057 (2008) I.f.: 2,897


Synthesis of enantiomeric spirooxazolines and spirooxazolidines by the regioselective ring closure of monoterpene-based aminodiols ARKIVOC part (iii) , 33-42 (2008) I.f.: 1,377

1. N. Hazeri, M. T. Maghsoodlou, S. M. Habibi-Khorassani, G. Marandi: ARKIVOC (xiv) 282-288 (2008)


Synthesis and application of monoterpene-based chiral aminodiols Tetrahedron 64, 1034-1039 (2008) I.f.: 2,897 1. D. Frain, F. Kirby, P. McArdle, P. O'Leary: Synlett 1261-1264 (2009)


Regio- and stereoselective synthesis of constrained enantiomeric β-amino acid derivatives Tetrahedron: Asymmetry, 19, 2296–2303 (2008) I.f.: 2,796

27. Anasztázia Hetényi, Zsolt Szakonyi, István M. Mándity, Éva Szolnoki, Gábor K.

Tóth, Tamás A. Martinek, Ferenc Fülöp Sculpting the β-peptide H12 helix via a designed side-chain shape Chem. Commun. 177–179 (2009) I.f.: 5,34

1. T. Beke, C. Somlai, G. Magyarfalvi, A. Perczel, G. Tarczay: J. Phys.

Chem. B, 113(22), 7918-7926 (2009) 28. Balázs, A. Hetényi, Z. Szakonyi, R. Sillanpää, F. Fülöp

Solvent Enhanced diastereo- and regioselectivity in the Pd(II)-catalyzed synthesis of six- and eight-membered heterocycles via cis-aminopalladation Chemistry - A European Journal, 15, 7376–7381 (2009) I.f.: 5,454

29. Z. Szakonyi, R. Sillanpää, F. Fülöp Synthesis of conformationally constrained tricyclic β-lactam enantiomers through Ugi four-centre three-component reactions of a monoterpene-based β-amino acid Mol. Div. kézirat elfogadva I.f.: 2,708

Össz I.f.: 67,04 II. Szabadalmak:

1. D. J. Smith, M. Jalkanen, F. Fülöp, L. Lázár, Z. Szakonyi, G. Bernáth: Inhibitors of copper-containing amine oxidases. (Biotie Therapies Corp., Finland). PCT Int. Appl. (2002),57 pp.; CAN 136:79760.



(2004), 269 pp., CAN 141:350160 3. S. S. Costa, M. De Souza, T. Ibrahim, G. Oliveira de Melo, A. P. De Almeida,

C. Guette, J.-P. Ferezou, V. L. G. Koatz J. Nat. Prod. 69(5), 815-818 (2006) 4. G. Negrón-Silva, C. X. Hernández-Reyes, D. Angeles-Beltrán, L. Lomas-

Romero, E. González-Zamora: Molecules, 13, 977-985 (2008) 5. P. Dunkel, A. Gelain, D. Barlocco, N. Haider, K. Gyires, B. Sperlágh, K.


2. D. J. Smith, J. David, M. Jalkanen, F. Fülöp, L. Lázár, Z. Szakonyi, G. Bernáth:

Oxadiazine derivatives as inhibitors of copper-containing amine oxidases. (Biotie Therapies Corp., Finland). PCT Int. Appl. (2002), 53 pp.; CA 136:102405.



(2004), 269 pp., CAN 141:350160 3. D. J. Smith, J. David; F. Fülöp, M. Pihlavisto, L. Lázár, S. Alaranta, P. Vainio, Z.

Szakonyi: Preparation of hydrazino indanes as inhibitors of copper-containing amine oxidases (Biotie Therapies Corporation, Finland). PCT Int. Appl. (2003), 58 pp.; CA 138:106506.

1. R. Ueno, A. Nagashima, T. Inoue, M. Ohkubo, K. Yoshihara: PCT Int. Appl.

(2004), 269 pp., CAN 141:350160 2. S. Jalkanen, SM. Salmi, M. Jalkanen: PCT Int. Appl. (2005), 31 pp., WO

2005072738, CAN 143:179666 3. S. Jalkanen, SM. Salmi, M. Jalkanen: PCT Int. Appl. (2005), 25 pp., WO

2005063261, CAN 143:109791 4. P. Dunkel, A. Gelain, D. Barlocco, N. Haider, K. Gyires, B. Sperlágh, K.


4. F. Fülöp, Z. Szakonyi: Chiral cyclic β-amino acids and their derivatives,

pharmaceutical compositions contaioning them and the use of such compounds

(Bioblocks Magyarország Gyógyszerkémiai és Fejlesztı Kft., Hungary) PCT Int. Appl., WO 2008/059299 A1, 36 pp.

Öszzes független idézettség az elmúlt 10 évben: 143 Szeged, 2009. augusztus 26.

tudományos munkásság: i. publikációk és független idézettségük · tudományos...

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